KR20080081021A - 산제의 맛 차단 - Google Patents

산제의 맛 차단 Download PDF

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Publication number
KR20080081021A
KR20080081021A KR1020087016451A KR20087016451A KR20080081021A KR 20080081021 A KR20080081021 A KR 20080081021A KR 1020087016451 A KR1020087016451 A KR 1020087016451A KR 20087016451 A KR20087016451 A KR 20087016451A KR 20080081021 A KR20080081021 A KR 20080081021A
Authority
KR
South Korea
Prior art keywords
solid
fine powder
coated solid
coated
taste
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020087016451A
Other languages
English (en)
Korean (ko)
Inventor
라이너 벨링하우젠
다니엘 루드하르트
프랭크 라이더
마틴 스타인백
제스코 장크
마틴 와이스
올라프 베렌드
스팁하우트 우도 판
Original Assignee
바이엘 테크놀로지 서비시즈 게엠베하
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 바이엘 테크놀로지 서비시즈 게엠베하 filed Critical 바이엘 테크놀로지 서비시즈 게엠베하
Publication of KR20080081021A publication Critical patent/KR20080081021A/ko
Ceased legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/007—Pulmonary tract; Aromatherapy
    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5015—Organic compounds, e.g. fats, sugars
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5089—Processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Otolaryngology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Seasonings (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020087016451A 2005-12-24 2006-12-20 산제의 맛 차단 Ceased KR20080081021A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005062270.4 2005-12-24
DE102005062270A DE102005062270A1 (de) 2005-12-24 2005-12-24 Geschmacksmaskierung von Pulvern

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020117031078A Division KR101245627B1 (ko) 2005-12-24 2006-12-20 산제의 맛 차단

Publications (1)

Publication Number Publication Date
KR20080081021A true KR20080081021A (ko) 2008-09-05

Family

ID=38042692

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020087016451A Ceased KR20080081021A (ko) 2005-12-24 2006-12-20 산제의 맛 차단
KR1020117031078A Expired - Fee Related KR101245627B1 (ko) 2005-12-24 2006-12-20 산제의 맛 차단

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1020117031078A Expired - Fee Related KR101245627B1 (ko) 2005-12-24 2006-12-20 산제의 맛 차단

Country Status (24)

