KR20210034039A - 다파글리플로진을 사용하는 HFpEF의 치료 방법 및 이를 포함하는 조성물 - Google Patents

다파글리플로진을 사용하는 HFpEF의 치료 방법 및 이를 포함하는 조성물 Download PDF

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KR20210034039A
KR20210034039A KR1020217004721A KR20217004721A KR20210034039A KR 20210034039 A KR20210034039 A KR 20210034039A KR 1020217004721 A KR1020217004721 A KR 1020217004721A KR 20217004721 A KR20217004721 A KR 20217004721A KR 20210034039 A KR20210034039 A KR 20210034039A
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day
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patient
treatment
diabetic patient
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안나 마리아 랭킬드
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아스트라제네카 아베
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020217004721A 2018-07-19 2019-07-18 다파글리플로진을 사용하는 HFpEF의 치료 방법 및 이를 포함하는 조성물 Ceased KR20210034039A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862700463P 2018-07-19 2018-07-19
US62/700,463 2018-07-19
PCT/EP2019/069323 WO2020016335A1 (en) 2018-07-19 2019-07-18 Methods of treating hfpef employing dapagliflozin and compositions comprising the same

Publications (1)

Publication Number Publication Date
KR20210034039A true KR20210034039A (ko) 2021-03-29

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KR1020217004721A Ceased KR20210034039A (ko) 2018-07-19 2019-07-18 다파글리플로진을 사용하는 HFpEF의 치료 방법 및 이를 포함하는 조성물

Country Status (21)

Country Link
US (2) US11826376B2 (https=)
EP (1) EP3823631A1 (https=)
JP (2) JP2021530517A (https=)
KR (1) KR20210034039A (https=)
CN (1) CN112512530A (https=)
AU (4) AU2019304032B2 (https=)
BR (1) BR112021000139A2 (https=)
CA (1) CA3105626A1 (https=)
CL (1) CL2021000107A1 (https=)
CR (1) CR20210029A (https=)
EA (1) EA202190226A1 (https=)
IL (2) IL319642A (https=)
JO (1) JOP20210009A1 (https=)
MA (1) MA53175A (https=)
MX (2) MX2021000601A (https=)
MY (1) MY210508A (https=)
PE (1) PE20210644A1 (https=)
PH (1) PH12021550121A1 (https=)
SG (1) SG11202100417RA (https=)
UA (1) UA129183C2 (https=)
WO (1) WO2020016335A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112021000139A2 (pt) 2018-07-19 2021-04-06 Astrazeneca Ab Métodos de tratamento da hfpef empregando dapagliflozina e composições compreendendo a mesma
WO2021037400A1 (en) 2019-08-30 2021-03-04 Astrazeneca Ab Methods of treating heart failure with reduced ejection fraction with dapagliflozin
CN117510447B (zh) * 2023-11-08 2025-08-12 河北医科大学 一种达格列净-吡格列酮共无定形物及其制备方法和应用

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