EE05197B1 - Linesoliid - kristallivorm II - Google Patents
Linesoliid - kristallivorm IIInfo
- Publication number
- EE05197B1 EE05197B1 EEP200200420A EEP200200420A EE05197B1 EE 05197 B1 EE05197 B1 EE 05197B1 EE P200200420 A EEP200200420 A EE P200200420A EE P200200420 A EEP200200420 A EE P200200420A EE 05197 B1 EE05197 B1 EE 05197B1
- Authority
- EE
- Estonia
- Prior art keywords
- linezolid
- crystalline form
- crystalline
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/22—Oxygen atoms attached in position 2 with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to other ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US17983700P | 2000-02-02 | 2000-02-02 | |
PCT/US2001/000657 WO2001057035A1 (en) | 2000-02-02 | 2001-01-29 | Linezolid-crystal form ii |
Publications (2)
Publication Number | Publication Date |
---|---|
EE200200420A EE200200420A (et) | 2003-12-15 |
EE05197B1 true EE05197B1 (et) | 2009-08-17 |
Family
ID=22658183
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EEP200200420A EE05197B1 (et) | 2000-02-02 | 2001-01-29 | Linesoliid - kristallivorm II |
Country Status (31)
Country | Link |
---|---|
EP (1) | EP1255754B1 (et) |
JP (1) | JP5235256B2 (et) |
KR (3) | KR100864745B1 (et) |
CN (1) | CN1221547C (et) |
AR (1) | AR027261A1 (et) |
AT (1) | ATE297920T1 (et) |
AU (1) | AU782138B2 (et) |
BR (1) | BR0107667A (et) |
CA (1) | CA2395603C (et) |
CO (1) | CO5261555A1 (et) |
CZ (1) | CZ302292B6 (et) |
DE (1) | DE60111497T2 (et) |
DK (1) | DK1255754T3 (et) |
EA (1) | EA004434B1 (et) |
EE (1) | EE05197B1 (et) |
ES (1) | ES2242728T3 (et) |
HK (1) | HK1051196A1 (et) |
HU (1) | HUP0301076A3 (et) |
IL (1) | IL151010A0 (et) |
MX (1) | MXPA02007471A (et) |
MY (1) | MY122829A (et) |
NO (2) | NO323459B1 (et) |
NZ (1) | NZ520541A (et) |
PE (1) | PE20011086A1 (et) |
PL (1) | PL356433A1 (et) |
PT (1) | PT1255754E (et) |
SI (1) | SI1255754T1 (et) |
SK (1) | SK287025B6 (et) |
TW (1) | TWI297687B (et) |
WO (1) | WO2001057035A1 (et) |
ZA (1) | ZA200205162B (et) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100490643B1 (ko) * | 2002-10-29 | 2005-05-19 | 한국과학기술연구원 | 새로운 메틸리덴 피페리딘일 옥사졸리딘온 유도체 및이들의 제조방법 |
ES2331454T1 (es) | 2003-10-16 | 2010-01-05 | Symed Labs Limited | Forma cristalina de linezolid. |
EP1737850B1 (en) | 2004-04-19 | 2007-10-03 | Symed Labs Limited | A novel process for the preparation of linezolid and related compounds |
WO2006004922A1 (en) * | 2004-06-29 | 2006-01-12 | Teva Pharmaceutical Industries Ltd. | Crystalline form iv of linezolid |
WO2006110155A1 (en) * | 2004-06-29 | 2006-10-19 | Teva Pharmaceutical Industries Ltd | Solid forms of linezolid and processes for preparation thereof |
CA2602073A1 (en) | 2005-02-24 | 2006-08-31 | Teva Pharmaceutical Industries Ltd. | Processes for the preparation of linezolid intermediate |
KR20070062504A (ko) * | 2005-06-22 | 2007-06-15 | 테바 파마슈티컬 인더스트리즈 리미티드 | 테가세로드 말레이트의 다형태 |
DE602006001699D1 (de) * | 2005-07-20 | 2008-08-21 | Teva Pharma | Stabile pharmazeutische Zusammensetzung mit Linezolid Form IV |
WO2007102082A1 (en) * | 2006-03-09 | 2007-09-13 | Glenmark Pharmaceuticals Limited | High oxazolidinone content solid dosage forms |
CA2703011A1 (en) * | 2006-10-23 | 2008-10-23 | Concert Pharmaceuticals Inc. | Oxazolidinone derivatives and methods of use |
WO2011050826A1 (en) | 2009-10-28 | 2011-05-05 | Synthon B.V. | Process for making crystalline form a of linezolid |
EP2563781B1 (en) | 2010-04-30 | 2016-10-26 | Indiana University Research and Technology Corporation | Processes for preparing linezolid |
EP2603506A1 (en) | 2010-08-11 | 2013-06-19 | Synthon BV | Process for making linezolid |
EP2603505A1 (en) | 2010-08-11 | 2013-06-19 | Synthon BV | Process for making linezolid |
EP2593440A1 (en) * | 2011-02-24 | 2013-05-22 | Lee Pharma Limited | Anhydrous linezolid crystalline form-ii |
WO2012119653A1 (en) | 2011-03-09 | 2012-09-13 | Synthon Bv | Process for making crystalline form a of linezolid |
CN102731341A (zh) * | 2011-04-13 | 2012-10-17 | 上海医药工业研究院 | 用于制备利奈唑胺的中间体及其制备方法 |
CN102766106A (zh) * | 2011-05-03 | 2012-11-07 | 江苏豪森医药集团有限公司 | 利奈唑胺的新晶型及其制备方法 |
CN102399200B (zh) * | 2011-12-14 | 2013-12-04 | 浙江新东港药业股份有限公司 | 一种利用悬浮结晶法制备利奈唑胺晶型ⅰ的方法 |
