JP2019151627A5 - - Google Patents

Download PDF

Info

Publication number
JP2019151627A5
JP2019151627A5 JP2019035140A JP2019035140A JP2019151627A5 JP 2019151627 A5 JP2019151627 A5 JP 2019151627A5 JP 2019035140 A JP2019035140 A JP 2019035140A JP 2019035140 A JP2019035140 A JP 2019035140A JP 2019151627 A5 JP2019151627 A5 JP 2019151627A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
diabetes
acceptable salt
compound according
therapeutic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2019035140A
Other languages
English (en)
Japanese (ja)
Other versions
JP2019151627A (ja
JP7206132B2 (ja
Filing date
Publication date
Application filed filed Critical
Publication of JP2019151627A publication Critical patent/JP2019151627A/ja
Publication of JP2019151627A5 publication Critical patent/JP2019151627A5/ja
Priority to JP2023000037A priority Critical patent/JP2023026566A/ja
Application granted granted Critical
Publication of JP7206132B2 publication Critical patent/JP7206132B2/ja
Priority to JP2024214451A priority patent/JP2025026615A/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2019035140A 2018-03-01 2019-02-28 メチルラクタム環化合物及びその医薬用途 Active JP7206132B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2023000037A JP2023026566A (ja) 2018-03-01 2023-01-04 メチルラクタム環化合物及びその医薬用途
JP2024214451A JP2025026615A (ja) 2018-03-01 2024-12-09 メチルラクタム環化合物及びその医薬用途

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2018036307 2018-03-01
JP2018036307 2018-03-01

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023000037A Division JP2023026566A (ja) 2018-03-01 2023-01-04 メチルラクタム環化合物及びその医薬用途

Publications (3)

Publication Number Publication Date
JP2019151627A JP2019151627A (ja) 2019-09-12
JP2019151627A5 true JP2019151627A5 (https=) 2022-03-07
JP7206132B2 JP7206132B2 (ja) 2023-01-17

Family

ID=67806229

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2019035140A Active JP7206132B2 (ja) 2018-03-01 2019-02-28 メチルラクタム環化合物及びその医薬用途
JP2023000037A Pending JP2023026566A (ja) 2018-03-01 2023-01-04 メチルラクタム環化合物及びその医薬用途
JP2024214451A Pending JP2025026615A (ja) 2018-03-01 2024-12-09 メチルラクタム環化合物及びその医薬用途

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2023000037A Pending JP2023026566A (ja) 2018-03-01 2023-01-04 メチルラクタム環化合物及びその医薬用途
JP2024214451A Pending JP2025026615A (ja) 2018-03-01 2024-12-09 メチルラクタム環化合物及びその医薬用途

Country Status (21)

Country Link
US (3) US11014910B2 (https=)
EP (1) EP3760624A4 (https=)
JP (3) JP7206132B2 (https=)
KR (1) KR102795351B1 (https=)
CN (1) CN111757877B (https=)
AR (1) AR114418A1 (https=)
AU (1) AU2019227770B2 (https=)
BR (1) BR112020016788A2 (https=)
CA (1) CA3087859A1 (https=)
CL (1) CL2020002199A1 (https=)
IL (1) IL276311B2 (https=)
MA (1) MA52427A (https=)
MX (1) MX2020009070A (https=)
MY (1) MY205197A (https=)
PE (1) PE20210123A1 (https=)
PH (1) PH12020551340A1 (https=)
SA (1) SA520420037B1 (https=)
SG (1) SG11202007120UA (https=)
TW (1) TWI805699B (https=)
WO (1) WO2019168096A1 (https=)
ZA (1) ZA202004600B (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI805699B (zh) * 2018-03-01 2023-06-21 日商日本煙草產業股份有限公司 甲基內醯胺環化合物及其用途
EP3778593A4 (en) 2018-04-04 2021-12-22 Japan Tobacco Inc. HETEROARYL-SUBSTITUTED PYRAZOLE COMPOUND AND ITS MEDICAL USE
JP7760370B2 (ja) * 2019-09-04 2025-10-27 日本たばこ産業株式会社 慢性腎臓病の治療又は予防方法
US20230119894A1 (en) * 2019-09-04 2023-04-20 Japan Tobacco Inc. Therapeutic or prophylactic method for diabetes using combination medicine
CA3175131A1 (en) 2020-03-19 2021-09-23 Chihiro Okuma Treatment or prevention method for chronic heart failure

