KR101245627B1 - 산제의 맛 차단 - Google Patents

산제의 맛 차단 Download PDF

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Publication number
KR101245627B1
KR101245627B1 KR1020117031078A KR20117031078A KR101245627B1 KR 101245627 B1 KR101245627 B1 KR 101245627B1 KR 1020117031078 A KR1020117031078 A KR 1020117031078A KR 20117031078 A KR20117031078 A KR 20117031078A KR 101245627 B1 KR101245627 B1 KR 101245627B1
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KR
South Korea
Prior art keywords
taste
powder
wax
temperature
mixture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR1020117031078A
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English (en)
Korean (ko)
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KR20120006085A (ko
Inventor
라이너 벨링하우젠
다니엘 루드하르트
프랭크 라이더
마틴 스타인백
제스코 장크
마틴 와이스
올라프 베렌드
스팁하우트 우도 판
Original Assignee
바이엘 인텔렉쳐 프로퍼티 게엠베하
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication of KR20120006085A publication Critical patent/KR20120006085A/ko
Application granted granted Critical
Publication of KR101245627B1 publication Critical patent/KR101245627B1/ko
Expired - Fee Related legal-status Critical Current
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/007—Pulmonary tract; Aromatherapy
    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5015—Organic compounds, e.g. fats, sugars
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5089—Processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Otolaryngology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Seasonings (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020117031078A 2005-12-24 2006-12-20 산제의 맛 차단 Expired - Fee Related KR101245627B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102005062270A DE102005062270A1 (de) 2005-12-24 2005-12-24 Geschmacksmaskierung von Pulvern
DE102005062270.4 2005-12-24
PCT/EP2006/012284 WO2007073911A2 (de) 2005-12-24 2006-12-20 Geschmacksmaskierung von pulvern

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020087016451A Division KR20080081021A (ko) 2005-12-24 2006-12-20 산제의 맛 차단

Publications (2)

Publication Number Publication Date
KR20120006085A KR20120006085A (ko) 2012-01-17
KR101245627B1 true KR101245627B1 (ko) 2013-03-20

Family

ID=38042692

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020087016451A Ceased KR20080081021A (ko) 2005-12-24 2006-12-20 산제의 맛 차단
KR1020117031078A Expired - Fee Related KR101245627B1 (ko) 2005-12-24 2006-12-20 산제의 맛 차단

Family Applications Before (1)

Application Number Title Priority Date Filing Date
KR1020087016451A Ceased KR20080081021A (ko) 2005-12-24 2006-12-20 산제의 맛 차단

Country Status (24)

