KR100850252B1 - 유기 화합물 - Google Patents

유기 화합물 Download PDF

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Publication number
KR100850252B1
KR100850252B1 KR1020037007242A KR20037007242A KR100850252B1 KR 100850252 B1 KR100850252 B1 KR 100850252B1 KR 1020037007242 A KR1020037007242 A KR 1020037007242A KR 20037007242 A KR20037007242 A KR 20037007242A KR 100850252 B1 KR100850252 B1 KR 100850252B1
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KR
South Korea
Prior art keywords
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london
halogen
page
crop protection
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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KR1020037007242A
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English (en)
Korean (ko)
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KR20030061414A (ko
Inventor
두크레이피에르
보비에르야쿠스
Original Assignee
노파르티스 아게
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Publication of KR20030061414A publication Critical patent/KR20030061414A/ko
Application granted granted Critical
Publication of KR100850252B1 publication Critical patent/KR100850252B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

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  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Paper (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020037007242A 2000-12-20 2001-12-18 유기 화합물 Expired - Fee Related KR100850252B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH2489/00 2000-12-20
CH24892000 2000-12-20
PCT/EP2001/014926 WO2002049641A2 (en) 2000-12-20 2001-12-18 Anti-endoparasitic amidoacetonitrils

Publications (2)

Publication Number Publication Date
KR20030061414A KR20030061414A (ko) 2003-07-18
KR100850252B1 true KR100850252B1 (ko) 2008-08-04

Family

ID=4569596

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020037007242A Expired - Fee Related KR100850252B1 (ko) 2000-12-20 2001-12-18 유기 화합물

Country Status (21)

