JPWO2023195530A5 - - Google Patents
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- Publication number
- JPWO2023195530A5 JPWO2023195530A5 JP2023560418A JP2023560418A JPWO2023195530A5 JP WO2023195530 A5 JPWO2023195530 A5 JP WO2023195530A5 JP 2023560418 A JP2023560418 A JP 2023560418A JP 2023560418 A JP2023560418 A JP 2023560418A JP WO2023195530 A5 JPWO2023195530 A5 JP WO2023195530A5
- Authority
- JP
- Japan
- Prior art keywords
- pharma
- acceptable salt
- compound according
- ceutically acceptable
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022064593 | 2022-04-08 | ||
| JP2022064593 | 2022-04-08 | ||
| JP2022094627 | 2022-06-10 | ||
| JP2022094627 | 2022-06-10 | ||
| JP2022207187 | 2022-12-23 | ||
| JP2022207187 | 2022-12-23 | ||
| PCT/JP2023/014318 WO2023195530A1 (ja) | 2022-04-08 | 2023-04-07 | ウイルス増殖阻害活性を有するウラシル誘導体およびそれらを含有する医薬組成物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2023195530A1 JPWO2023195530A1 (https=) | 2023-10-12 |
| JPWO2023195530A5 true JPWO2023195530A5 (https=) | 2025-01-14 |
| JP7624093B2 JP7624093B2 (ja) | 2025-01-29 |
Family
ID=88243017
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023560418A Active JP7624093B2 (ja) | 2022-04-08 | 2023-04-07 | ウイルス増殖阻害活性を有するウラシル誘導体およびそれらを含有する医薬組成物 |
| JP2023560417A Pending JPWO2023195529A1 (https=) | 2022-04-08 | 2023-04-07 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023560417A Pending JPWO2023195529A1 (https=) | 2022-04-08 | 2023-04-07 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US12545687B2 (https=) |
| EP (1) | EP4506342A1 (https=) |
| JP (2) | JP7624093B2 (https=) |
| KR (1) | KR20250004704A (https=) |
| CN (1) | CN117510472B (https=) |
| AU (1) | AU2023249953A1 (https=) |
| CA (1) | CA3246981A1 (https=) |
| CO (1) | CO2024013781A2 (https=) |
| IL (1) | IL315710A (https=) |
| MX (1) | MX2024012320A (https=) |
| TW (1) | TW202345801A (https=) |
| WO (2) | WO2023195529A1 (https=) |
| ZA (1) | ZA202407589B (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP7624093B2 (ja) * | 2022-04-08 | 2025-01-29 | 塩野義製薬株式会社 | ウイルス増殖阻害活性を有するウラシル誘導体およびそれらを含有する医薬組成物 |
| WO2024031089A1 (en) | 2022-08-05 | 2024-02-08 | Gilead Sciences, Inc. | Sars-cov2 main protease inhibitors |
| WO2025074997A1 (ja) * | 2023-10-02 | 2025-04-10 | 塩野義製薬株式会社 | ウイルス増殖阻害活性を有する縮合複素環誘導体およびそれらを含有する医薬組成物 |
| AU2024307335A1 (en) * | 2023-10-05 | 2026-04-16 | Shionogi & Co., Ltd. | Pharmaceutical composition containing uracil derivative |
| AU2024309726A1 (en) * | 2023-10-05 | 2026-04-16 | Shionogi & Co., Ltd. | Preparation containing uracil derivative |
| WO2025018428A2 (ja) * | 2023-10-05 | 2025-01-23 | 塩野義製薬株式会社 | ウラシル誘導体の製造方法 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7550480B2 (en) * | 2003-02-14 | 2009-06-23 | Smithkline Beecham Corporation | Compounds |
| UA85871C2 (uk) | 2004-03-15 | 2009-03-10 | Такеда Фармасьютікал Компані Лімітед | Інгібітори дипептидилпептидази |
