BRPI0620618A2 - sólido revestido para o mascaramento do sabor de pós, processo para preparação e uso do mesmo - Google Patents
sólido revestido para o mascaramento do sabor de pós, processo para preparação e uso do mesmo Download PDFInfo
- Publication number
- BRPI0620618A2 BRPI0620618A2 BRPI0620618-2A BRPI0620618A BRPI0620618A2 BR PI0620618 A2 BRPI0620618 A2 BR PI0620618A2 BR PI0620618 A BRPI0620618 A BR PI0620618A BR PI0620618 A2 BRPI0620618 A2 BR PI0620618A2
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- Prior art keywords
- solid
- coated
- powder
- process according
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5015—Organic compounds, e.g. fats, sugars
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5089—Processes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Biophysics (AREA)
- Otolaryngology (AREA)
- Pulmonology (AREA)
- Molecular Biology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Preparation (AREA)
- Seasonings (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005062270.4 | 2005-12-24 | ||
| DE102005062270A DE102005062270A1 (de) | 2005-12-24 | 2005-12-24 | Geschmacksmaskierung von Pulvern |
| PCT/EP2006/012284 WO2007073911A2 (de) | 2005-12-24 | 2006-12-20 | Geschmacksmaskierung von pulvern |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0620618A2 true BRPI0620618A2 (pt) | 2011-11-16 |
Family
ID=38042692
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0620618-2A BRPI0620618A2 (pt) | 2005-12-24 | 2006-12-20 | sólido revestido para o mascaramento do sabor de pós, processo para preparação e uso do mesmo |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US20090269411A1 (enExample) |
| EP (1) | EP1968555A2 (enExample) |
| JP (2) | JP5275039B2 (enExample) |
| KR (2) | KR20080081021A (enExample) |
| CN (1) | CN101346133A (enExample) |
| AU (1) | AU2006331009B2 (enExample) |
| BR (1) | BRPI0620618A2 (enExample) |
| CA (1) | CA2634481A1 (enExample) |
| CR (1) | CR10112A (enExample) |
| CU (1) | CU23877B1 (enExample) |
| DE (1) | DE102005062270A1 (enExample) |
| EC (1) | ECSP088577A (enExample) |
| GT (1) | GT200800126A (enExample) |
| HN (1) | HN2008000964A (enExample) |
| IL (1) | IL192085A0 (enExample) |
| MA (1) | MA30072B1 (enExample) |
| MY (1) | MY149601A (enExample) |
| NZ (1) | NZ569279A (enExample) |
| RU (1) | RU2440103C2 (enExample) |
| SV (1) | SV2009002971A (enExample) |
| TN (1) | TNSN08284A1 (enExample) |
| UA (1) | UA93072C2 (enExample) |
| WO (1) | WO2007073911A2 (enExample) |
| ZA (1) | ZA200805498B (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0327723D0 (en) | 2003-09-15 | 2003-12-31 | Vectura Ltd | Pharmaceutical compositions |
| EP2050437A1 (en) * | 2007-10-15 | 2009-04-22 | Laboratoires SMB | Improved pharmaceutical dry powder compositions for inhalation. |
| CA2714598A1 (en) * | 2008-02-13 | 2009-08-20 | Bayer Schering Pharma Aktiengesellschaft | Drug delivery system with stabilising effect |
| US20110097405A1 (en) * | 2008-02-13 | 2011-04-28 | Bayer Schering Pharma Aktiengesellschaft | Estradiol-containing drug delivery system |
| NZ593217A (en) * | 2008-12-05 | 2013-05-31 | Bayer Ip Gmbh | Extrudate having spicular active substances |
| EP2411137B1 (en) | 2009-03-27 | 2016-09-07 | Bend Research, Inc. | Spray-drying process |
| UY32836A (es) | 2009-08-12 | 2011-03-31 | Bayer Schering Pharma Ag | Partículas estabilizadas que comprenden 5-metil-(6s)-tetrahidrofolato |
| EP2467126A1 (en) | 2009-08-19 | 2012-06-27 | Bayer Pharma Aktiengesellschaft | Drug delivery systems (wafer) for pediatric use |
| US9084944B2 (en) | 2010-09-03 | 2015-07-21 | Bend Research, Inc. | Spray-drying apparatus and methods of using the same |
| US8815294B2 (en) | 2010-09-03 | 2014-08-26 | Bend Research, Inc. | Pharmaceutical compositions of dextran polymer derivatives and a carrier material |
| PT2611529T (pt) | 2010-09-03 | 2019-05-09 | Bend Res Inc | Método de secagem por pulverização |
| KR101869114B1 (ko) | 2010-09-20 | 2018-06-19 | 다이앤 골 | 마이크로캡슐화 방법 및 제품 |
| WO2012040502A1 (en) | 2010-09-24 | 2012-03-29 | Bend Research, Inc. | High-temperature spray drying process and apparatus |
| HU231017B1 (hu) | 2012-05-08 | 2019-11-28 | LAVET Gyógyszeripari Kft. | Praziquantel tartalmú ízfedett formulációk |
| US8993041B2 (en) * | 2012-10-15 | 2015-03-31 | New Jersey Institute Of Technology | Taste masked active pharmaceutical powder compositions and processes for making them |
