KR100265529B1 - 고지혈증 치료에 유용한 벤조티아제핀 화합물 - Google Patents

고지혈증 치료에 유용한 벤조티아제핀 화합물 Download PDF

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Publication number
KR100265529B1
KR100265529B1 KR1019940702834A KR19940702834A KR100265529B1 KR 100265529 B1 KR100265529 B1 KR 100265529B1 KR 1019940702834 A KR1019940702834 A KR 1019940702834A KR 19940702834 A KR19940702834 A KR 19940702834A KR 100265529 B1 KR100265529 B1 KR 100265529B1
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KR
South Korea
Prior art keywords
compound
formula
ethyl
integer
benzothiazepine
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Expired - Fee Related
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KR1019940702834A
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English (en)
Korean (ko)
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KR950700265A (ko
Inventor
로렌스 에드워드 브라이어디
Original Assignee
그레이엄 브레레톤
더 웰컴 파운데이션 리미티드
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Publication of KR950700265A publication Critical patent/KR950700265A/ko
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Publication of KR100265529B1 publication Critical patent/KR100265529B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Steroid Compounds (AREA)
KR1019940702834A 1992-02-17 1993-02-16 고지혈증 치료에 유용한 벤조티아제핀 화합물 Expired - Fee Related KR100265529B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB929203347A GB9203347D0 (en) 1992-02-17 1992-02-17 Hypolipidaemic compounds
GB9203347.1 1992-02-17
PCT/GB1993/000328 WO1993016055A1 (en) 1992-02-17 1993-02-16 Hypolipidaemic benzothiazepine compounds

Publications (2)

Publication Number Publication Date
KR950700265A KR950700265A (ko) 1995-01-16
KR100265529B1 true KR100265529B1 (ko) 2000-11-01

Family

ID=10710542

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019940702834A Expired - Fee Related KR100265529B1 (ko) 1992-02-17 1993-02-16 고지혈증 치료에 유용한 벤조티아제핀 화합물

Country Status (21)

Country Link
US (2) US5663165A (enExample)
EP (1) EP0626952B1 (enExample)
JP (1) JP2904926B2 (enExample)
KR (1) KR100265529B1 (enExample)
AT (1) ATE178897T1 (enExample)
AU (1) AU675419B2 (enExample)
CA (1) CA2117485A1 (enExample)
DE (1) DE69324479T2 (enExample)
DK (1) DK0626952T3 (enExample)
ES (1) ES2131106T3 (enExample)
FI (1) FI943775A7 (enExample)
GB (1) GB9203347D0 (enExample)
GR (1) GR3030491T3 (enExample)
HU (1) HUT71487A (enExample)
IL (1) IL104740A (enExample)
MX (1) MX9300821A (enExample)
MY (1) MY129970A (enExample)
NZ (1) NZ249189A (enExample)
TW (1) TW274547B (enExample)
WO (1) WO1993016055A1 (enExample)
ZA (1) ZA931073B (enExample)

Families Citing this family (126)

* Cited by examiner, † Cited by third party
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EP0626952A1 (en) 1994-12-07
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WO1993016055A1 (en) 1993-08-19
ES2131106T3 (es) 1999-07-16
AU675419B2 (en) 1997-02-06
US5859240A (en) 1999-01-12
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HU9402365D0 (en) 1994-10-28
HUT71487A (en) 1995-11-28
CA2117485A1 (en) 1993-08-19
IL104740A0 (en) 1993-06-10
KR950700265A (ko) 1995-01-16
JPH07503724A (ja) 1995-04-20
ZA931073B (en) 1994-08-16
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AU3508293A (en) 1993-09-03
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US5663165A (en) 1997-09-02
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FI943775L (fi) 1994-08-16
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TW274547B (enExample) 1996-04-21
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IL104740A (en) 1996-09-12
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ATE178897T1 (de) 1999-04-15
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