Family Cites Families (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3657282A (en) * 1969-01-23 1972-04-18 Merck & Co Inc Carboxyepoxyethyl-1-phosphonic acid and derivatives
FR2665898B1 (fr) 1990-08-20 1994-03-11 Sanofi Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
JPH04247081A (ja) 1991-02-01 1992-09-03 Takeda Chem Ind Ltd 5員複素環酸アミド類
FR2692575B1 (fr) 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
US7622471B2 (en) 2003-02-07 2009-11-24 Daiichi Pharmaceutical Co., Ltd. Pyrazole derivatives having a pyridazine and pyridine functionality
AU2004200420A1 (en) 2003-03-11 2004-09-30 Astellas Pharma Inc. Inhibitor of cyclooxygenase
JP2006182648A (ja) 2003-04-08 2006-07-13 Dai Ichi Seiyaku Co Ltd 7員複素環誘導体
WO2004110351A2 (en) 2003-05-14 2004-12-23 Anadys Pharmaceuticals, Inc. Heterocyclic compounds for treating hepatitis c virus
TW200526588A (en) 2003-11-17 2005-08-16 Smithkline Beecham Corp Chemical compounds
TW200526641A (en) 2003-12-26 2005-08-16 Daiichi Seiyaku Co Amidopyrazole derivatives
CN1980665A (zh) 2004-07-07 2007-06-13 默克公司 吡唑酰胺衍生物,包含这些化合物的组合物和使用方法
AU2005305675B2 (en) 2004-11-16 2012-12-13 Jazz Pharmaceuticals Operations Uk Limited New use for cannabinoid
JP2008007405A (ja) 2004-12-07 2008-01-17 Takeda Chem Ind Ltd カルボキサミド誘導体
JP4137956B2 (ja) * 2005-06-08 2008-08-20 日本たばこ産業株式会社 複素環化合物
KR100970294B1 (ko) 2005-06-08 2010-07-15 니뽄 다바코 산교 가부시키가이샤 복소환 화합물
ZA200800142B (en) * 2005-06-08 2009-05-27 Japan Tobacco Inc Heterocyclic compound
WO2007034279A2 (en) * 2005-09-19 2007-03-29 Pfizer Products Inc. C3a antagonists and pharmaceutical compositions thereof
WO2007098826A2 (en) 2006-01-18 2007-09-07 Siena Biotech S.P.A. Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof
EP2026798A1 (en) * 2006-04-27 2009-02-25 Solvay Pharmaceuticals GmbH Pharmaceutical compositions comprising cbx cannabinoid receptor modulators and potassium channel modulators
US20080027014A1 (en) 2006-07-28 2008-01-31 Tanabe Seiyaku Co., Ltd. Novel SGLT inhibitors
KR101450356B1 (ko) 2006-11-24 2014-10-15 에이씨 이뮨 에스.에이. 알츠하이머와 같은 아밀로이드 또는 아밀로이드-유사 단백질과 관련된 질환의 치료를 위한 n-(메틸)-1h-피라졸-3-아민, n-(메틸)-피리딘-2-아민 및 n-(메틸)-티아졸-2-아민 유도체
EP2121619A2 (en) 2006-11-24 2009-11-25 AC Immune S.A. Compounds for the treatment of diseases associated with amyloid or amyloid-like proteins
TW200901974A (en) 2007-01-16 2009-01-16 Wyeth Corp Compounds, compositions, and methods of making and using them
JP5583003B2 (ja) * 2007-04-02 2014-09-03 セラコス・インコーポレイテッド ベンジルグルコシド誘導体およびその用途
WO2009091813A1 (en) 2008-01-14 2009-07-23 Wyeth Compounds useful as alpha7 nicotinic acetylcholine receptor agonists
EP2349484A2 (en) 2008-07-15 2011-08-03 Novartis AG Heteroaryl derivatives as dgat1 inhibitors
CN102918034B (zh) 2010-03-30 2015-06-03 维颂公司 多取代芳族化合物作为凝血酶的抑制剂
AR087701A1 (es) * 2011-08-31 2014-04-09 Japan Tobacco Inc Derivados de pirazol con actividad inhibidora de sglt1
KR102727059B1 (ko) * 2015-02-16 2024-11-05 더 유니버서티 어브 퀸슬랜드 설포닐우레아와 관련 화합물 및 그 용도
CN109071454B (zh) * 2016-02-16 2023-02-17 昆士兰大学 磺酰脲和相关化合物及其用途
TWI805699B (zh) * 2018-03-01 2023-06-21 日商日本煙草產業股份有限公司 甲基內醯胺環化合物及其用途
EP3778593A4 (en) 2018-04-04 2021-12-22 Japan Tobacco Inc. HETEROARYL-SUBSTITUTED PYRAZOLE COMPOUND AND ITS MEDICAL USE

Similar Documents

Publication Publication Date Title
JP2019151627A5 (https=)
JP2019048894A5 (https=)
JP2020097577A5 (https=)
JP2021191784A5 (https=)
JP2024516371A5 (https=)
JP2013032389A5 (https=)
JP2015078230A5 (https=)
JP2013518107A5 (https=)
JP2012255026A5 (https=)
FI3256218T3 (fi) Kdm1a-estäjät sairauksien hoidossa
JP2017524735A5 (https=)
JP2016501221A5 (https=)
JP2011518833A5 (https=)
JP2011527299A5 (https=)
JP2015024998A5 (https=)
JP2006526031A5 (https=)
JP2016518337A5 (https=)
JP2013542247A5 (https=)
JP2013525444A5 (https=)
JP2015155440A5 (https=)
JP2017517565A5 (https=)
EP4663637A3 (en) Novel deuterium substituted positron emission tomography (pet) imaging agents and their pharmacological application
JP2014530818A5 (https=)
CN103717571B8 (zh) 9‑氨基甲基取代的四环素类化合物
JP2018145180A5 (https=)