KR20050087791A - 클로로메틸 세펨 유도체 제조를 위한 개선된 제조방법 - Google Patents

클로로메틸 세펨 유도체 제조를 위한 개선된 제조방법 Download PDF

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Publication number
KR20050087791A
KR20050087791A KR1020057007694A KR20057007694A KR20050087791A KR 20050087791 A KR20050087791 A KR 20050087791A KR 1020057007694 A KR1020057007694 A KR 1020057007694A KR 20057007694 A KR20057007694 A KR 20057007694A KR 20050087791 A KR20050087791 A KR 20050087791A
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KR
South Korea
Prior art keywords
formula
para
chloromethyl
iii
methoxybenzyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
KR1020057007694A
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English (en)
Korean (ko)
Inventor
파라니사미 센띠쿠마 우다얌파라얌
산제이 니브루티 카라리
파드마나브한 라마
판두랑 볼원트 데쉬판데
Original Assignee
오키드 케미칼즈 앤드 파마수티컬즈 리미티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by 오키드 케미칼즈 앤드 파마수티컬즈 리미티드 filed Critical 오키드 케미칼즈 앤드 파마수티컬즈 리미티드
Publication of KR20050087791A publication Critical patent/KR20050087791A/ko
Withdrawn legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02—Preparation
    • C07D501/08—Preparation by forming the ring or condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Cephalosporin Compounds (AREA)
KR1020057007694A 2002-11-01 2003-10-23 클로로메틸 세펨 유도체 제조를 위한 개선된 제조방법 Withdrawn KR20050087791A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN808CH2002 2002-11-01
IN808/MAS/2002 2002-11-01

Publications (1)

Publication Number Publication Date
KR20050087791A true KR20050087791A (ko) 2005-08-31

Family

ID=35561711

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020057007694A Withdrawn KR20050087791A (ko) 2002-11-01 2003-10-23 클로로메틸 세펨 유도체 제조를 위한 개선된 제조방법

Country Status (5)

Country Link
JP (1) JP2006507289A (enExample)
KR (1) KR20050087791A (enExample)
CN (1) CN1315841C (enExample)
AU (1) AU2003269416A1 (enExample)
WO (1) WO2004039813A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005026176A1 (ja) * 2003-09-09 2005-03-24 Nippon Chemical Industrial Co.,Ltd. ３−クロロメチル-３-セフェム誘導体の製造方法
CN101260116A (zh) * 2008-04-21 2008-09-10 湖南有色凯铂生物药业有限公司 7-苯乙酰胺-3-氯甲基-4-头孢烷酸对甲氧苄酯的合成方法
CN102344459B (zh) * 2011-07-27 2014-08-06 山西新天源医药化工有限公司 一种头孢中间体gcle的制备方法
CN102643294B (zh) * 2012-04-18 2014-11-26 山东普洛得邦医药有限公司 一种头孢母核中间体的制备方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE35152B1 (en) * 1969-08-26 1975-11-26 Glaxo Lab Ltd Improvements in or relating to cephalosporin compounds
NL7411505A (nl) * 1973-09-06 1975-03-10 Rhone Poulenc Sa Werkwijze voor de bereiding en toepassing van nieuwe 7-trichlooraceetamido-3-desacetoxy-cefa- losporanzuurpreparaten.
AU498131B2 (en) * 1974-02-26 1979-02-15 Ciba-Geigy Ag Production of cephems by cyclization
JPS5874689A (ja) * 1981-10-29 1983-05-06 Otsuka Chem Co Ltd ３−クロロメチル−３−セフエム誘導体の製造法
JPS6043340B2 (ja) * 1981-04-10 1985-09-27 大塚化学薬品株式会社 塩素化アゼチジノン誘導体及びその製造法
GB2099817B (en) * 1981-04-10 1985-05-15 Otsuka Kagaku Yakuhin Azetidinone derivatives and process for the preparation of the same
JPS59164771A (ja) * 1983-03-10 1984-09-17 Otsuka Chem Co Ltd 塩素化アゼチジノン誘導体の製造方法
JPS60237061A (ja) * 1984-05-08 1985-11-25 Otsuka Chem Co Ltd アゼチジノン誘導体の製造法
JPS60115562A (ja) * 1983-11-28 1985-06-22 Otsuka Chem Co Ltd アゼチジノン誘導体の製造法
DE3933934A1 (de) * 1989-10-03 1991-04-11 Bayer Ag Verfahren zur herstellung von 7-amino-3-((z)-1-propen-1-yl)-3-cephem-4-carbonsaeure
JP3224279B2 (ja) * 1992-07-27 2001-10-29 大塚化学株式会社 セフエム化合物の製造法
JP4157177B2 (ja) * 1997-06-04 2008-09-24 大塚化学ホールディングス株式会社 ３−アルケニルセフェム化合物の製造法

Also Published As

Publication number Publication date
CN1315841C (zh) 2007-05-16
CN1708501A (zh) 2005-12-14
AU2003269416A1 (en) 2004-05-25
WO2004039813A1 (en) 2004-05-13
JP2006507289A (ja) 2006-03-02

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