KR100242397B1 - 트리아졸 유도체와 그의 염,그들의 제조방법 및 그들을 함유한 항진균제 - Google Patents

트리아졸 유도체와 그의 염,그들의 제조방법 및 그들을 함유한 항진균제 Download PDF

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KR100242397B1
KR100242397B1 KR1019920023597A KR920023597A KR100242397B1 KR 100242397 B1 KR100242397 B1 KR 100242397B1 KR 1019920023597 A KR1019920023597 A KR 1019920023597A KR 920023597 A KR920023597 A KR 920023597A KR 100242397 B1 KR100242397 B1 KR 100242397B1
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South Korea
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substituted
unsubstituted
alkyl
phenyl
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Korean (ko)
Inventor
히로유끼 이마이즈미
데쯔야 가지따
겐니찌 다까시마
미나꼬 요쯔지
게이꼬 다까꾸라
아끼라 요쯔지
쥬니찌 미쯔야마
가쯔미 시미즈
히로시 사까이
히로까즈 나리따
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나카노 가쓰히코
도야마 가가쿠 고교 가부시키가이샤
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1019920023597A 1991-12-09 1992-12-08 트리아졸 유도체와 그의 염,그들의 제조방법 및 그들을 함유한 항진균제 Expired - Fee Related KR100242397B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP91-350318 1991-12-09
JP35031891 1991-12-09
JP92-293961 1992-10-08
JP29396192A JP3471831B2 (ja) 1991-12-09 1992-10-08 新規なトリアゾール誘導体およびその塩

Publications (1)

Publication Number Publication Date
KR100242397B1 true KR100242397B1 (ko) 2000-03-02

Family

ID=26559630

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019920023597A Expired - Fee Related KR100242397B1 (ko) 1991-12-09 1992-12-08 트리아졸 유도체와 그의 염,그들의 제조방법 및 그들을 함유한 항진균제

Country Status (7)

Country Link
US (2) US5366989A (https=)
EP (1) EP0546529A1 (https=)
JP (1) JP3471831B2 (https=)
KR (1) KR100242397B1 (https=)
AU (1) AU655089B2 (https=)
CA (1) CA2084334A1 (https=)
TW (1) TW225476B (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3471831B2 (ja) * 1991-12-09 2003-12-02 富山化学工業株式会社 新規なトリアゾール誘導体およびその塩
ES2062941B1 (es) * 1993-03-15 1995-10-01 Uriach & Cia Sa J Nuevos derivados de azol activos por via oral.
ES2159676T3 (es) * 1995-12-22 2001-10-16 Ss Pharmaceutical Co Derivados de triazol con actividad antimicotica e intermediarios.
US6002028A (en) * 1995-12-22 1999-12-14 Ss Pharmaceutical Co., Ltd. Triazole derivative, preparation process thereof and pharmaceutical comprising the same as an effective ingredient
US5939448A (en) * 1996-06-21 1999-08-17 Ss Pharmaceutical Co., Ltd. Triazole derivative or salt thereof
US5965188A (en) * 1996-07-31 1999-10-12 Anitox Corporation Anti-bacterial amine derivatives
DK1399402T3 (da) * 2001-06-26 2010-11-15 Basilea Pharmaceutica Ag Intermediære halophenylderivater og deres anvendelse i en fremgangsmåde til fremstilling af azolderivater
JP2006182765A (ja) * 2004-11-30 2006-07-13 Sumitomo Chemical Co Ltd エポキシトリアゾール誘導体の製造方法
WO2006059759A1 (ja) * 2004-11-30 2006-06-08 Sumitomo Chemical Company, Limited エポキシトリアゾール誘導体の製造方法
EP2440518B1 (de) * 2009-06-08 2014-08-20 Bayer Cropscience AG Verfahren zur herstellung von fluoralkylnitrilen
US20150246898A1 (en) * 2012-09-12 2015-09-03 Dow Agrosciences Llc Metalloenzyme inhibitor compounds
CN102993052B (zh) * 2012-12-29 2014-07-09 吉首大学 芳基丙酰氧肟酸类尿素酶抑制剂及其合成和用途
CN103012207B (zh) * 2012-12-29 2015-05-27 吉首大学 二芳基丙酰-n-甲基氧肟酸类尿素酶抑制剂及其合成和用途
WO2023243700A1 (ja) * 2022-06-17 2023-12-21 シンクレスト株式会社 ジフルオロアルデヒド、エポキシ及びその誘導体

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4616027A (en) * 1982-08-14 1986-10-07 Pfizer Inc. Antifungal 1-aryl-1-fluoroalkyl-2-(1H-1,2,4-triazol-1-yl)ethanols
PH19347A (en) * 1982-09-30 1986-04-02 Pfizer Triazole derivatives,pharmaceutical composition containing same and method of use thereof
DE3378764D1 (en) * 1982-09-30 1989-02-02 Pfizer Ltd Triazole anti-fungal agents
GB8312624D0 (en) * 1983-05-07 1983-06-08 Pfizer Ltd Triazole antifungal agents
BG48681A3 (bg) * 1982-12-14 1991-04-15 Ciba - Geigy Ag Фунгицидно средство
DE3461637D1 (en) * 1983-02-16 1987-01-22 Pfizer Ltd Triazole antifungal agents
GB8304282D0 (en) * 1983-02-16 1983-03-23 Pfizer Ltd Antifungal agents
GB8305377D0 (en) 1983-02-25 1983-03-30 Pfizer Ltd Antifungal agents
US4518604A (en) * 1983-07-25 1985-05-21 Pfizer Inc. Antifungal 1-aryl-2-(1H-1,2,4-triazol-1yl)-1-perfluoroalkylethyl halides
GB8322983D0 (en) * 1983-08-26 1983-09-28 Pfizer Ltd Triazole antifungal agents
GB8601952D0 (en) * 1986-01-28 1986-03-05 Ici Plc Heterocyclic compounds
DE3736773A1 (de) * 1987-10-30 1989-05-11 Bayer Ag 3-(4-chlorphenyl)-2,2-dimethyl-3-hydroxy-4- (1,2,4-triazol-1-yl)-butyronitril
KR910700237A (ko) * 1989-01-23 1991-03-14 리챠드 지. 워터맨 치환된 트리아졸, 그의 제조방법 및 살진균제로서 사용하기 위한 조성물
DE59108565D1 (de) * 1990-08-09 1997-04-03 Bayer Ag Halogenalkyl-azolyl-Derivate
JP3471831B2 (ja) * 1991-12-09 2003-12-02 富山化学工業株式会社 新規なトリアゾール誘導体およびその塩

Also Published As

Publication number Publication date
AU2985892A (en) 1993-07-01
JP3471831B2 (ja) 2003-12-02
CA2084334A1 (en) 1993-06-10
TW225476B (https=) 1994-06-21
EP0546529A1 (en) 1993-06-16
JPH05213906A (ja) 1993-08-24
US5366989A (en) 1994-11-22
US5605921A (en) 1997-02-25
AU655089B2 (en) 1994-12-01

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