KR20120107991A - Ｃ형 간염 바이러스 억제제 - Google Patents

Ｃ형 간염 바이러스 억제제 Download PDF

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Publication number
KR20120107991A
KR20120107991A KR1020127018317A KR20127018317A KR20120107991A KR 20120107991 A KR20120107991 A KR 20120107991A KR 1020127018317 A KR1020127018317 A KR 1020127018317A KR 20127018317 A KR20127018317 A KR 20127018317A KR 20120107991 A KR20120107991 A KR 20120107991A
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KR
South Korea
Prior art keywords
cap
mmol
mixture
hcv
added
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KR1020127018317A
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English (en)
Korean (ko)
Inventor
마코넨 벨레마
제프리 리 로마인
반 엔. 응우옌
간 왕
오마르 디. 로페즈
데니스 알. 생 로랑
퀴 첸
존 에이. 벤더
종 양
피야세나 헤와와삼
닝닝 수
니콜라스 에이. 민웰
존 에이. 이스터
바오-닝 수
미카엘 제이. 스미스
Original Assignee
브리스톨-마이어스 스큅 컴퍼니
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43479603&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20120107991(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 브리스톨-마이어스 스큅 컴퍼니 filed Critical 브리스톨-마이어스 스큅 컴퍼니
Publication of KR20120107991A publication Critical patent/KR20120107991A/ko
Withdrawn legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/19—Cytokines; Lymphokines; Interferons
    • A61K38/21—Interferons [IFN]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Zoology (AREA)
  • Molecular Biology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020127018317A 2009-12-16 2010-12-13 Ｃ형 간염 바이러스 억제제 Withdrawn KR20120107991A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US28694209P 2009-12-16 2009-12-16
US61/286,942 2009-12-16
US12/957,512 US8377980B2 (en) 2009-12-16 2010-12-01 Hepatitis C virus inhibitors
US12/957,512 2010-12-01

Publications (1)

Publication Number Publication Date
KR20120107991A true KR20120107991A (ko) 2012-10-04

Family

ID=43479603

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020127018317A Withdrawn KR20120107991A (ko) 2009-12-16 2010-12-13 Ｃ형 간염 바이러스 억제제

Country Status (21)

Country Link
US (1) US8377980B2 (enExample)
EP (1) EP2513091B1 (enExample)
JP (1) JP5785189B2 (enExample)
KR (1) KR20120107991A (enExample)
CN (1) CN102741242B (enExample)
AR (1) AR079634A1 (enExample)
AU (1) AU2010332034B2 (enExample)
BR (1) BR112012014677A2 (enExample)
CA (1) CA2784662A1 (enExample)
CL (1) CL2012001637A1 (enExample)
CO (1) CO6561788A2 (enExample)
EA (1) EA020815B1 (enExample)
MA (1) MA33806B1 (enExample)
MX (1) MX2012006635A (enExample)
NZ (1) NZ601220A (enExample)
PE (1) PE20121479A1 (enExample)
PH (1) PH12012500979A1 (enExample)
SG (1) SG181700A1 (enExample)
TN (1) TN2012000264A1 (enExample)
TW (1) TWI487702B (enExample)
WO (1) WO2011075439A1 (enExample)

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MA33806B1 (fr) 2012-12-03
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