KR20110031349A - 티아졸릴 피페리딘 유도체 - Google Patents
티아졸릴 피페리딘 유도체 Download PDFInfo
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- KR20110031349A KR20110031349A KR1020117001604A KR20117001604A KR20110031349A KR 20110031349 A KR20110031349 A KR 20110031349A KR 1020117001604 A KR1020117001604 A KR 1020117001604A KR 20117001604 A KR20117001604 A KR 20117001604A KR 20110031349 A KR20110031349 A KR 20110031349A
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Classifications
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- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/28—Radicals substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
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- Ophthalmology & Optometry (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Neurosurgery (AREA)
- Endocrinology (AREA)
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- Biomedical Technology (AREA)
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- Obesity (AREA)
- Oncology (AREA)
- Gastroenterology & Hepatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102008029734A DE102008029734A1 (de) | 2008-06-23 | 2008-06-23 | Thiazolyl-piperidinderivate |
| DE102008029734.8 | 2008-06-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20110031349A true KR20110031349A (ko) | 2011-03-25 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020117001604A Withdrawn KR20110031349A (ko) | 2008-06-23 | 2009-05-28 | 티아졸릴 피페리딘 유도체 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US8436186B2 (https=) |
| EP (1) | EP2313403B1 (https=) |
| JP (1) | JP5607038B2 (https=) |
| KR (1) | KR20110031349A (https=) |
| CN (1) | CN102066367A (https=) |
| AR (1) | AR072192A1 (https=) |
| AU (1) | AU2009262631B2 (https=) |
| BR (1) | BRPI0913234A2 (https=) |
| CA (1) | CA2728851A1 (https=) |
| DE (1) | DE102008029734A1 (https=) |
| EA (1) | EA201100035A1 (https=) |
| IL (1) | IL210164A0 (https=) |
| MX (1) | MX2010013915A (https=) |
| WO (1) | WO2009156041A2 (https=) |
| ZA (1) | ZA201100566B (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
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| CN101679404B (zh) * | 2007-06-01 | 2012-06-13 | 霍夫曼-拉罗奇有限公司 | 哌啶-酰胺衍生物 |
| AU2010341229A1 (en) * | 2009-12-17 | 2012-08-02 | Merck Patent Gmbh | Sphingosine kinase inhibitors |
| US9845489B2 (en) | 2010-07-26 | 2017-12-19 | Biomatrica, Inc. | Compositions for stabilizing DNA, RNA and proteins in saliva and other biological samples during shipping and storage at ambient temperatures |
| GB201020161D0 (en) | 2010-11-26 | 2011-01-12 | Almac Discovery Ltd | Pharmaceutical compounds |
| GB2493142A (en) | 2011-07-20 | 2013-01-30 | Johann Wolfgang Goethe Uni T Frankfurt | Ceramide and ceramide synthase in the diagnosis and treatment of multiple sclerosis |
| JP6033791B2 (ja) * | 2011-12-23 | 2016-11-30 | Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 | 新規ｓ１ｐ受容体調整薬 |
| US9725703B2 (en) | 2012-12-20 | 2017-08-08 | Biomatrica, Inc. | Formulations and methods for stabilizing PCR reagents |
| WO2014157382A1 (ja) * | 2013-03-29 | 2014-10-02 | 味の素株式会社 | スフィンゴシンキナーゼ阻害剤 |
| CN106572650B (zh) | 2014-06-10 | 2021-08-31 | 生物马特里卡公司 | 在环境温度下稳定凝血细胞 |
| US9546151B2 (en) | 2014-07-31 | 2017-01-17 | Oregon Health & Science University | VMAT inhibitory compounds |
| EP3223807B1 (en) * | 2014-11-24 | 2021-09-15 | The Board of Trustees of the University of Illinois | Method of preventing or treating a pulmonary disease or condition |
| SG11201804776SA (en) | 2015-12-08 | 2018-07-30 | Biomatrica Inc | Reduction of erythrocyte sedimentation rate |
