ATE354360T1 - Amidoacetonitrile zur bekämpfung von endoparasiten - Google Patents

Amidoacetonitrile zur bekämpfung von endoparasiten

Info

Publication number
ATE354360T1
ATE354360T1 AT01985421T AT01985421T ATE354360T1 AT E354360 T1 ATE354360 T1 AT E354360T1 AT 01985421 T AT01985421 T AT 01985421T AT 01985421 T AT01985421 T AT 01985421T AT E354360 T1 ATE354360 T1 AT E354360T1
Authority
AT
Austria
Prior art keywords
amidoacetonitriles
endoparasites
fight
fight endoparasites
Prior art date
Application number
AT01985421T
Other languages
German (de)
English (en)
Inventor
Pierre Ducray
Jacques Bouvier
Original Assignee
Novartis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh
Application granted granted Critical
Publication of ATE354360T1 publication Critical patent/ATE354360T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Paper (AREA)
AT01985421T 2000-12-20 2001-12-18 Amidoacetonitrile zur bekämpfung von endoparasiten ATE354360T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH24892000 2000-12-20

Publications (1)

Publication Number Publication Date
ATE354360T1 true ATE354360T1 (de) 2007-03-15

Family

ID=4569596

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01985421T ATE354360T1 (de) 2000-12-20 2001-12-18 Amidoacetonitrile zur bekämpfung von endoparasiten

Country Status (21)