Country Link
US (1) US20090269411A1 (enExample)
EP (1) EP1968555A2 (enExample)
JP (2) JP5275039B2 (enExample)
KR (2) KR20080081021A (enExample)
CN (1) CN101346133A (enExample)
AU (1) AU2006331009B2 (enExample)
BR (1) BRPI0620618A2 (enExample)
CA (1) CA2634481A1 (enExample)
CR (1) CR10112A (enExample)
CU (1) CU23877B1 (enExample)
DE (1) DE102005062270A1 (enExample)
EC (1) ECSP088577A (enExample)
GT (1) GT200800126A (enExample)
HN (1) HN2008000964A (enExample)
IL (1) IL192085A0 (enExample)
MA (1) MA30072B1 (enExample)
MY (1) MY149601A (enExample)
NZ (1) NZ569279A (enExample)
RU (1) RU2440103C2 (enExample)
SV (1) SV2009002971A (enExample)
TN (1) TNSN08284A1 (enExample)
UA (1) UA93072C2 (enExample)
WO (1) WO2007073911A2 (enExample)
ZA (1) ZA200805498B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0327723D0 (en) 2003-09-15 2003-12-31 Vectura Ltd Pharmaceutical compositions
EP2050437A1 (en) * 2007-10-15 2009-04-22 Laboratoires SMB Improved pharmaceutical dry powder compositions for inhalation.
CN102006857B (zh) * 2008-02-13 2013-06-26 拜耳先灵医药股份有限公司 具有稳定作用的药物递送系统
WO2009101021A2 (en) * 2008-02-13 2009-08-20 Bayer Schering Pharma Aktiengesellschaft Estradiol-containing drug delivery system
NZ593217A (en) * 2008-12-05 2013-05-31 Bayer Ip Gmbh Extrudate having spicular active substances
PT3130396T (pt) 2009-03-27 2021-05-12 Bend Res Inc Processo de secagem por pulverização
UY32836A (es) * 2009-08-12 2011-03-31 Bayer Schering Pharma Ag Partículas estabilizadas que comprenden 5-metil-(6s)-tetrahidrofolato
WO2011020610A1 (en) 2009-08-19 2011-02-24 Bayer Schering Pharma Aktiengesellschaft Drug delivery systems (wafer) for pediatric use
EP2611529B1 (en) 2010-09-03 2019-01-23 Bend Research, Inc. Spray-drying method
US8815294B2 (en) 2010-09-03 2014-08-26 Bend Research, Inc. Pharmaceutical compositions of dextran polymer derivatives and a carrier material
EP2611530B1 (en) 2010-09-03 2019-01-16 Bend Research, Inc. Spray-drying apparatus and methods of using the same
EP2629913B1 (en) 2010-09-20 2020-08-26 SPI Pharma, INC. Microencapsulation process and product
EP2618924A1 (en) 2010-09-24 2013-07-31 Bend Research, Inc. High-temperature spray drying process and apparatus
HU231017B1 (hu) 2012-05-08 2019-11-28 LAVET Gyógyszeripari Kft. Praziquantel tartalmú ízfedett formulációk
US8993041B2 (en) * 2012-10-15 2015-03-31 New Jersey Institute Of Technology Taste masked active pharmaceutical powder compositions and processes for making them
EP3212169B1 (en) 2014-10-31 2021-01-13 Bend Research, Inc. Process for forming active domains dispersed in a matrix
CN114993892B (zh) * 2019-05-13 2024-10-18 南京制药厂有限公司 吡喹酮粒度的光散射检测法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999052510A1 (en) * 1998-04-09 1999-10-21 Eurand International S.P.A. Wettable microcapsules having hydrophobic polymer coated cores

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4568559A (en) * 1984-02-06 1986-02-04 Biotek, Inc. Composite core coated microparticles and process of preparing same
NL193682C (nl) * 1987-05-14 2000-07-04 Glaxo Group Ltd Beklede cefuroximaxetilsamenstelling.
FR2811913B1 (fr) * 2000-07-19 2003-09-19 Separex Sa Procede d'encapsulation sous forme de micro-capsules de fines particules solides
GB2405798A (en) * 2003-09-15 2005-03-16 Vectura Ltd Dry powder inhaler with primary and secondary piercing elements and a medicament pack for use with an inhalation device.

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999052510A1 (en) * 1998-04-09 1999-10-21 Eurand International S.P.A. Wettable microcapsules having hydrophobic polymer coated cores

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
Journal of Applied Physiology. 1998, 제84권 717-725쪽. *
Journal of Applied Physiology. 1998, 제84권 717-725쪽.*

Also Published As

Publication number Publication date
EP1968555A2 (de) 2008-09-17
NZ569279A (en) 2011-06-30
CR10112A (es) 2009-01-07
KR20080081021A (ko) 2008-09-05
KR20120006085A (ko) 2012-01-17
WO2007073911A3 (de) 2007-08-23
US20090269411A1 (en) 2009-10-29
CU23877B1 (es) 2013-04-19
MY149601A (en) 2013-09-13
JP2013144695A (ja) 2013-07-25
JP5275039B2 (ja) 2013-08-28
JP2009521419A (ja) 2009-06-04
CN101346133A (zh) 2009-01-14
BRPI0620618A2 (pt) 2011-11-16
CU20080124A7 (es) 2010-08-30
MA30072B1 (fr) 2008-12-01
AU2006331009A1 (en) 2007-07-05
RU2008130171A (ru) 2010-01-27
ECSP088577A (es) 2008-07-30
GT200800126A (es) 2010-06-25
IL192085A0 (en) 2008-12-29
RU2440103C2 (ru) 2012-01-20
TNSN08284A1 (en) 2009-10-30
AU2006331009B2 (en) 2012-10-04
DE102005062270A1 (de) 2007-06-28
CA2634481A1 (en) 2007-07-05
WO2007073911A2 (de) 2007-07-05
HN2008000964A (es) 2013-03-11
UA93072C2 (ru) 2011-01-10
ZA200805498B (en) 2009-11-25
SV2009002971A (es) 2009-04-28

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