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| GB9624482D0 (en) | 1995-12-18 | 1997-01-15 | Zeneca Phaema S A | Chemical compounds |
| BR9707495A (pt) | 1996-02-13 | 1999-07-27 | Zeneca Ltd | Derivado de quinazolina processo para a preparação do mesmo composição farmacêutica e processo para a produç o de um efeito antiangiogênico e/ou de redução de permeabilidade vascular em um animal de sangue quente |
| US6291455B1 (en) | 1996-03-05 | 2001-09-18 | Zeneca Limited | 4-anilinoquinazoline derivatives |
| GB9718972D0 (en) | 1996-09-25 | 1997-11-12 | Zeneca Ltd | Chemical compounds |
| GB9714249D0 (en) | 1997-07-08 | 1997-09-10 | Angiogene Pharm Ltd | Vascular damaging agents |
| GB9900334D0 (en) | 1999-01-07 | 1999-02-24 | Angiogene Pharm Ltd | Tricylic vascular damaging agents |
| GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
| NZ522074A (en) | 2000-05-31 | 2004-06-25 | Astrazeneca Ab | Indole derivatives with vascular damaging activity |
| IL153484A0 (en) | 2000-07-07 | 2003-07-06 | Angiogene Pharm Ltd | Colchinol derivatives as angiogenesis inhibitors |
| CN1255392C (zh) | 2000-07-07 | 2006-05-10 | 安吉奥金尼药品有限公司 | 作为血管生成抑制剂的秋水仙醇衍生物 |
| KR101280096B1 (ko) | 2005-06-29 | 2013-06-28 | 컴퓨메딕스 리미티드 | 전도성 브리지를 포함하는 센서 어셈블리 |
| JP2009503107A (ja) | 2005-08-04 | 2009-01-29 | アポジー・バイオテクノロジー・コーポレイション | スフィンゴシンキナーゼ阻害剤およびそれらの使用方法 |
| MX2008002061A (es) | 2005-08-18 | 2008-04-16 | Hoffmann La Roche | Derivados de tiazolil piperidina utiles como moduladores del receptor h3. |
| EP1957076A2 (en) | 2005-11-29 | 2008-08-20 | Merck & Co., Inc. | Thiazole derivatives as cxcr3 receptor modulators |
-
2008
- 2008-06-23 DE DE102008029734A patent/DE102008029734A1/de not_active Withdrawn
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2009
- 2009-05-28 KR KR1020117001604A patent/KR20110031349A/ko not_active Withdrawn
- 2009-05-28 CA CA2728851A patent/CA2728851A1/en not_active Abandoned
- 2009-05-28 CN CN2009801234988A patent/CN102066367A/zh active Pending
- 2009-05-28 JP JP2011515144A patent/JP5607038B2/ja not_active Expired - Fee Related
- 2009-05-28 EA EA201100035A patent/EA201100035A1/ru unknown
- 2009-05-28 MX MX2010013915A patent/MX2010013915A/es not_active Application Discontinuation
- 2009-05-28 BR BRPI0913234A patent/BRPI0913234A2/pt not_active IP Right Cessation
- 2009-05-28 US US13/000,573 patent/US8436186B2/en not_active Expired - Fee Related
- 2009-05-28 AU AU2009262631A patent/AU2009262631B2/en not_active Ceased
- 2009-05-28 EP EP09768890.7A patent/EP2313403B1/de not_active Not-in-force
- 2009-05-28 WO PCT/EP2009/003817 patent/WO2009156041A2/de not_active Ceased
- 2009-06-19 AR ARP090102229A patent/AR072192A1/es unknown
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2010
- 2010-12-21 IL IL210164A patent/IL210164A0/en unknown
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2011
- 2011-01-21 ZA ZA2011/00566A patent/ZA201100566B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2011525502A (ja) | 2011-09-22 |
| EP2313403A2 (de) | 2011-04-27 |
| CN102066367A (zh) | 2011-05-18 |
| CA2728851A1 (en) | 2009-12-30 |
| ZA201100566B (en) | 2011-10-26 |
| AR072192A1 (es) | 2010-08-11 |
| BRPI0913234A2 (pt) | 2016-01-19 |
| IL210164A0 (en) | 2011-03-31 |
| JP5607038B2 (ja) | 2014-10-15 |
| AU2009262631A1 (en) | 2009-12-30 |
| AU2009262631B2 (en) | 2013-08-22 |
| WO2009156041A2 (de) | 2009-12-30 |
| EA201100035A1 (ru) | 2011-08-30 |
| DE102008029734A1 (de) | 2009-12-24 |
| US8436186B2 (en) | 2013-05-07 |
| US20110105505A1 (en) | 2011-05-05 |
| EP2313403B1 (de) | 2015-04-08 |
| MX2010013915A (es) | 2011-02-21 |
| WO2009156041A3 (de) | 2010-06-10 |
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