KR20140034743A - 체외기생충 구제용 활성 화합물의 배합물 - Google Patents

체외기생충 구제용 활성 화합물의 배합물 Download PDF

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Publication number
KR20140034743A
KR20140034743A KR1020137018518A KR20137018518A KR20140034743A KR 20140034743 A KR20140034743 A KR 20140034743A KR 1020137018518 A KR1020137018518 A KR 1020137018518A KR 20137018518 A KR20137018518 A KR 20137018518A KR 20140034743 A KR20140034743 A KR 20140034743A
Authority
KR
South Korea
Prior art keywords
alkyl
spp
haloalkyl
alkoxy
halogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020137018518A
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English (en)
Korean (ko)
Inventor
안드레아스 투르베르크
울리히 괴르겐스
한스-게오르크 슈바르츠
슈테판 베르너
Original Assignee
바이엘 인텔렉쳐 프로퍼티 게엠베하
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 바이엘 인텔렉쳐 프로퍼티 게엠베하 filed Critical 바이엘 인텔렉쳐 프로퍼티 게엠베하
Publication of KR20140034743A publication Critical patent/KR20140034743A/ko
Ceased legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020137018518A 2010-12-21 2011-12-19 체외기생충 구제용 활성 화합물의 배합물 Ceased KR20140034743A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102010063691A DE102010063691A1 (de) 2010-12-21 2010-12-21 Ektoparasitizide Wirkstoffkombinationen
DE102010063691.6 2010-12-21
PCT/EP2011/073280 WO2012084852A2 (de) 2010-12-21 2011-12-19 Ektoparasitizide wirkstoffkombinationen

Publications (1)

Publication Number Publication Date
KR20140034743A true KR20140034743A (ko) 2014-03-20

Family

ID=45476470

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020137018518A Ceased KR20140034743A (ko) 2010-12-21 2011-12-19 체외기생충 구제용 활성 화합물의 배합물

Country Status (26)

Country Link
US (1) US9066945B2 (enExample)
EP (1) EP2654425A2 (enExample)
JP (1) JP6018580B2 (enExample)
KR (1) KR20140034743A (enExample)
CN (1) CN103442569B (enExample)
AR (1) AR084509A1 (enExample)
AU (1) AU2011347551B2 (enExample)
BR (1) BR112013015952A2 (enExample)
CA (1) CA2822080A1 (enExample)
CL (1) CL2013001794A1 (enExample)
CO (1) CO6751235A2 (enExample)
CR (1) CR20130303A (enExample)
CU (1) CU20130081A7 (enExample)
DE (1) DE102010063691A1 (enExample)
DO (1) DOP2013000143A (enExample)
EC (1) ECSP13012706A (enExample)
GT (1) GT201300157A (enExample)
MX (1) MX2013006866A (enExample)
MY (1) MY164916A (enExample)
NI (1) NI201300056A (enExample)
NZ (1) NZ612221A (enExample)
PH (1) PH12013501317A1 (enExample)
RU (1) RU2013133704A (enExample)
TW (1) TWI593685B (enExample)
UY (1) UY33822A (enExample)
WO (1) WO2012084852A2 (enExample)

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CN110305115A (zh) * 2019-08-19 2019-10-08 南通大学 一种含1-(6-氯吡嗪-2-基)-3-甲氧基吡唑单元的吡唑肟衍生物的制备和应用
US12655138B2 (en) 2020-07-24 2026-06-16 Elanco Us Inc. Process for making an isoxazoline compound and intermediate thereof
AU2021335500A1 (en) 2020-09-04 2023-05-04 Elanco Us Inc. Palatable formulations
WO2024121262A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121261A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121264A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121263A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives

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Also Published As

Publication number Publication date
US20140179623A1 (en) 2014-06-26
WO2012084852A2 (de) 2012-06-28
CN103442569B (zh) 2017-04-05
MX2013006866A (es) 2013-07-29
AU2011347551A1 (en) 2013-07-11
CR20130303A (es) 2013-07-18
MY164916A (en) 2018-02-15
BR112013015952A2 (pt) 2018-07-10
PH12013501317A1 (en) 2019-09-02
US9066945B2 (en) 2015-06-30
TW201305141A (zh) 2013-02-01
JP6018580B2 (ja) 2016-11-02
DOP2013000143A (es) 2013-08-15
DE102010063691A1 (de) 2012-06-21
AU2011347551B2 (en) 2016-03-17
RU2013133704A (ru) 2015-01-27
WO2012084852A3 (de) 2012-11-15
TWI593685B (zh) 2017-08-01
CU20130081A7 (es) 2013-09-27
CO6751235A2 (es) 2013-09-16
AR084509A1 (es) 2013-05-22
NZ612221A (en) 2016-01-29
CN103442569A (zh) 2013-12-11
GT201300157A (es) 2014-09-02
EP2654425A2 (de) 2013-10-30
UY33822A (es) 2012-07-31
CA2822080A1 (en) 2012-06-28
CL2013001794A1 (es) 2014-04-04
ECSP13012706A (es) 2013-08-30
NI201300056A (es) 2014-06-06
JP2014505677A (ja) 2014-03-06

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