KR20240156409A - 주요 우울 장애 치료에 사용을 위한 아티카프란트의 다형 형태 - Google Patents

주요 우울 장애 치료에 사용을 위한 아티카프란트의 다형 형태 Download PDF

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Publication number
KR20240156409A
KR20240156409A KR1020247033176A KR20247033176A KR20240156409A KR 20240156409 A KR20240156409 A KR 20240156409A KR 1020247033176 A KR1020247033176 A KR 1020247033176A KR 20247033176 A KR20247033176 A KR 20247033176A KR 20240156409 A KR20240156409 A KR 20240156409A
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KR
South Korea
Prior art keywords
articaprant
crystalline form
amorphous
anhedonia
treatment
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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KR1020247033176A
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English (en)
Korean (ko)
Inventor
필리프 페르난데스
마크 쉬밋
바니나 포포바
아담 사비츠
라마 멜코트
웨인 씨. 드레베츠
스리하리 고팔
데럴 펨버톤
차크라다르 라기셰티
아이바 케직
Original Assignee
얀센 파마슈티칼즈, 인코포레이티드
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Application filed by 얀센 파마슈티칼즈, 인코포레이티드 filed Critical 얀센 파마슈티칼즈, 인코포레이티드
Publication of KR20240156409A publication Critical patent/KR20240156409A/ko
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020247033176A 2022-03-07 2023-03-06 주요 우울 장애 치료에 사용을 위한 아티카프란트의 다형 형태 Pending KR20240156409A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263317475P 2022-03-07 2022-03-07
US63/317,475 2022-03-07
PCT/IB2023/052088 WO2023170550A1 (en) 2022-03-07 2023-03-06 Polymorph forms of aticaprant for use in treating major depressive disorder

Publications (1)

Publication Number Publication Date
KR20240156409A true KR20240156409A (ko) 2024-10-29

Family

ID=85706849

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020247033176A Pending KR20240156409A (ko) 2022-03-07 2023-03-06 주요 우울 장애 치료에 사용을 위한 아티카프란트의 다형 형태

Country Status (14)

Country Link
US (3) US11998524B2 (https=)
EP (1) EP4489747A1 (https=)
JP (1) JP2025508051A (https=)
KR (1) KR20240156409A (https=)
CN (1) CN119156211A (https=)
AU (1) AU2023232536A1 (https=)
CA (1) CA3254365A1 (https=)
CL (1) CL2024002627A1 (https=)
CO (1) CO2024012158A2 (https=)
IL (1) IL315409A (https=)
JO (1) JOP20240197A1 (https=)
MX (1) MX2024010980A (https=)
TW (1) TW202345796A (https=)
WO (1) WO2023170550A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12161622B2 (en) 2021-05-04 2024-12-10 Janssen Pharmaceuticals, Inc. Compositions and methods for the treatment of depression
WO2023170554A1 (en) 2022-03-07 2023-09-14 Janssen Pharmaceuticals, Inc. Compositions comprising aticaprant

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AU2023232536A1 (en) 2024-10-24
US20230277499A1 (en) 2023-09-07
US11998524B2 (en) 2024-06-04
IL315409A (en) 2024-11-01
CL2024002627A1 (es) 2025-01-24
CN119156211A (zh) 2024-12-17
JOP20240197A1 (ar) 2024-09-05
US12171743B2 (en) 2024-12-24
WO2023170550A1 (en) 2023-09-14
CO2024012158A2 (es) 2024-09-30
JP2025508051A (ja) 2025-03-21
CA3254365A1 (en) 2023-09-14
EP4489747A1 (en) 2025-01-15
US20240316003A1 (en) 2024-09-26
US20250325515A1 (en) 2025-10-23
MX2024010980A (es) 2024-12-06
TW202345796A (zh) 2023-12-01

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