KR20110011653A - 테트라히드로이소퀴놀린의 제조 방법 - Google Patents

테트라히드로이소퀴놀린의 제조 방법 Download PDF

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KR20110011653A
KR20110011653A KR1020107027200A KR20107027200A KR20110011653A KR 20110011653 A KR20110011653 A KR 20110011653A KR 1020107027200 A KR1020107027200 A KR 1020107027200A KR 20107027200 A KR20107027200 A KR 20107027200A KR 20110011653 A KR20110011653 A KR 20110011653A
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compound
formula
solution
compounds
mmol
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Inventor
폴 로벤
루린 자오
베이 왕
방-치 천
슈앙 류
민 후
유-린 앨런 양
매튜 이셔우드
라시둘 아민
원거 추이
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브리스톨-마이어스 스큅 컴퍼니
알바니 몰레큘라 리써치, 인크.
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    • C07C217/58—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by singly-bound oxygen atoms with amino groups and the six-membered aromatic ring, or the condensed ring system containing that ring, bound to the same carbon atom of the carbon chain
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
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KR1020107027200A 2008-06-04 2009-06-04 테트라히드로이소퀴놀린의 제조 방법 Ceased KR20110011653A (ko)

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US5871708P 2008-06-04 2008-06-04
US61/058,717 2008-06-04

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KR20110011653A true KR20110011653A (ko) 2011-02-08

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US (4) US8420811B2 (cg-RX-API-DMAC10.html)
EP (2) EP2280955B8 (cg-RX-API-DMAC10.html)
JP (3) JP2011522827A (cg-RX-API-DMAC10.html)
KR (1) KR20110011653A (cg-RX-API-DMAC10.html)
CN (2) CN102112465B (cg-RX-API-DMAC10.html)
AR (1) AR071997A1 (cg-RX-API-DMAC10.html)
ES (1) ES2652462T3 (cg-RX-API-DMAC10.html)
TW (1) TW201002682A (cg-RX-API-DMAC10.html)
WO (2) WO2009149258A2 (cg-RX-API-DMAC10.html)

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CN102595902B (zh) * 2009-05-12 2015-04-29 阿尔巴尼分子研究公司 7-([1,2,4]三唑并[1,5-a]吡啶-6-基)-4-(3,4-二氯苯基)-1,2,3,4-四氢异喹啉及其用途
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JP5739415B2 (ja) * 2009-05-12 2015-06-24 ブリストル−マイヤーズ スクウィブ カンパニー （Ｓ）−７−（［１，２，４］トリアゾロ［１，５−ａ］ピリジン−６−イル）−４−（３，４−ジクロロフェニル）−１，２，３，４−テトラヒドロイソキノリンの結晶形態およびその使用
WO2012024397A2 (en) 2010-08-17 2012-02-23 Albany Molecular Research, Inc. 2,5-methano-and 2,5-ethano-tetrahydrobenzazepine derivatives and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
NO2686520T3 (cg-RX-API-DMAC10.html) 2011-06-06 2018-03-17
US10154988B2 (en) 2012-11-14 2018-12-18 The Johns Hopkins University Methods and compositions for treating schizophrenia
WO2014159501A2 (en) * 2013-03-14 2014-10-02 Bristol-Myers Squibb Company Processes for preparing tetrahydroisoquinolines
CN103601699A (zh) * 2013-11-04 2014-02-26 南京大学 一类1,3,4-噻二唑-2-酰胺衍生物及其制备方法
TWI665190B (zh) 2013-11-15 2019-07-11 阿克比治療有限公司 ｛［５－（３－氯苯基）－３－羥基吡啶－２－羰基］胺基｝乙酸之固體型式，其組合物及用途
US11713298B2 (en) 2018-05-09 2023-08-01 Akebia Therapeutics, Inc. Process for preparing 2-[[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino]acetic acid
US11524939B2 (en) 2019-11-13 2022-12-13 Akebia Therapeutics, Inc. Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino} acetic acid
US12612367B2 (en) 2019-12-10 2026-04-28 Akebia Therapeutics, Inc. Method for producing nitrogen-containing heteroarylcarboxamide acetic acid derivative
CN116351731B (zh) * 2023-03-10 2026-06-23 合肥博焱视芯电子科技有限公司 一种基于色选机的在线分拣方法及系统

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