EP2852580A1 (en) | 2012-01-24 | 2015-04-01 | Jubilant Life Sciences Ltd. | Improved process for the preparation of stable crystalline form-i of linezolid, substantially free of residual solvent |
WO2013120496A1 (en) | 2012-02-14 | 2013-08-22 | Pharmathen S.A. | Process for the preparation of linezolid in crystalline form and salts thereof |
CN102643245A (zh) * | 2012-04-10 | 2012-08-22 | 杭州华东医药集团生物工程研究所有限公司 | 一种利奈唑胺晶型及其制备方法 |
ES2603252T3 (es) | 2012-11-09 | 2017-02-24 | Synthon Bv | Proceso para preparar linezolid |
JP7251813B2 (ja) * | 2017-11-16 | 2023-04-04 | ペルシカ ファーマシューティカルズ リミテッド | リネゾリド製剤 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
US5688792A (en) * | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
MY115155A (en) * | 1993-09-09 | 2003-04-30 | Upjohn Co | Substituted oxazine and thiazine oxazolidinone antimicrobials. |
CN1167701C (zh) * | 1996-04-11 | 2004-09-22 | 法玛西雅厄普约翰美国公司 | 制备噁唑烷酮胺的方法 |
WO1999024393A1 (en) * | 1997-11-07 | 1999-05-20 | Pharmacia & Upjohn Company | Process to produce oxazolidinones |
-
2001
- 2001-01-22 AR ARP010100269A patent/AR027261A1/es not_active Application Discontinuation
- 2001-01-25 PE PE2001000080A patent/PE20011086A1/es not_active Application Discontinuation
- 2001-01-26 CO CO01005901A patent/CO5261555A1/es not_active Application Discontinuation
- 2001-01-29 AU AU32755/01A patent/AU782138B2/en not_active Ceased
- 2001-01-29 KR KR1020077016678A patent/KR100864745B1/ko not_active IP Right Cessation
- 2001-01-29 MY MYPI20010371A patent/MY122829A/en unknown
- 2001-01-29 IL IL15101001A patent/IL151010A0/xx active IP Right Grant
- 2001-01-29 CA CA2395603A patent/CA2395603C/en not_active Expired - Lifetime
- 2001-01-29 EE EEP200200420A patent/EE05197B1/et not_active IP Right Cessation
- 2001-01-29 CN CNB018034489A patent/CN1221547C/zh not_active Expired - Fee Related
- 2001-01-29 MX MXPA02007471A patent/MXPA02007471A/es active IP Right Grant
- 2001-01-29 KR KR1020027009923A patent/KR100781815B1/ko not_active IP Right Cessation
- 2001-01-29 CZ CZ20022635A patent/CZ302292B6/cs not_active IP Right Cessation
- 2001-01-29 DE DE60111497T patent/DE60111497T2/de not_active Expired - Lifetime
- 2001-01-29 HU HU0301076A patent/HUP0301076A3/hu unknown
- 2001-01-29 SI SI200130405T patent/SI1255754T1/sl unknown
- 2001-01-29 WO PCT/US2001/000657 patent/WO2001057035A1/en active IP Right Grant
- 2001-01-29 NZ NZ520541A patent/NZ520541A/en not_active IP Right Cessation
- 2001-01-29 JP JP2001557867A patent/JP5235256B2/ja not_active Expired - Lifetime
- 2001-01-29 ES ES01904805T patent/ES2242728T3/es not_active Expired - Lifetime
- 2001-01-29 BR BR0107667-1A patent/BR0107667A/pt not_active Application Discontinuation
- 2001-01-29 PL PL01356433A patent/PL356433A1/xx unknown
- 2001-01-29 KR KR1020087010742A patent/KR20080044358A/ko not_active Application Discontinuation
- 2001-01-29 PT PT01904805T patent/PT1255754E/pt unknown
- 2001-01-29 EP EP01904805A patent/EP1255754B1/en not_active Expired - Lifetime
- 2001-01-29 EA EA200200819A patent/EA004434B1/ru not_active IP Right Cessation
- 2001-01-29 AT AT01904805T patent/ATE297920T1/de active
- 2001-01-29 SK SK994-2002A patent/SK287025B6/sk not_active IP Right Cessation
- 2001-01-29 DK DK01904805T patent/DK1255754T3/da active
- 2001-02-02 TW TW090102231A patent/TWI297687B/zh not_active IP Right Cessation
-
2002
- 2002-06-27 ZA ZA200205162A patent/ZA200205162B/en unknown
- 2002-08-01 NO NO20023654A patent/NO323459B1/no not_active IP Right Cessation
-
2003
- 2003-05-16 HK HK03103460A patent/HK1051196A1/xx not_active IP Right Cessation
-
2006
- 2006-12-15 NO NO20065836A patent/NO20065836L/no not_active Application Discontinuation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AA1Y | Spc filed |
Free format text: PRODUCT NAME: ZYVOX; REG NO/DATE: 00032/0259 05.01.2001 Spc suppl protection certif: C20100003 Filing date: 20100215 |
|
FC1Y | Spc application refused |
Free format text: PRODUCT NAME: ZYVOX; REG NO/DATE: 00032/0259 05.01.2001 Spc suppl protection certif: C20100003 Filing date: 20100215 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20101231 |
|
MM4A | Lapsed by not paying the annual fees |
Effective date: 20120129 |