JP2021530453A5 - - Google Patents

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Publication number
JP2021530453A5
JP2021530453A5 JP2020571855A JP2020571855A JP2021530453A5 JP 2021530453 A5 JP2021530453 A5 JP 2021530453A5 JP 2020571855 A JP2020571855 A JP 2020571855A JP 2020571855 A JP2020571855 A JP 2020571855A JP 2021530453 A5 JP2021530453 A5 JP 2021530453A5
Authority
JP
Japan
Prior art keywords
disease
pharmaceutically acceptable
pharmaceutical composition
stereoisomer
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020571855A
Other languages
English (en)
Japanese (ja)
Other versions
JP7328263B2 (ja
JP2021530453A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/039509 external-priority patent/WO2020006233A1/en
Publication of JP2021530453A publication Critical patent/JP2021530453A/ja
Publication of JP2021530453A5 publication Critical patent/JP2021530453A5/ja
Priority to JP2023126807A priority Critical patent/JP2023145694A/ja
Application granted granted Critical
Publication of JP7328263B2 publication Critical patent/JP7328263B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020571855A 2018-06-29 2019-06-27 免疫調節化合物 Active JP7328263B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023126807A JP2023145694A (ja) 2018-06-29 2023-08-03 免疫調節化合物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862692176P 2018-06-29 2018-06-29
US62/692,176 2018-06-29
PCT/US2019/039509 WO2020006233A1 (en) 2018-06-29 2019-06-27 Immunomodulatory compounds

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023126807A Division JP2023145694A (ja) 2018-06-29 2023-08-03 免疫調節化合物

Publications (3)

Publication Number Publication Date
JP2021530453A JP2021530453A (ja) 2021-11-11
JP2021530453A5 true JP2021530453A5 (https=) 2022-07-05
JP7328263B2 JP7328263B2 (ja) 2023-08-16

Family

ID=68987232

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020571855A Active JP7328263B2 (ja) 2018-06-29 2019-06-27 免疫調節化合物
JP2023126807A Pending JP2023145694A (ja) 2018-06-29 2023-08-03 免疫調節化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023126807A Pending JP2023145694A (ja) 2018-06-29 2023-08-03 免疫調節化合物

Country Status (8)

Country Link
US (1) US12234220B2 (https=)
EP (1) EP3814330A4 (https=)
JP (2) JP7328263B2 (https=)
KR (1) KR102834593B1 (https=)
CN (1) CN113166100A (https=)
AU (1) AU2019293235B2 (https=)
CA (1) CA3102212A1 (https=)
WO (1) WO2020006233A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN118108706A (zh) * 2017-09-04 2024-05-31 C4医药公司 戊二酰亚胺
EP3814330A4 (en) * 2018-06-29 2022-07-20 Dana-Farber Cancer Institute, Inc. Immunomodulatory compounds
WO2020210630A1 (en) 2019-04-12 2020-10-15 C4 Therapeutics, Inc. Tricyclic degraders of ikaros and aiolos
JP7852923B2 (ja) * 2019-11-27 2026-04-28 キャプター セラピューティクス エス.エー. セレブロンに結合するピペリジン-2,6-ジオン誘導体、及びその使用方法
PH12022551482A1 (en) 2019-12-18 2023-11-29 Novartis Ag 3-(5-methoxy-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof
WO2022255889A1 (en) * 2021-06-01 2022-12-08 Captor Therapeutics S.A. Compounds which bind to cereblon, and use thereof
WO2022254362A1 (en) 2021-06-03 2022-12-08 Novartis Ag 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and medical uses thereof
EP4584259A1 (en) 2022-09-09 2025-07-16 Innovo Therapeutics, Inc. Ck1alpha and dual ck1alpha / gspt1 degrading compounds
CN116655595A (zh) * 2023-06-05 2023-08-29 中国人民解放军军事科学院军事医学研究院 2,6-哌啶二酮衍生物及其制备和用途
WO2025063888A1 (en) 2023-09-19 2025-03-27 Kancure Pte. Ltd. Survivin-targeted compounds
WO2025179161A1 (en) 2024-02-21 2025-08-28 Innovo Therapeutics, Inc. Protein degrading compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5698579A (en) 1993-07-02 1997-12-16 Celgene Corporation Cyclic amides
WO2008007979A1 (en) * 2006-07-12 2008-01-17 Auckland Uniservices Limited (2,6-dioxo-3-piperinyl)amidobenzoic immunomodulatory and anti-cancer derivatives
BR112018068906A2 (pt) * 2016-03-16 2019-01-22 H. Lee Moffitt Cancer Center And Research Institute, Inc. composição, método, método de redução de risco, prevenção ou tratamento de um indivíduo que tem uma doença ou distúrbio autoimune, método de indução de degradação de uma proteína-alvo numa célula, método para reduzir o risco, prevenir ou tratar um estado da doença ou afecção num paciente em que a atividade proteica desregulada é responsável pelo referido estado da doença ou afecção, método para reduzir o risco, prevenir ou tratar câncer num indivíduo e método de tratamento de uma doença ou distúrbio genético num indivíduo
CN109790143A (zh) * 2016-05-10 2019-05-21 C4医药公司 用于靶蛋白降解的胺连接的c3-戊二酰亚胺降解决定子体
IL312367A (en) * 2017-01-31 2024-06-01 Arvinas Operations Inc Cereblon ligands and bifunctional compounds comprising the same
CN118108706A (zh) 2017-09-04 2024-05-31 C4医药公司 戊二酰亚胺
WO2019140387A1 (en) 2018-01-12 2019-07-18 Kymera Therapeutics, Inc. Crbn ligands and uses thereof
EP3814330A4 (en) * 2018-06-29 2022-07-20 Dana-Farber Cancer Institute, Inc. Immunomodulatory compounds

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