KR101541203B1 - 피라지논 유도체 및 폐 질환의 치료에서 그의 용도 - Google Patents
피라지논 유도체 및 폐 질환의 치료에서 그의 용도 Download PDFInfo
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- KR101541203B1 KR101541203B1 KR1020107001749A KR20107001749A KR101541203B1 KR 101541203 B1 KR101541203 B1 KR 101541203B1 KR 1020107001749 A KR1020107001749 A KR 1020107001749A KR 20107001749 A KR20107001749 A KR 20107001749A KR 101541203 B1 KR101541203 B1 KR 101541203B1
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- alkyl
- methyl
- amino
- oxo
- benzamide
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- 0 CC(c1cc(*(C(*2)=C(*3)I)C(*)=C3I)c2c(*)c1)=O Chemical compound CC(c1cc(*(C(*2)=C(*3)I)C(*)=C3I)c2c(*)c1)=O 0.000 description 5
- SAZVRXTVWZAHBI-UHFFFAOYSA-N CC(C)(c1ccccc1OCCNC)NC1=NC=CN(c2c(C)ccc(C(NC3CC3)=O)c2)C1=O Chemical compound CC(C)(c1ccccc1OCCNC)NC1=NC=CN(c2c(C)ccc(C(NC3CC3)=O)c2)C1=O SAZVRXTVWZAHBI-UHFFFAOYSA-N 0.000 description 1
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- MPIMGWLQRISQEA-UHFFFAOYSA-N CCNC(c1ccc(C)c(N(C=CN=C2NCc3ccccc3)C2=O)c1)=O Chemical compound CCNC(c1ccc(C)c(N(C=CN=C2NCc3ccccc3)C2=O)c1)=O MPIMGWLQRISQEA-UHFFFAOYSA-N 0.000 description 1
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- AEJXIGXJEDGFLR-UHFFFAOYSA-N Cc(c(N(C=CN=C1NC2(CC2)c(cccc2)c2OCCNC)C1=O)c1)cc(F)c1C(NC1CC1)=O Chemical compound Cc(c(N(C=CN=C1NC2(CC2)c(cccc2)c2OCCNC)C1=O)c1)cc(F)c1C(NC1CC1)=O AEJXIGXJEDGFLR-UHFFFAOYSA-N 0.000 description 1
- OYKIDFXQQWIOQP-XMMPIXPASA-N Cc(c(N(C=CN=C1N[C@H](CC(N2CCN(C)CC2)=O)c2ccccc2)C1=O)c1)ccc1C(NC1CC1)=O Chemical compound Cc(c(N(C=CN=C1N[C@H](CC(N2CCN(C)CC2)=O)c2ccccc2)C1=O)c1)ccc1C(NC1CC1)=O OYKIDFXQQWIOQP-XMMPIXPASA-N 0.000 description 1
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- NAIILALUCIFGCO-UHFFFAOYSA-N Cc(ccc(C(NC1CC1)=O)c1)c1N(C=CN=C1NCc(cccc2)c2OCCN2CCCC2)C1=O Chemical compound Cc(ccc(C(NC1CC1)=O)c1)c1N(C=CN=C1NCc(cccc2)c2OCCN2CCCC2)C1=O NAIILALUCIFGCO-UHFFFAOYSA-N 0.000 description 1
- CHODZWUTQMXBGR-UHFFFAOYSA-N Cc(ccc(C(NC1CC1)=O)c1)c1N(C=CN=C1c2ccccc2)C1=O Chemical compound Cc(ccc(C(NC1CC1)=O)c1)c1N(C=CN=C1c2ccccc2)C1=O CHODZWUTQMXBGR-UHFFFAOYSA-N 0.000 description 1
- ORGIAWBDTNBZMA-UHFFFAOYSA-N Cc(ccc(C(NOC)=O)c1)c1N(C=CN=C1NCc2c(CN3CCN(C)CC3)cccc2)C1=O Chemical compound Cc(ccc(C(NOC)=O)c1)c1N(C=CN=C1NCc2c(CN3CCN(C)CC3)cccc2)C1=O ORGIAWBDTNBZMA-UHFFFAOYSA-N 0.000 description 1
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| WO2013057322A1 (en) | 2011-10-20 | 2013-04-25 | Oryzon Genomics, S.A. | (hetero)aryl cyclopropylamine compounds as lsd1 inhibitors |
| BR112014009306B1 (pt) | 2011-10-20 | 2021-07-20 | Oryzon Genomics S.A. | Compostos de (hetero)aril ciclopropilamina como inibidores de lsd1 |
| KR20150000900A (ko) | 2012-04-10 | 2015-01-05 | 다이닛본 스미토모 세이야꾸 가부시끼가이샤 | 신규한 1-치환된 인다졸 유도체 |
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