JP2021522345A5 - - Google Patents

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Publication number
JP2021522345A5
JP2021522345A5 JP2021509963A JP2021509963A JP2021522345A5 JP 2021522345 A5 JP2021522345 A5 JP 2021522345A5 JP 2021509963 A JP2021509963 A JP 2021509963A JP 2021509963 A JP2021509963 A JP 2021509963A JP 2021522345 A5 JP2021522345 A5 JP 2021522345A5
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
cancer
subject
administering
Prior art date
Application number
JP2021509963A
Other languages
English (en)
Japanese (ja)
Other versions
JPWO2020033019A5 (https=
JP2021522345A (ja
JP7115671B2 (ja
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Priority claimed from PCT/US2019/029192 external-priority patent/WO2020033019A2/en
Publication of JP2021522345A publication Critical patent/JP2021522345A/ja
Publication of JPWO2020033019A5 publication Critical patent/JPWO2020033019A5/ja
Publication of JP2021522345A5 publication Critical patent/JP2021522345A5/ja
Application granted granted Critical
Publication of JP7115671B2 publication Critical patent/JP7115671B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021509963A 2018-04-25 2019-04-25 新規なmct4阻害剤及びその使用 Active JP7115671B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862662637P 2018-04-25 2018-04-25
US62/662,637 2018-04-25
PCT/US2019/029192 WO2020033019A2 (en) 2018-04-25 2019-04-25 Novel mct4 inhibitors and uses thereof

Publications (4)

Publication Number Publication Date
JP2021522345A JP2021522345A (ja) 2021-08-30
JPWO2020033019A5 JPWO2020033019A5 (https=) 2022-04-28
JP2021522345A5 true JP2021522345A5 (https=) 2022-04-28
JP7115671B2 JP7115671B2 (ja) 2022-08-09

Family

ID=68532786

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021509963A Active JP7115671B2 (ja) 2018-04-25 2019-04-25 新規なmct4阻害剤及びその使用

Country Status (7)

Country Link
US (1) US10919878B2 (https=)
EP (1) EP3784650B1 (https=)
JP (1) JP7115671B2 (https=)
CN (1) CN112888673B (https=)
AU (1) AU2019317518B2 (https=)
CA (1) CA3098189C (https=)
WO (1) WO2020033019A2 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12544375B2 (en) * 2019-09-05 2026-02-10 The Board Of Trustees Of The Leland Junior University Small molecule therapeutic for parkinson's disease paired with a biomarker of therapeutic activity
WO2021249969A1 (en) * 2020-06-10 2021-12-16 Merck Patent Gmbh Combination product for the treatment of cancer diseases
WO2022243573A1 (en) 2021-05-21 2022-11-24 Cemm - Forschungszentrum Für Molekulare Medizin Gmbh 1,2,4-triazolo[1,5-a]pyrimidine-based slc16a3 inhibitors and their therapeutic use
WO2022243574A1 (en) 2021-05-21 2022-11-24 Cemm - Forschungszentrum Für Molekulare Medizin Gmbh 3-(phthalazin-1-yl)benzenesulfonamide-based slc16a3 inhibitors and their therapeutic use

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1226438A (https=) 1968-12-03 1971-03-31
GB0327734D0 (en) * 2003-11-28 2003-12-31 Novartis Ag Organic compounds
TW200804349A (en) * 2005-12-23 2008-01-16 Kalypsys Inc Novel substituted pyrimidinyloxy ureas as inhibitors of protein kinases
WO2010089580A1 (en) * 2009-02-06 2010-08-12 Astrazeneca Ab Use of a mct1 inhibitor in the treatment of cancers expressing mct1 over mct4
CN102731413A (zh) * 2011-04-15 2012-10-17 上海医药工业研究院 一种脲类化合物、其制备方法、其中间体及其应用
CN105263484B (zh) 2013-05-24 2018-08-03 株式会社加龄.营养研究所 包含二甲双胍和二氢槲皮素的药物组合及其用于治疗癌症的用途
CN107406390B (zh) * 2014-11-17 2021-04-16 奈吉治疗公司 单羧酸转运蛋白调节剂及其用途
EP3247349B1 (en) * 2015-01-22 2019-12-11 The Scripps Research Institute Chromenone inhibitors of monocarboxylate transporters
US10328078B2 (en) * 2015-01-22 2019-06-25 The Scripps Research Institute Pteridine dione monocarboxylate transporter inhibitors
BR112017026535B1 (pt) * 2015-06-12 2023-12-19 Vettore, LLC Composto e composição farmacêutica
CN108368060B (zh) * 2017-12-21 2020-09-15 中国科学院合肥物质科学研究院 一类嘧啶类衍生物激酶抑制剂

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