Country Link
US (1) US7700656B2 (https=)
EP (1) EP1392281B1 (https=)
JP (1) JP2004521097A (https=)
KR (1) KR100850252B1 (https=)
CN (1) CN1531426A (https=)
AR (1) AR035523A1 (https=)
AT (1) ATE354360T1 (https=)
AU (2) AU3458802A (https=)
BR (1) BR0116326A (https=)
CA (1) CA2432388C (https=)
CY (1) CY1106509T1 (https=)
DE (1) DE60126838T2 (https=)
DK (1) DK1392281T3 (https=)
ES (1) ES2281453T3 (https=)
MX (1) MXPA03005701A (https=)
NZ (1) NZ526538A (https=)
PT (1) PT1392281E (https=)
RU (1) RU2286775C2 (https=)
TW (1) TWI292712B (https=)
WO (1) WO2002049641A2 (https=)
ZA (1) ZA200304331B (https=)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
AR036054A1 (es) 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR037746A1 (es) * 2001-12-06 2004-12-01 Novartis Ag Compuestos derivados de amidoacetonitrilo, un procedimiento para su preparacion, un procedimiento para la preparacion de compuestos intermediarios, una composicion para combatir parasitos, un procedimiento para combatir dichos parasitos, y el empleo de dichos derivados para la preparacion de una com
TW200305556A (en) * 2002-03-21 2003-11-01 Novartis Ag Organic compounds
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
AR042420A1 (es) 2002-09-11 2005-06-22 Novartis Ag Benzotriazolil- aminoacetonitril compuestos, proceso para su preparacion, metodo y uso de los mismos en el control de endo- y ecto-parasitos dentro y sobre ganado productor de sangre caliente y animales domesticos y plantas, y en la preparacion de una composicion farmaceutica
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
AR049391A1 (es) * 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) * 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
AU2005303993B2 (en) * 2004-11-09 2009-10-29 Elanco Tiergesundheit Ag Process for the preparation of enantiomers of amidoacetonitrile compounds from their racemates
US20080227863A1 (en) * 2005-07-25 2008-09-18 Novartis Ag Organic Compounds
DE102006025874A1 (de) 2006-06-02 2007-12-06 Bayer Cropscience Ag Alkoxyalkyl-substituierte cyclische Ketoenole
WO2008062005A1 (en) * 2006-11-24 2008-05-29 Novartis Ag The use of aminoacetonitril compounds in the control of endoparasites in warm- blood animals.
KR20110098012A (ko) 2007-02-09 2011-08-31 화이자 리미티드 구충제
ES2367332T3 (es) * 2007-02-21 2011-11-02 Pfizer Limited Agentes antiparasitarios de benzofurano.
RS55271B1 (sr) 2007-05-15 2017-02-28 Merial Sas Ariloazol-2-il cijanoetilamino jedinjenja, postupci dobijanja i postupci njihove primene
MX2011004217A (es) 2008-10-21 2011-06-20 Merial Ltd Compuestos de tioamida, metodo de elaboracion y metodo para usarlos.
AR074024A1 (es) 2008-11-14 2010-12-15 Merial Ltd Compuesto de arilazol-2-il-cianoetilamino enantiomericamente enriquecidos, composicion plaguicida y su uso para prevenir la infeccion parasitaria
UY33282A (es) * 2010-03-25 2011-09-30 Novartis Ag Composiciones endoparasiticidas
PH12013501809A1 (en) 2011-03-02 2013-10-14 Nihon Nohyaku Co Ltd Endoparasite control agent
RU2638830C2 (ru) * 2011-11-25 2017-12-18 Байер Интеллектуэль Проперти Гмбх Применение арильных и гетарильных карбоксамидов в качестве эндопаразитицидов
CA2863384C (en) * 2012-02-14 2017-08-29 Nippon Soda Co., Ltd. Aryloxyacetamide compound and pesticide
PL2880014T3 (pl) * 2012-08-06 2017-10-31 Pitney Pharmaceuticals Pty Ltd Związki do leczenia chorób związanych ze szlakiem mTOR
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
AR094961A1 (es) 2013-03-15 2015-09-09 Lilly Co Eli 1-hidroxi-benzooxaboroles como agentes antiparasitarios
EP2821412A1 (en) * 2013-07-01 2015-01-07 Universität Zürich Organometallic 2-cyano-2-aminobenzoate-propyl derivates and their use as anthelmintics
ES2727531T3 (es) * 2013-09-13 2019-10-16 Pitney Pharmaceuticals Pty Ltd Antineoplásico que comprende un compuesto de aminoacetonitrilo como ingrediente activo
US10391076B2 (en) * 2015-02-24 2019-08-27 Pitney Pharmaceuticals Pty Ltd. Anti-cancer agent comprising aminoacetonitrile compound as active ingredient
EP3235815A1 (de) 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3457294A (en) 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
FR1520925A (fr) 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
US4515731A (en) 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
GB8517279D0 (en) 1985-07-08 1985-08-14 Ici Plc Benzamide derivatives
JP2994182B2 (ja) * 1992-07-23 1999-12-27 石原産業株式会社 アミド系化合物又はその塩、それらの製造方法及びそれらを含有する有害動物防除剤
US6239077B1 (en) * 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
CA2447084A1 (en) 2001-05-15 2002-11-21 Novartis Ag Benzamidoacetonitriles and their use as antiparasitics
AR036054A1 (es) 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR038156A1 (es) * 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica

Also Published As

Publication number Publication date
KR20030061414A (ko) 2003-07-18
US20040082624A1 (en) 2004-04-29
CY1106509T1 (el) 2012-01-25
ES2281453T3 (es) 2007-10-01
CN1531426A (zh) 2004-09-22
PT1392281E (pt) 2007-05-31
ZA200304331B (en) 2004-04-28
US7700656B2 (en) 2010-04-20
EP1392281A2 (en) 2004-03-03
CA2432388C (en) 2010-06-08
EP1392281B1 (en) 2007-02-21
WO2002049641A3 (en) 2003-12-04
AU3458802A (en) 2002-07-01
RU2003122196A (ru) 2005-03-20
DE60126838D1 (de) 2007-04-05
MXPA03005701A (es) 2003-10-06
JP2004521097A (ja) 2004-07-15
AR035523A1 (es) 2004-06-02
KR100850252B1 (ko) 2008-08-04
RU2286775C2 (ru) 2006-11-10
AU2002234588B2 (en) 2005-03-24
DE60126838T2 (de) 2007-11-08
DK1392281T3 (da) 2007-06-11
TWI292712B (en) 2008-01-21
NZ526538A (en) 2005-12-23
BR0116326A (pt) 2004-07-06
CA2432388A1 (en) 2002-06-27
WO2002049641A2 (en) 2002-06-27

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