Country Link
US (1) US20090269411A1 (enExample)
EP (1) EP1968555A2 (enExample)
JP (2) JP5275039B2 (enExample)
KR (2) KR20080081021A (enExample)
CN (1) CN101346133A (enExample)
AU (1) AU2006331009B2 (enExample)
BR (1) BRPI0620618A2 (enExample)
CA (1) CA2634481A1 (enExample)
CR (1) CR10112A (enExample)
CU (1) CU23877B1 (enExample)
DE (1) DE102005062270A1 (enExample)
EC (1) ECSP088577A (enExample)
GT (1) GT200800126A (enExample)
HN (1) HN2008000964A (enExample)
IL (1) IL192085A0 (enExample)
MA (1) MA30072B1 (enExample)
MY (1) MY149601A (enExample)
NZ (1) NZ569279A (enExample)
RU (1) RU2440103C2 (enExample)
SV (1) SV2009002971A (enExample)
TN (1) TNSN08284A1 (enExample)
UA (1) UA93072C2 (enExample)
WO (1) WO2007073911A2 (enExample)
ZA (1) ZA200805498B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0327723D0 (en) 2003-09-15 2003-12-31 Vectura Ltd Pharmaceutical compositions
EP2050437A1 (en) * 2007-10-15 2009-04-22 Laboratoires SMB Improved pharmaceutical dry powder compositions for inhalation.
EP2252261A2 (en) * 2008-02-13 2010-11-24 Bayer Schering Pharma Aktiengesellschaft Drug delivery system with stabilising effect
US20110097405A1 (en) * 2008-02-13 2011-04-28 Bayer Schering Pharma Aktiengesellschaft Estradiol-containing drug delivery system
CA2745456A1 (en) * 2008-12-05 2010-06-10 Bayer Animal Health Gmbh Extrudate having spicular active substances
EP2411137B1 (en) 2009-03-27 2016-09-07 Bend Research, Inc. Spray-drying process
UY32836A (es) * 2009-08-12 2011-03-31 Bayer Schering Pharma Ag Partículas estabilizadas que comprenden 5-metil-(6s)-tetrahidrofolato
US20120207836A1 (en) 2009-08-19 2012-08-16 Bayer Pharma Aktiengesellschaft Drug delivery systems (wafer) for pediatric use
US8815294B2 (en) 2010-09-03 2014-08-26 Bend Research, Inc. Pharmaceutical compositions of dextran polymer derivatives and a carrier material
PT2611530T (pt) 2010-09-03 2019-05-09 Bend Res Inc Aparelho de secagem por pulverização e métodos de utilização do mesmo
WO2012031129A2 (en) 2010-09-03 2012-03-08 Bend Research, Inc. Spray-drying apparatus and methods of using the same
CN103619514B (zh) 2010-09-20 2016-09-28 Spi制药公司 微包囊方法和制品
WO2012040502A1 (en) 2010-09-24 2012-03-29 Bend Research, Inc. High-temperature spray drying process and apparatus
HU231017B1 (hu) 2012-05-08 2019-11-28 LAVET Gyógyszeripari Kft. Praziquantel tartalmú ízfedett formulációk
US8993041B2 (en) * 2012-10-15 2015-03-31 New Jersey Institute Of Technology Taste masked active pharmaceutical powder compositions and processes for making them
JP6650933B2 (ja) 2014-10-31 2020-02-19 ベンド リサーチ， インコーポレイテッド マトリックス中に分散された活性薬剤ドメインを形成するためのプロセス
CN114993892B (zh) * 2019-05-13 2024-10-18 南京制药厂有限公司 吡喹酮粒度的光散射检测法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4568559A (en) * 1984-02-06 1986-02-04 Biotek, Inc. Composite core coated microparticles and process of preparing same
NL193682C (nl) * 1987-05-14 2000-07-04 Glaxo Group Ltd Beklede cefuroximaxetilsamenstelling.
NZ507951A (en) * 1998-04-09 2002-12-20 Eurand Internat S Wettable microcapsules having hydrophobic polymer coated cores
FR2811913B1 (fr) * 2000-07-19 2003-09-19 Separex Sa Procede d'encapsulation sous forme de micro-capsules de fines particules solides
GB2405798A (en) * 2003-09-15 2005-03-16 Vectura Ltd Dry powder inhaler with primary and secondary piercing elements and a medicament pack for use with an inhalation device.

Also Published As

Publication number Publication date
TNSN08284A1 (en) 2009-10-30
AU2006331009A1 (en) 2007-07-05
UA93072C2 (ru) 2011-01-10
IL192085A0 (en) 2008-12-29
AU2006331009B2 (en) 2012-10-04
BRPI0620618A2 (pt) 2011-11-16
ZA200805498B (en) 2009-11-25
WO2007073911A3 (de) 2007-08-23
GT200800126A (es) 2010-06-25
SV2009002971A (es) 2009-04-28
CA2634481A1 (en) 2007-07-05
KR101245627B1 (ko) 2013-03-20
CR10112A (es) 2009-01-07
US20090269411A1 (en) 2009-10-29
DE102005062270A1 (de) 2007-06-28
CU20080124A7 (es) 2010-08-30
JP2013144695A (ja) 2013-07-25
RU2008130171A (ru) 2010-01-27
KR20120006085A (ko) 2012-01-17
JP5275039B2 (ja) 2013-08-28
MY149601A (en) 2013-09-13
MA30072B1 (fr) 2008-12-01
EP1968555A2 (de) 2008-09-17
NZ569279A (en) 2011-06-30
CN101346133A (zh) 2009-01-14
HN2008000964A (es) 2013-03-11
ECSP088577A (es) 2008-07-30
CU23877B1 (es) 2013-04-19
WO2007073911A2 (de) 2007-07-05
JP2009521419A (ja) 2009-06-04
RU2440103C2 (ru) 2012-01-20

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