JPWO2020033955A5 - - Google Patents

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Publication number
JPWO2020033955A5
JPWO2020033955A5 JP2021531626A JP2021531626A JPWO2020033955A5 JP WO2020033955 A5 JPWO2020033955 A5 JP WO2020033955A5 JP 2021531626 A JP2021531626 A JP 2021531626A JP 2021531626 A JP2021531626 A JP 2021531626A JP WO2020033955 A5 JPWO2020033955 A5 JP WO2020033955A5
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JP
Japan
Prior art keywords
alkyl
disease
cycloalkyl
formula
pruritus
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Pending
Application number
JP2021531626A
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English (en)
Japanese (ja)
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JP2021534244A (ja
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Priority claimed from PCT/US2019/046182 external-priority patent/WO2020033955A1/en
Publication of JP2021534244A publication Critical patent/JP2021534244A/ja
Publication of JPWO2020033955A5 publication Critical patent/JPWO2020033955A5/ja
Pending legal-status Critical Current

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JP2021531626A 2018-08-10 2019-08-12 ピロロピリミジンitk阻害剤 Pending JP2021534244A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862717400P 2018-08-10 2018-08-10
US62/717,400 2018-08-10
PCT/US2019/046182 WO2020033955A1 (en) 2018-08-10 2019-08-12 Pyrrolopyrimidine itk inhibitors

Publications (2)

Publication Number Publication Date
JP2021534244A JP2021534244A (ja) 2021-12-09
JPWO2020033955A5 true JPWO2020033955A5 (es) 2022-08-29

Family

ID=69405523

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021531626A Pending JP2021534244A (ja) 2018-08-10 2019-08-12 ピロロピリミジンitk阻害剤

Country Status (13)

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US (3) US11021482B2 (es)
EP (1) EP3833350A4 (es)
JP (1) JP2021534244A (es)
KR (1) KR20210044822A (es)
CN (1) CN112823005A (es)
AU (1) AU2019317625A1 (es)
BR (1) BR112021002479A2 (es)
CA (1) CA3109192A1 (es)
IL (1) IL280593A (es)
MX (1) MX2021001558A (es)
PH (1) PH12021550187A1 (es)
SG (1) SG11202100525SA (es)
WO (1) WO2020033955A1 (es)

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WO2023014049A1 (ko) * 2021-08-02 2023-02-09 한국화학연구원 신규한 피롤로 피리미딘 유도체 화합물, 이의 제조방법, 및 이를 유효성분으로 포함하는 대사성 간질환의 예방 또는 치료용 약학적 조성물
CN113571191A (zh) * 2021-08-31 2021-10-29 复旦大学附属中山医院 免疫检查点抑制剂相关mace发生风险的预测方法
WO2023110843A1 (en) * 2021-12-15 2023-06-22 Almirall, S.A. Heterobicyclic derivatives as itk inhibitors
WO2024102778A1 (en) * 2022-11-08 2024-05-16 Aclaris Therapeutics, Inc. Pyrrolopyrimidine compositions for treatment of itk mediated conditions

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