KE3078A - 3-amino-indazoecarboxylic acid derivatives,process for their preparation and their use as medicaments - Google Patents

3-amino-indazoecarboxylic acid derivatives,process for their preparation and their use as medicaments

Info

Publication number
KE3078A
KE3078A KE3078A KE307880A KE3078A KE 3078 A KE3078 A KE 3078A KE 3078 A KE3078 A KE 3078A KE 307880 A KE307880 A KE 307880A KE 3078 A KE3078 A KE 3078A
Authority
KE
Kenya
Prior art keywords
indazoecarboxylic
medicaments
amino
preparation
acid derivatives
Prior art date
Application number
KE3078A
Other languages
English (en)
Inventor
K H Mayer
W Wuttke
E Klauke
S Petersen
F Hoffmeister
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of KE3078A publication Critical patent/KE3078A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
KE3078A 1974-12-13 1980-08-29 3-amino-indazoecarboxylic acid derivatives,process for their preparation and their use as medicaments KE3078A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
KE3078A true KE3078A (en) 1980-10-03

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
KE3078A KE3078A (en) 1974-12-13 1980-08-29 3-amino-indazoecarboxylic acid derivatives,process for their preparation and their use as medicaments

Country Status (27)

Country Link
US (1) US4051252A (de)
JP (1) JPS5182266A (de)
AT (1) AT343653B (de)
BE (1) BE836528A (de)
CA (1) CA1059523A (de)
CH (1) CH622250A5 (de)
CS (1) CS189731B2 (de)
DD (1) DD125484A5 (de)
DE (1) DE2458965C3 (de)
DK (1) DK137082C (de)
ES (1) ES443429A1 (de)
FI (1) FI753493A (de)
FR (1) FR2293928A1 (de)
GB (1) GB1490306A (de)
HK (1) HK52580A (de)
HU (1) HU173557B (de)
IE (1) IE42208B1 (de)
IL (1) IL48642A (de)
KE (1) KE3078A (de)
LU (1) LU73993A1 (de)
NL (1) NL7514521A (de)
NO (1) NO145382C (de)
PL (1) PL99858B1 (de)
SE (1) SE419645B (de)
SU (1) SU604487A3 (de)
YU (1) YU315275A (de)
ZA (1) ZA757777B (de)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
CN1926132B (zh) * 2000-09-15 2010-12-29 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡唑化合物
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
AU2001292670A1 (en) 2000-09-15 2002-03-26 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
MXPA03005606A (es) 2000-12-21 2003-10-06 Vertex Pharma Compuestos de pirazol utiles como inhibidores de la proteina cinasa.
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
ES2380054T3 (es) 2001-09-26 2012-05-08 Pfizer Italia S.R.L. Derivados de aminoindazol activos como inhibidores de quinasas, procedimientos para su preparación, y composiciones farmacéuticas que los contienen
PL372198A1 (en) * 2002-02-06 2005-07-11 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
ATE468336T1 (de) 2002-03-15 2010-06-15 Vertex Pharma Azolylaminoazine als proteinkinasehemmer
MXPA04011417A (es) 2002-05-17 2005-02-14 Pharmacia Italia Spa Derivados de aminoindazol activos como inhibidores de cinasa, procedimiento para su preparacion y composiciones farmaceuticas que los comprenden.
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
DK1532145T3 (da) 2002-08-02 2007-01-15 Vertex Pharma Pyrazolpræparater der er anvendelige som inhibitorer af GSK-3
WO2004041285A1 (en) * 2002-10-31 2004-05-21 Amgen Inc. Antiinflammation agents
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
US7592340B2 (en) * 2003-12-04 2009-09-22 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
US7737151B2 (en) 2005-08-18 2010-06-15 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
SG166827A1 (en) 2005-11-03 2010-12-29 Vertex Pharma Aminopyrimidines useful as kinase inhibitors
CA2647261A1 (en) * 2006-04-14 2007-10-25 Abbott Laboratories Process for the preparation of indazolyl ureas that inhibit vanilloid subtype 1 (vr1) receptors
CA2668429A1 (en) 2006-11-02 2008-05-15 Vertex Pharmaceuticals Incorporated Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
MX2009006690A (es) 2006-12-19 2009-07-31 Vertex Pharma Aminopirimidinas utiles como inhibidores de proteinas cinasas.
MX2009009592A (es) 2007-03-09 2009-11-10 Vertex Pharma Aminopiridinas utiles como inhibidores de proteinas cinasas.
MX2009009590A (es) 2007-03-09 2009-11-10 Vertex Pharma Aminopirimidinas utiles como inhibidores de proteinas cinasas.
MX2009009591A (es) 2007-03-09 2009-11-10 Vertex Pharma Aminopirimidinas utiles como inhibidores de proteinas cinasas.
CA2683785A1 (en) 2007-04-13 2008-10-23 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
AU2008247594A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
MX2009011810A (es) * 2007-05-02 2010-01-14 Vertex Pharma Tiazoles y pirazoles utiles como inhibidores de cinasa.
MX2009011811A (es) * 2007-05-02 2010-01-14 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasa.
JP2010528021A (ja) * 2007-05-24 2010-08-19 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼのインヒビターとして有用なチアゾールおよびピラゾール
EP2176261B1 (de) * 2007-07-31 2012-12-19 Vertex Pharmaceuticals Incorporated Verfahren für die zubereitung von 5-fluor-1h-pyrazolo [3, 4-b] pyridin-3-amin und derivaten davon
JP2012501971A (ja) * 2008-09-03 2012-01-26 バーテックス ファーマシューティカルズ インコーポレイテッド 共結晶および共結晶を含む薬学的処方物
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
HUE037085T2 (hu) 2012-07-24 2018-08-28 Bial Portela & Ca Sa Karbamid vegyületek és enzim-inhibitorként történõ alkalmazásuk
CN104662002A (zh) * 2012-07-27 2015-05-27 比亚尔-珀特拉和Ca股份公司 取代脲类化合物的合成方法
DK3024825T3 (en) 2013-07-24 2017-10-02 BIAL - PORTELA & Cª S A IMIDAZOLE CARBOXAMIDES AND THEIR USE AS FAAH INHIBITORS

