JPWO2020257571A5 - - Google Patents

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JPWO2020257571A5
JPWO2020257571A5 JP2021575993A JP2021575993A JPWO2020257571A5 JP WO2020257571 A5 JPWO2020257571 A5 JP WO2020257571A5 JP 2021575993 A JP2021575993 A JP 2021575993A JP 2021575993 A JP2021575993 A JP 2021575993A JP WO2020257571 A5 JPWO2020257571 A5 JP WO2020257571A5
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Japan
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formula
compound
contacting
pharmaceutical material
group
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JP2021575993A
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English (en)
Japanese (ja)
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JP2022537049A (ja
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Priority claimed from PCT/US2020/038622 external-priority patent/WO2020257571A1/en
Publication of JP2022537049A publication Critical patent/JP2022537049A/ja
Publication of JPWO2020257571A5 publication Critical patent/JPWO2020257571A5/ja
Priority to JP2024211105A priority Critical patent/JP2025032197A/ja
Pending legal-status Critical Current

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JP2021575993A 2019-06-21 2020-06-19 ベンペド酸の製造方法及びその組成物 Pending JP2022537049A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024211105A JP2025032197A (ja) 2019-06-21 2024-12-04 ベンペド酸を含む製薬材料、医薬製剤及び医薬組成物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962864873P 2019-06-21 2019-06-21
US62/864,873 2019-06-21
PCT/US2020/038622 WO2020257571A1 (en) 2019-06-21 2020-06-19 Methods of making bempedoic acid and compositions of the same

Related Child Applications (1)

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JP2024211105A Division JP2025032197A (ja) 2019-06-21 2024-12-04 ベンペド酸を含む製薬材料、医薬製剤及び医薬組成物

Publications (2)

Publication Number Publication Date
JP2022537049A JP2022537049A (ja) 2022-08-23
JPWO2020257571A5 true JPWO2020257571A5 (enExample) 2023-06-16

Family

ID=71528020

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2021575993A Pending JP2022537049A (ja) 2019-06-21 2020-06-19 ベンペド酸の製造方法及びその組成物
JP2021575994A Withdrawn JP2022536979A (ja) 2019-06-21 2020-06-19 塩形態のベンペド酸及びそれを使用する方法
JP2024211105A Pending JP2025032197A (ja) 2019-06-21 2024-12-04 ベンペド酸を含む製薬材料、医薬製剤及び医薬組成物

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2021575994A Withdrawn JP2022536979A (ja) 2019-06-21 2020-06-19 塩形態のベンペド酸及びそれを使用する方法
JP2024211105A Pending JP2025032197A (ja) 2019-06-21 2024-12-04 ベンペド酸を含む製薬材料、医薬製剤及び医薬組成物

Country Status (13)

Country Link
US (10) US12344578B2 (enExample)
EP (3) EP3986860A1 (enExample)
JP (3) JP2022537049A (enExample)
KR (3) KR20220024816A (enExample)
CN (3) CN112437766A (enExample)
AU (3) AU2020295503A1 (enExample)
BR (2) BR112021025928A2 (enExample)
CA (2) CA3144372A1 (enExample)
ES (1) ES3032779T3 (enExample)
HU (1) HUE072061T2 (enExample)
IL (3) IL288909A (enExample)
MX (2) MX2021015936A (enExample)
WO (2) WO2020257571A1 (enExample)

Families Citing this family (17)

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CA3144372A1 (en) 2019-06-21 2020-12-24 Esperion Therapeutics, Inc. Salt forms of bempedoic acid and methods for using the same
EP4038045A1 (en) 2019-10-03 2022-08-10 Synthon B.V. Crystalline forms of bempedoic acid
WO2021110929A1 (en) * 2019-12-06 2021-06-10 Synthon B.V. Crystalline forms of sodium salt of bempedoic acid
CN111559961A (zh) * 2020-05-26 2020-08-21 杭州科巢生物科技有限公司 一种贝派地酸晶型及其制备方法
WO2021255180A1 (en) * 2020-06-19 2021-12-23 Synthon B.V. Salts of bempedoic acid
CN112521282A (zh) * 2020-12-02 2021-03-19 苏州汉德创宏生化科技有限公司 一种贝派地酸中间体及其合成方法
WO2022149161A1 (en) * 2021-01-05 2022-07-14 Dr. Reddy's Laboratories Limited Process for preparation of bempedoic acid and its intermediates
US20240366625A1 (en) 2021-06-02 2024-11-07 Esperion Therapeutics, Inc. Compositions containing and therapies using bempedoic acid and tolvaptan
CN115504914B (zh) * 2021-06-23 2024-05-07 武汉武药科技有限公司 一种贝派地酸中间体的制备方法
CN114436837B (zh) * 2021-12-27 2024-02-20 甘李药业股份有限公司 一种贝派地酸中间体的纯化方法
WO2023187833A1 (en) * 2022-03-30 2023-10-05 Enaltec Labs Private Limited A novel salt of bempedoic acid
WO2024151311A1 (en) 2023-01-09 2024-07-18 Esperion Therapeutics, Inc. Methods of treatment using bempedoic acid
CN116589341A (zh) * 2023-04-14 2023-08-15 苏州汉德创宏生化科技有限公司 一种抗高血酯药物中间体的制备方法
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WO2025196155A1 (en) 2024-03-20 2025-09-25 Astrazeneca Ab Pcsk9 inhibitors and methods of use thereof
WO2025238159A1 (en) 2024-05-16 2025-11-20 Astrazeneca Ab Combination therapy comprising azd0780 and ezetimibe

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