TWI593685B - 殺外寄生蟲之活性化合物組合物 - Google Patents

殺外寄生蟲之活性化合物組合物 Download PDF

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Publication number
TWI593685B
TWI593685B TW100147255A TW100147255A TWI593685B TW I593685 B TWI593685 B TW I593685B TW 100147255 A TW100147255 A TW 100147255A TW 100147255 A TW100147255 A TW 100147255A TW I593685 B TWI593685 B TW I593685B
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Taiwan
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TW100147255A
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English (en)
Chinese (zh)
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TW201305141A (zh
Inventor
安德烈斯 特伯格
尤瑞奇 葛根斯
漢斯喬格 舒瓦茲
史蒂芬 華納
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拜耳智慧財產有限公司
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Publication of TW201305141A publication Critical patent/TW201305141A/zh
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/601,4-Diazines; Hydrogenated 1,4-diazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
TW100147255A 2010-12-21 2011-12-20 殺外寄生蟲之活性化合物組合物 TWI593685B (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102010063691A DE102010063691A1 (de) 2010-12-21 2010-12-21 Ektoparasitizide Wirkstoffkombinationen

Publications (2)

Publication Number Publication Date
TW201305141A TW201305141A (zh) 2013-02-01
TWI593685B true TWI593685B (zh) 2017-08-01

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
TW100147255A TWI593685B (zh) 2010-12-21 2011-12-20 殺外寄生蟲之活性化合物組合物

Country Status (26)

Country Link
US (1) US9066945B2 (enExample)
EP (1) EP2654425A2 (enExample)
JP (1) JP6018580B2 (enExample)
KR (1) KR20140034743A (enExample)
CN (1) CN103442569B (enExample)
AR (1) AR084509A1 (enExample)
AU (1) AU2011347551B2 (enExample)
BR (1) BR112013015952A2 (enExample)
CA (1) CA2822080A1 (enExample)
CL (1) CL2013001794A1 (enExample)
CO (1) CO6751235A2 (enExample)
CR (1) CR20130303A (enExample)
CU (1) CU20130081A7 (enExample)
DE (1) DE102010063691A1 (enExample)
DO (1) DOP2013000143A (enExample)
EC (1) ECSP13012706A (enExample)
GT (1) GT201300157A (enExample)
MX (1) MX2013006866A (enExample)
MY (1) MY164916A (enExample)
NI (1) NI201300056A (enExample)
NZ (1) NZ612221A (enExample)
PH (1) PH12013501317A1 (enExample)
RU (1) RU2013133704A (enExample)
TW (1) TWI593685B (enExample)
UY (1) UY33822A (enExample)
WO (1) WO2012084852A2 (enExample)

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RU2641916C2 (ru) * 2012-10-02 2018-01-23 Байер Кропсайенс Аг Гетероциклические соединения в качестве пестицидов
CN111246743B (zh) * 2017-10-18 2022-10-11 拜耳公司 具有杀虫/杀螨性质的活性化合物结合物
CN110305115A (zh) * 2019-08-19 2019-10-08 南通大学 一种含1-(6-氯吡嗪-2-基)-3-甲氧基吡唑单元的吡唑肟衍生物的制备和应用
KR20230043904A (ko) 2020-07-24 2023-03-31 엘랑코 유에스 인코포레이티드 이속사졸린 화합물 및 이의 중간체의 제조 공정
EP4208157A1 (en) 2020-09-04 2023-07-12 Elanco Us Inc. Palatable formulations
WO2024121263A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121261A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121262A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121264A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives

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Also Published As

Publication number Publication date
DOP2013000143A (es) 2013-08-15
CU20130081A7 (es) 2013-09-27
US20140179623A1 (en) 2014-06-26
MX2013006866A (es) 2013-07-29
AU2011347551B2 (en) 2016-03-17
US9066945B2 (en) 2015-06-30
TW201305141A (zh) 2013-02-01
JP2014505677A (ja) 2014-03-06
NZ612221A (en) 2016-01-29
DE102010063691A1 (de) 2012-06-21
UY33822A (es) 2012-07-31
GT201300157A (es) 2014-09-02
CN103442569B (zh) 2017-04-05
NI201300056A (es) 2014-06-06
CR20130303A (es) 2013-07-18
WO2012084852A2 (de) 2012-06-28
JP6018580B2 (ja) 2016-11-02
CA2822080A1 (en) 2012-06-28
BR112013015952A2 (pt) 2018-07-10
RU2013133704A (ru) 2015-01-27
CN103442569A (zh) 2013-12-11
CL2013001794A1 (es) 2014-04-04
CO6751235A2 (es) 2013-09-16
AU2011347551A1 (en) 2013-07-11
ECSP13012706A (es) 2013-08-30
AR084509A1 (es) 2013-05-22
EP2654425A2 (de) 2013-10-30
KR20140034743A (ko) 2014-03-20
WO2012084852A3 (de) 2012-11-15
MY164916A (en) 2018-02-15
PH12013501317A1 (en) 2019-09-02

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