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3274203A (en) * 1963-05-31 1966-09-20 Du Pont 1-carbamyl and thiocarbamyl-3-amino-4-nonsubstituted and substituted pyrazoles
NL6707299A (de) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
HU173557B (hu) 1979-06-28
SE7513990L (sv) 1976-06-14
SE419645B (sv) 1981-08-17
PL99858B1 (pl) 1978-08-31
ATA939775A (de) 1977-10-15
AU8717075A (en) 1977-06-09
BE836528A (fr) 1976-06-11
JPS5182266A (en) 1976-07-19
LU73993A1 (de) 1976-11-11
FR2293928A1 (fr) 1976-07-09
NO754024L (de) 1976-06-15
US4051252A (en) 1977-09-27
DK567275A (da) 1976-06-14
NO145382B (no) 1981-11-30
SU604487A3 (ru) 1978-04-25
DE2458965C3 (de) 1979-10-11
DE2458965B2 (de) 1979-02-22
NO145382C (no) 1982-03-10
CS189731B2 (en) 1979-04-30
AT343653B (de) 1978-06-12
IL48642A (en) 1979-12-30
HK52580A (en) 1980-09-26
DK137082C (da) 1978-06-19
IE42208L (en) 1976-06-13
IL48642A0 (en) 1976-02-29
FI753493A (de) 1976-06-14
CA1059523A (en) 1979-07-31
YU315275A (en) 1982-02-28
DK137082B (da) 1978-01-16
GB1490306A (en) 1977-11-02
NL7514521A (nl) 1976-06-15
DE2458965A1 (de) 1976-06-16
IE42208B1 (en) 1980-06-18
ZA757777B (en) 1976-11-24
CH622250A5 (de) 1981-03-31
FR2293928B1 (de) 1979-09-21
ES443429A1 (es) 1977-04-16
DD125484A5 (de) 1977-04-20

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