| US11364203B2 (en) | 2014-10-31 | 2022-06-21 | Bend Reserch, Inc. | Process for forming active domains dispersed in a matrix |
| CN114993892B (zh) * | 2019-05-13 | 2024-10-18 | 南京制药厂有限公司 | 吡喹酮粒度的光散射检测法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4568559A (en) * | 1984-02-06 | 1986-02-04 | Biotek, Inc. | Composite core coated microparticles and process of preparing same |
| NL193682C (nl) * | 1987-05-14 | 2000-07-04 | Glaxo Group Ltd | Beklede cefuroximaxetilsamenstelling. |
| CA2328080C (en) * | 1998-04-09 | 2008-08-12 | Eurand International S.P.A. | Wettable microcapsules having hydrophobic polymer coated cores |
| FR2811913B1 (fr) * | 2000-07-19 | 2003-09-19 | Separex Sa | Procede d'encapsulation sous forme de micro-capsules de fines particules solides |
| GB2405798A (en) * | 2003-09-15 | 2005-03-16 | Vectura Ltd | Dry powder inhaler with primary and secondary piercing elements and a medicament pack for use with an inhalation device. |
-
2005
- 2005-12-24 DE DE102005062270A patent/DE102005062270A1/de not_active Withdrawn
-
2006
- 2006-12-20 US US12/158,725 patent/US20090269411A1/en not_active Abandoned
- 2006-12-20 EP EP06829765A patent/EP1968555A2/de not_active Withdrawn
- 2006-12-20 CA CA002634481A patent/CA2634481A1/en not_active Abandoned
- 2006-12-20 RU RU2008130171/15A patent/RU2440103C2/ru not_active IP Right Cessation
- 2006-12-20 BR BRPI0620618-2A patent/BRPI0620618A2/pt not_active IP Right Cessation
- 2006-12-20 AU AU2006331009A patent/AU2006331009B2/en not_active Ceased
- 2006-12-20 JP JP2008546239A patent/JP5275039B2/ja not_active Expired - Fee Related
- 2006-12-20 KR KR1020087016451A patent/KR20080081021A/ko not_active Ceased
- 2006-12-20 NZ NZ569279A patent/NZ569279A/en not_active IP Right Cessation
- 2006-12-20 UA UAA200809702A patent/UA93072C2/ru unknown
- 2006-12-20 MY MYPI20082294A patent/MY149601A/en unknown
- 2006-12-20 CN CNA2006800490555A patent/CN101346133A/zh active Pending
- 2006-12-20 KR KR1020117031078A patent/KR101245627B1/ko not_active Expired - Fee Related
- 2006-12-20 WO PCT/EP2006/012284 patent/WO2007073911A2/de not_active Ceased
-
2008
- 2008-06-12 IL IL192085A patent/IL192085A0/en unknown
- 2008-06-19 MA MA31056A patent/MA30072B1/fr unknown
- 2008-06-23 GT GT200800126A patent/GT200800126A/es unknown
- 2008-06-23 CU CU20080124A patent/CU23877B1/es not_active IP Right Cessation
- 2008-06-23 EC EC2008008577A patent/ECSP088577A/es unknown
- 2008-06-23 CR CR10112A patent/CR10112A/es not_active Application Discontinuation
- 2008-06-23 SV SV2008002971A patent/SV2009002971A/es unknown
- 2008-06-23 TN TNP2008000284A patent/TNSN08284A1/en unknown
- 2008-06-24 ZA ZA200805498A patent/ZA200805498B/xx unknown
- 2008-06-24 HN HN2008000964A patent/HN2008000964A/es unknown
-
2013
- 2013-03-05 JP JP2013042861A patent/JP2013144695A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| UA93072C2 (ru) | 2011-01-10 |
| AU2006331009A1 (en) | 2007-07-05 |
| DE102005062270A1 (de) | 2007-06-28 |
| CU23877B1 (es) | 2013-04-19 |
| JP2013144695A (ja) | 2013-07-25 |
| JP5275039B2 (ja) | 2013-08-28 |
| KR20080081021A (ko) | 2008-09-05 |
| RU2440103C2 (ru) | 2012-01-20 |
| JP2009521419A (ja) | 2009-06-04 |
| MY149601A (en) | 2013-09-13 |
| SV2009002971A (es) | 2009-04-28 |
| AU2006331009B2 (en) | 2012-10-04 |
| KR101245627B1 (ko) | 2013-03-20 |
| US20090269411A1 (en) | 2009-10-29 |
| CA2634481A1 (en) | 2007-07-05 |
| ECSP088577A (es) | 2008-07-30 |
| CR10112A (es) | 2009-01-07 |
| EP1968555A2 (de) | 2008-09-17 |
| TNSN08284A1 (en) | 2009-10-30 |
| NZ569279A (en) | 2011-06-30 |
| CN101346133A (zh) | 2009-01-14 |
| WO2007073911A2 (de) | 2007-07-05 |
| HN2008000964A (es) | 2013-03-11 |
| CU20080124A7 (es) | 2010-08-30 |
| KR20120006085A (ko) | 2012-01-17 |
| ZA200805498B (en) | 2009-11-25 |
| IL192085A0 (en) | 2008-12-29 |
| GT200800126A (es) | 2010-06-25 |
| RU2008130171A (ru) | 2010-01-27 |
| WO2007073911A3 (de) | 2007-08-23 |
| MA30072B1 (fr) | 2008-12-01 |
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| B25A | Requested transfer of rights approved |
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| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 8A ANUIDADE. |
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| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
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