KR20110033299A - 트리-사이클릭 피라졸로피리딘 키나제 억제제 - Google Patents
트리-사이클릭 피라졸로피리딘 키나제 억제제 Download PDFInfo
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- KR20110033299A KR20110033299A KR1020117004087A KR20117004087A KR20110033299A KR 20110033299 A KR20110033299 A KR 20110033299A KR 1020117004087 A KR1020117004087 A KR 1020117004087A KR 20117004087 A KR20117004087 A KR 20117004087A KR 20110033299 A KR20110033299 A KR 20110033299A
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
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- Oncology (AREA)
- Endocrinology (AREA)
- Transplantation (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8291908P | 2008-07-23 | 2008-07-23 | |
| US61/082,919 | 2008-07-23 | ||
| US11603208P | 2008-11-19 | 2008-11-19 | |
| US61/116,032 | 2008-11-19 | ||
| US14010008P | 2008-12-23 | 2008-12-23 | |
| US61/140,100 | 2008-12-23 | ||
| US16315209P | 2009-03-25 | 2009-03-25 | |
| US61/163,152 | 2009-03-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20110033299A true KR20110033299A (ko) | 2011-03-30 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020117004087A Withdrawn KR20110033299A (ko) | 2008-07-23 | 2009-07-22 | 트리-사이클릭 피라졸로피리딘 키나제 억제제 |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP2318408B1 (OSRAM) |
| JP (2) | JP2011529066A (OSRAM) |
| KR (1) | KR20110033299A (OSRAM) |
| CN (1) | CN102159574A (OSRAM) |
| AR (1) | AR074171A1 (OSRAM) |
| AU (1) | AU2009274027A1 (OSRAM) |
| BR (1) | BRPI0916295A2 (OSRAM) |
| CA (1) | CA2731432A1 (OSRAM) |
| IL (1) | IL210822A0 (OSRAM) |
| MX (1) | MX2011000843A (OSRAM) |
| TW (1) | TW201018680A (OSRAM) |
| WO (1) | WO2010011772A2 (OSRAM) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3140759B2 (ja) | 1990-04-02 | 2001-03-05 | キンセキ株式会社 | 弾性表面波素子の製造方法 |
| JP3362860B2 (ja) | 1991-01-09 | 2003-01-07 | 大日本印刷株式会社 | 表面弾性波素子の製造方法 |
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| US8846712B2 (en) | 2011-09-12 | 2014-09-30 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| EP2567959B1 (en) * | 2011-09-12 | 2014-04-16 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| WO2013045413A1 (en) * | 2011-09-27 | 2013-04-04 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| WO2013060636A1 (en) * | 2011-10-25 | 2013-05-02 | Sanofi | 6-(4-hydroxy-phenyl)-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| WO2013167403A1 (en) * | 2012-05-09 | 2013-11-14 | Sanofi | Substituted 6-(4-hydroxy-phenyl)-1h-pyrazolo[3,4-b]pyridine derivatives as kinase inhibitors |
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| JP6878316B2 (ja) * | 2015-06-19 | 2021-05-26 | ノバルティス アーゲー | Ｓｈｐ２の活性を阻害するための化合物および組成物 |
| JP6828271B2 (ja) | 2016-05-18 | 2021-02-10 | ソニー株式会社 | 通信装置、通信方法、プログラム、および、通信システム |
| KR102642378B1 (ko) * | 2017-03-24 | 2024-02-28 | 픽사이 인코포레이티드 | 유용한 약학적 적용을 갖는 융합된 트리아졸로-피리미딘 화합물 |
| CN111032045B (zh) * | 2017-08-15 | 2023-08-15 | 安吉奥斯医药品有限公司 | 用于治疗血液病症的丙酮酸激酶激活剂 |
| CN111620866A (zh) * | 2019-02-27 | 2020-09-04 | 南京药石科技股份有限公司 | 一种顺式-7,7-二氟-六氢-1H 吡咯并[3,4-c]吡啶衍生物及其制备方法 |
| KR20240157788A (ko) * | 2022-02-08 | 2024-11-01 | 테라스, 인크. | 암 및 기타 적응증의 치료에 사용하기 위한 적어도 4개의 환에 의해서 형성된 t 구조를 갖는 화합물 |
| CN118834206A (zh) * | 2023-04-24 | 2024-10-25 | 北京宇繁科技有限责任公司 | 一种map4k4抑制剂及其制备方法和应用 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10222550A1 (de) * | 2002-05-17 | 2003-11-27 | Bayer Ag | Substituierte Benzyl-pyrazolopyridine |
| MXPA05001688A (es) * | 2002-08-12 | 2005-04-19 | Sugen Inc | 3-pirrolil-piridopirazoles y 3-pirrolil-indazoles como inhibidores de cinasa novedosos. |
| US7507826B2 (en) * | 2004-03-30 | 2009-03-24 | Vertex Pharmaceuticals Incorporated | Azaindoles useful as inhibitors of JAK and other protein kinases |
| WO2005103050A2 (en) * | 2004-04-02 | 2005-11-03 | Vertex Pharmaceuticals Incorporated | Azaindoles useful as inhibitors of rock and other protein kinases |
| BRPI0610828A2 (pt) * | 2005-05-16 | 2010-07-27 | Irm Llc | compostos e composições como inibidores de proteìna quinase |
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- 2009-07-22 BR BRPI0916295A patent/BRPI0916295A2/pt not_active IP Right Cessation
- 2009-07-22 KR KR1020117004087A patent/KR20110033299A/ko not_active Withdrawn
- 2009-07-22 JP JP2011520175A patent/JP2011529066A/ja not_active Withdrawn
- 2009-07-22 AU AU2009274027A patent/AU2009274027A1/en not_active Abandoned
- 2009-07-22 CN CN2009801367212A patent/CN102159574A/zh active Pending
- 2009-07-22 MX MX2011000843A patent/MX2011000843A/es not_active Application Discontinuation
- 2009-07-22 CA CA2731432A patent/CA2731432A1/en not_active Abandoned
- 2009-07-22 WO PCT/US2009/051437 patent/WO2010011772A2/en not_active Ceased
- 2009-07-23 TW TW098124909A patent/TW201018680A/zh unknown
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| WO2010011772A3 (en) | 2010-04-29 |
| EP2318408B1 (en) | 2016-02-17 |
| BRPI0916295A2 (pt) | 2019-09-24 |
| AR074171A1 (es) | 2010-12-29 |
| JP2014208710A (ja) | 2014-11-06 |
| JP5931976B2 (ja) | 2016-06-08 |
| CA2731432A1 (en) | 2010-01-28 |
| WO2010011772A2 (en) | 2010-01-28 |
| AU2009274027A1 (en) | 2010-01-28 |
| EP2318408A2 (en) | 2011-05-11 |
| JP2011529066A (ja) | 2011-12-01 |
| TW201018680A (en) | 2010-05-16 |
| CN102159574A (zh) | 2011-08-17 |
| IL210822A0 (en) | 2011-04-28 |
| MX2011000843A (es) | 2011-04-11 |
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