KR101273614B1 - 중합체 부분을 포함하는 다가 ｖｌａ―４ 길항제 - Google Patents

중합체 부분을 포함하는 다가 ｖｌａ―４ 길항제 Download PDF

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Publication number
KR101273614B1
KR101273614B1 KR1020077003108A KR20077003108A KR101273614B1 KR 101273614 B1 KR101273614 B1 KR 101273614B1 KR 1020077003108 A KR1020077003108 A KR 1020077003108A KR 20077003108 A KR20077003108 A KR 20077003108A KR 101273614 B1 KR101273614 B1 KR 101273614B1
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KR
South Korea
Prior art keywords
substituted
alkyl
aryl
group
heteroaryl
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KR1020077003108A
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English (en)
Korean (ko)
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KR20070051267A (ko
Inventor
안드레이 더블유. 콘라디
마이클 에이. 플레이스
크리스토퍼 엠. 셈코
테오도르 예드노크
제니퍼 엘. 스미스
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엘란 파마슈티칼스, 인크.
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Publication of KR20070051267A publication Critical patent/KR20070051267A/ko
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/74—Synthetic polymeric materials
    • A61K31/785—Polymers containing nitrogen
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
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KR1020077003108A 2004-07-08 2005-07-08 중합체 부분을 포함하는 다가 ｖｌａ―４ 길항제 KR101273614B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US58697504P 2004-07-08 2004-07-08
US60/586,975 2004-07-08
PCT/US2005/024369 WO2006010054A2 (en) 2004-07-08 2005-07-08 Multivalent vla-4 antagonists comprising polyethylene glycol moieties

Publications (2)

Publication Number Publication Date
KR20070051267A KR20070051267A (ko) 2007-05-17
KR101273614B1 true KR101273614B1 (ko) 2013-06-12

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US (4) US7794700B2 (US07794700-20100914-C00065.png)
EP (4) EP2298356A3 (US07794700-20100914-C00065.png)
JP (1) JP2008505927A (US07794700-20100914-C00065.png)
KR (1) KR101273614B1 (US07794700-20100914-C00065.png)
CN (1) CN101035563B (US07794700-20100914-C00065.png)
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MA (1) MA28786B1 (US07794700-20100914-C00065.png)
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