| CN100502868C (zh) * | 2005-11-18 | 2009-06-24 | 北京大学 | 非肽类sars冠状病毒3cl蛋白酶抑制剂及其用途 |
| KR20110089463A (ko) | 2006-07-24 | 2011-08-08 | 한국화학연구원 | 신규 hiv 역전사 효소 억제제 |
| ES2533863T3 (es) | 2007-06-29 | 2015-04-15 | Korea Research Institute Of Chemical Technology | Inhibidores novedosos de la transcriptasa inversa de VIH |
| JP6075621B2 (ja) | 2010-08-10 | 2017-02-08 | 塩野義製薬株式会社 | 新規複素環誘導体およびそれらを含有する医薬組成物 |
| WO2013118855A1 (ja) * | 2012-02-09 | 2013-08-15 | 塩野義製薬株式会社 | 複素環および炭素環誘導体 |
| CN115515593A (zh) * | 2020-02-17 | 2022-12-23 | 勒芬天主教大学 | 作为药物的新的6-取代的7-脱氮嘌呤和相应的核苷 |
| PH12021552872A1 (en) | 2020-04-05 | 2022-03-21 | Pfizer | Compounds and methods for the treatment of covid-19 |
| CN113801187A (zh) * | 2020-06-12 | 2021-12-17 | 南开大学 | 靶向新型冠状病毒的迈克尔受体类主蛋白酶抑制剂的制备及用途 |
| US11351149B2 (en) | 2020-09-03 | 2022-06-07 | Pfizer Inc. | Nitrile-containing antiviral compounds |
| LT4122926T (lt) | 2021-04-14 | 2025-07-25 | Shionogi & Co., Ltd. | Triazino dariniai, turintys virusų replikaciją slopinantį poveikį, ir juos apimanti farmacinė kompozicija |
| WO2022224223A1 (en) | 2021-04-23 | 2022-10-27 | Novartis Ag | Compounds and compositions for the treatment of coronaviral related diseases |
| UY39863A (es) | 2021-07-22 | 2023-02-28 | Novartis Ag | Compuestos y composiciones para el tratamiento de enfermedades relacionadas con el coronavirus |
| CN113801097B (zh) | 2021-09-27 | 2022-11-22 | 成都施贝康生物医药科技有限公司 | 二氢嘧啶类化合物、其制备方法及用途 |
| CN113735838B (zh) | 2021-09-27 | 2022-07-08 | 成都施贝康生物医药科技有限公司 | 二氢嘧啶类化合物、其制备方法及用途 |
| CN113620888B (zh) * | 2021-09-27 | 2023-06-06 | 成都施贝康生物医药科技有限公司 | 二氢嘧啶类化合物及其制备方法和应用 |
| CN113666914B (zh) | 2021-09-27 | 2022-06-07 | 成都施贝康生物医药科技有限公司 | 二氢嘧啶类化合物及其制备方法和用途 |
| CN113773300B (zh) | 2021-09-27 | 2022-10-11 | 成都施贝康生物医药科技有限公司 | 磺酰胺类化合物、其制备方法及用途 |
| JP7624093B2 (ja) * | 2022-04-08 | 2025-01-29 | 塩野義製薬株式会社 | ウイルス増殖阻害活性を有するウラシル誘導体およびそれらを含有する医薬組成物 |
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2023
- 2023-04-07 JP JP2023560418A patent/JP7624093B2/ja active Active
- 2023-04-07 CN CN202311441304.7A patent/CN117510472B/zh active Active
- 2023-04-07 EP EP23784813.0A patent/EP4506342A1/en active Pending
- 2023-04-07 TW TW112113106A patent/TW202345801A/zh unknown
- 2023-04-07 IL IL315710A patent/IL315710A/en unknown
- 2023-04-07 WO PCT/JP2023/014316 patent/WO2023195529A1/ja not_active Ceased
- 2023-04-07 JP JP2023560417A patent/JPWO2023195529A1/ja active Pending
- 2023-04-07 US US18/554,130 patent/US12545687B2/en active Active
- 2023-04-07 WO PCT/JP2023/014318 patent/WO2023195530A1/ja not_active Ceased
- 2023-04-07 KR KR1020247036205A patent/KR20250004704A/ko active Pending
- 2023-04-07 AU AU2023249953A patent/AU2023249953A1/en active Pending
- 2023-04-07 CA CA3246981A patent/CA3246981A1/en active Pending
-
2024
- 2024-10-04 MX MX2024012320A patent/MX2024012320A/es unknown
- 2024-10-07 ZA ZA2024/07589A patent/ZA202407589B/en unknown
- 2024-10-11 CO CONC2024/0013781A patent/CO2024013781A2/es unknown