JPS5993096A - ５−フルオロ−２′−デオキシウリジン誘導体及びその製造法 - Google Patents

５−フルオロ−２′−デオキシウリジン誘導体及びその製造法

Info

Publication number
JPS5993096A
JPS5993096A JP57201847A JP20184782A JPS5993096A JP S5993096 A JPS5993096 A JP S5993096A JP 57201847 A JP57201847 A JP 57201847A JP 20184782 A JP20184782 A JP 20184782A JP S5993096 A JPS5993096 A JP S5993096A
Authority
JP
Japan
Prior art keywords
group
fluoro
deoxyuridine
mmole
phosphate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP57201847A
Other languages
English (en)
Japanese (ja)
Other versions
JPS635038B2 (esLanguage
Inventor
Kenzo Watanabe
兼三 渡辺
Yoshinori Kato
加藤　喜規
Masahiko Saito
斉藤　政彦
Takeo Oba
大場　丈夫
Hisashi Fukushima
福島　久
Takeshi Hara
健 原
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Teijin Ltd
Original Assignee
Teijin Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teijin Ltd filed Critical Teijin Ltd
Priority to JP57201847A priority Critical patent/JPS5993096A/ja
Publication of JPS5993096A publication Critical patent/JPS5993096A/ja
Publication of JPS635038B2 publication Critical patent/JPS635038B2/ja
Granted legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP57201847A 1982-11-19 1982-11-19 ５−フルオロ−２′−デオキシウリジン誘導体及びその製造法 Granted JPS5993096A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP57201847A JPS5993096A (ja) 1982-11-19 1982-11-19 ５−フルオロ−２′−デオキシウリジン誘導体及びその製造法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP57201847A JPS5993096A (ja) 1982-11-19 1982-11-19 ５−フルオロ−２′−デオキシウリジン誘導体及びその製造法

Publications (2)

Publication Number Publication Date
JPS5993096A true JPS5993096A (ja) 1984-05-29
JPS635038B2 JPS635038B2 (esLanguage) 1988-02-01

Family

ID=16447871

Family Applications (1)

Application Number Title Priority Date Filing Date
JP57201847A Granted JPS5993096A (ja) 1982-11-19 1982-11-19 ５−フルオロ−２′−デオキシウリジン誘導体及びその製造法

Country Status (1)

Country Link
JP (1) JPS5993096A (esLanguage)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4605645A (en) * 1981-12-09 1986-08-12 Teijin Limited 5-fluoro-2'-deoxyuridine derivatives and a process for the preparation thereof
US4684631A (en) * 1984-10-09 1987-08-04 Toyama Chemical Co., Ltd. Novel 5-fluoro-2-deoxyuridine derivatives and salts thereof, process for producing the same, and antitumor agents containing the same
US5032680A (en) * 1988-02-29 1991-07-16 Kuraray Co., Ltd. 2'-deoxy-5-fluorouridine derivatives
US5414077A (en) * 1990-02-20 1995-05-09 Gilead Sciences Non-nucleoside linkers for convenient attachment of labels to oligonucleotides using standard synthetic methods

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS52139082A (en) * 1976-05-07 1977-11-19 Mitsui Toatsu Chem Inc 5-fluorouridinephosphates
JPS5329938A (en) * 1976-08-27 1978-03-20 Mitsui Toatsu Chem Inc Carcinostatic agent
JPS57128699A (en) * 1981-02-03 1982-08-10 Tokyo Kinzoku Kogyo Kk 5-fluorouracil derivative and its medical composition
JPS5899499A (ja) * 1981-12-09 1983-06-13 Teijin Ltd ５−フルオロ−２′−デオキシウリジン誘導体を有効成分とする抗腫瘍剤
JPS58192899A (ja) * 1982-05-06 1983-11-10 Teijin Ltd ３′−アシル−５−フルオロ−２′−デオキシウリジン誘導体及びその製造法
JPS5970699A (ja) * 1982-10-13 1984-04-21 Teijin Ltd ５−フルオロ−２′−デオキシウリジン誘導体及びその製造法

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS52139082A (en) * 1976-05-07 1977-11-19 Mitsui Toatsu Chem Inc 5-fluorouridinephosphates
JPS5329938A (en) * 1976-08-27 1978-03-20 Mitsui Toatsu Chem Inc Carcinostatic agent
JPS57128699A (en) * 1981-02-03 1982-08-10 Tokyo Kinzoku Kogyo Kk 5-fluorouracil derivative and its medical composition
JPS5899499A (ja) * 1981-12-09 1983-06-13 Teijin Ltd ５−フルオロ−２′−デオキシウリジン誘導体を有効成分とする抗腫瘍剤
JPS58192899A (ja) * 1982-05-06 1983-11-10 Teijin Ltd ３′−アシル−５−フルオロ−２′−デオキシウリジン誘導体及びその製造法
JPS5970699A (ja) * 1982-10-13 1984-04-21 Teijin Ltd ５−フルオロ−２′−デオキシウリジン誘導体及びその製造法

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4605645A (en) * 1981-12-09 1986-08-12 Teijin Limited 5-fluoro-2'-deoxyuridine derivatives and a process for the preparation thereof
US4684631A (en) * 1984-10-09 1987-08-04 Toyama Chemical Co., Ltd. Novel 5-fluoro-2-deoxyuridine derivatives and salts thereof, process for producing the same, and antitumor agents containing the same
US4740503A (en) * 1984-10-09 1988-04-26 Toyama Chemical Co., Ltd. Novel 5-fluoro-2'-deoxyuridine derivatives and salts thereof, process for producing the same, and antitumor agents containing the same
US5032680A (en) * 1988-02-29 1991-07-16 Kuraray Co., Ltd. 2'-deoxy-5-fluorouridine derivatives
US5414077A (en) * 1990-02-20 1995-05-09 Gilead Sciences Non-nucleoside linkers for convenient attachment of labels to oligonucleotides using standard synthetic methods

Also Published As

Publication number Publication date
JPS635038B2 (esLanguage) 1988-02-01

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