Country Link
US (1) US7700656B2 (https=)
EP (1) EP1392281B1 (https=)
JP (1) JP2004521097A (https=)
KR (1) KR100850252B1 (https=)
CN (1) CN1531426A (https=)
AR (1) AR035523A1 (https=)
AT (1) ATE354360T1 (https=)
AU (2) AU3458802A (https=)
BR (1) BR0116326A (https=)
CA (1) CA2432388C (https=)
CY (1) CY1106509T1 (https=)
DE (1) DE60126838T2 (https=)
DK (1) DK1392281T3 (https=)
ES (1) ES2281453T3 (https=)
MX (1) MXPA03005701A (https=)
NZ (1) NZ526538A (https=)
PT (1) PT1392281E (https=)
RU (1) RU2286775C2 (https=)
TW (1) TWI292712B (https=)
WO (1) WO2002049641A2 (https=)
ZA (1) ZA200304331B (https=)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035531A1 (es) * 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
AR036054A1 (es) 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
TWI261053B (en) * 2001-12-06 2006-09-01 Novartis Ag Amidoacetonitrile compounds, their preparation, compositions and use as pesticides
AR039020A1 (es) * 2002-03-21 2005-02-02 Novartis Ag Compuestos de aminoacetonitrilo
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
AR042420A1 (es) * 2002-09-11 2005-06-22 Novartis Ag Benzotriazolil- aminoacetonitril compuestos, proceso para su preparacion, metodo y uso de los mismos en el control de endo- y ecto-parasitos dentro y sobre ganado productor de sangre caliente y animales domesticos y plantas, y en la preparacion de una composicion farmaceutica
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
AR049391A1 (es) * 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) * 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
EP1812385B1 (en) * 2004-11-09 2012-07-18 Novartis AG Process for the preparation of enantiomers of amidoacetonitrile compounds from their racemates
EP1910278A1 (en) * 2005-07-25 2008-04-16 Novartis AG Amidonitrile compounds
DE102006025874A1 (de) 2006-06-02 2007-12-06 Bayer Cropscience Ag Alkoxyalkyl-substituierte cyclische Ketoenole
WO2008062005A1 (en) * 2006-11-24 2008-05-29 Novartis Ag The use of aminoacetonitril compounds in the control of endoparasites in warm- blood animals.
KR20110098012A (ko) 2007-02-09 2011-08-31 화이자 리미티드 구충제
ES2367332T3 (es) 2007-02-21 2011-11-02 Pfizer Limited Agentes antiparasitarios de benzofurano.
ES2597083T3 (es) * 2007-05-15 2017-01-13 Merial, Inc. Compuestos de ariloazol-2-il cianoetilamino, procedimiento de fabricación y procedimiento de utilización de los mismos
KR101782308B1 (ko) * 2008-10-21 2017-09-27 메리얼 인코포레이티드 티오아미드 화합물, 이의 제조 방법 및 사용 방법
MY153715A (en) 2008-11-14 2015-03-13 Merial Ltd Enantiomerically enriched aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
UY33282A (es) * 2010-03-25 2011-09-30 Novartis Ag Composiciones endoparasiticidas
AU2012224015B2 (en) 2011-03-02 2017-04-13 Nihon Nohyaku Co., Ltd. Internal parasiticide
MX349802B (es) * 2011-11-25 2017-08-14 Bayer Ip Gmbh Uso de aril- y hetarilcarboxamidas como endoparasiticidas.
CN104105688A (zh) * 2012-02-14 2014-10-15 日本曹达株式会社 芳氧基乙酰胺化合物和有害生物防除剂
EP2880014B1 (en) 2012-08-06 2017-05-17 Pitney Pharmaceuticals Pty Limited Compounds for the treatment of mtor pathway related diseases
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
AR094961A1 (es) 2013-03-15 2015-09-09 Lilly Co Eli 1-hidroxi-benzooxaboroles como agentes antiparasitarios
EP2821412A1 (en) * 2013-07-01 2015-01-07 Universität Zürich Organometallic 2-cyano-2-aminobenzoate-propyl derivates and their use as anthelmintics
JP6556700B2 (ja) * 2013-09-13 2019-08-07 ピットニー ファーマシューティカル ピーティーワイ リミテッド アミノアセトニトリル化合物を有効成分として含有する抗癌剤
AU2016224395A1 (en) * 2015-02-24 2017-08-31 Pitney Pharmaceuticals Pty Limited Anti cancer agent comprising aminoacetonitrile compound as active ingredient
EP3235815A1 (de) 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1520925A (fr) 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
EP0953565A2 (en) * 1998-05-01 1999-11-03 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative, agricultural and horticultural insecticide containing the same, and use thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3457294A (en) * 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
US4515731A (en) * 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
GB8517279D0 (en) * 1985-07-08 1985-08-14 Ici Plc Benzamide derivatives
JP2994182B2 (ja) * 1992-07-23 1999-12-27 石原産業株式会社 アミド系化合物又はその塩、それらの製造方法及びそれらを含有する有害動物防除剤
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
MXPA03010404A (es) * 2001-05-15 2004-03-09 Novartis Ag Benzamidoacetonitrilos y su uso como antiparasitarios.
AR036054A1 (es) * 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR038156A1 (es) * 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1520925A (fr) 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
EP0953565A2 (en) * 1998-05-01 1999-11-03 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative, agricultural and horticultural insecticide containing the same, and use thereof

Also Published As

Publication number Publication date
EP1392281A2 (en) 2004-03-03
ES2281453T3 (es) 2007-10-01
WO2002049641A2 (en) 2002-06-27
US7700656B2 (en) 2010-04-20
US20040082624A1 (en) 2004-04-29
DE60126838T2 (de) 2007-11-08
DE60126838D1 (de) 2007-04-05
AU2002234588B2 (en) 2005-03-24
CA2432388A1 (en) 2002-06-27
CA2432388C (en) 2010-06-08
KR20030061414A (ko) 2003-07-18
DK1392281T3 (da) 2007-06-11
PT1392281E (pt) 2007-05-31
EP1392281B1 (en) 2007-02-21
CN1531426A (zh) 2004-09-22
JP2004521097A (ja) 2004-07-15
AU3458802A (en) 2002-07-01
RU2286775C2 (ru) 2006-11-10
TWI292712B (en) 2008-01-21
ZA200304331B (en) 2004-04-28
AR035523A1 (es) 2004-06-02
CY1106509T1 (el) 2012-01-25
NZ526538A (en) 2005-12-23
RU2003122196A (ru) 2005-03-20
ATE354360T1 (de) 2007-03-15
WO2002049641A3 (en) 2003-12-04
MXPA03005701A (es) 2003-10-06
BR0116326A (pt) 2004-07-06

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