JPH1129545A5 - - Google Patents
Info
- Publication number
- JPH1129545A5 JPH1129545A5 JP1997202756A JP20275697A JPH1129545A5 JP H1129545 A5 JPH1129545 A5 JP H1129545A5 JP 1997202756 A JP1997202756 A JP 1997202756A JP 20275697 A JP20275697 A JP 20275697A JP H1129545 A5 JPH1129545 A5 JP H1129545A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- aryl
- alkylaryl
- formula
- substituted aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE96112275:1 | 1996-07-30 | ||
| EP96112275A EP0837055A1 (en) | 1996-07-30 | 1996-07-30 | Substituted Indanylidineacetylguanidines, process for their preparation, their use as medicaments or diagnostic and medicaments containing them |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPH1129545A JPH1129545A (ja) | 1999-02-02 |
| JPH1129545A5 true JPH1129545A5 (cg-RX-API-DMAC7.html) | 2005-05-26 |
| JP4039589B2 JP4039589B2 (ja) | 2008-01-30 |
Family
ID=8223055
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP20275697A Expired - Fee Related JP4039589B2 (ja) | 1996-07-30 | 1997-07-29 | 置換インダニリジンアセチルグアニジン類、それらの製造方法、医薬または診断剤としてのそれらの使用およびそれらを含有する医薬 |
Country Status (29)
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20220042487A (ko) | 2008-12-31 | 2022-04-05 | 알데릭스, 인코포레이티드 | 체액 저류 또는 염 과부하와 연관된 장애 및 위장관 장애의 치료 시에 nhe-매개된 역수송을 억제하는 화합물 및 방법 |
| WO2018129556A1 (en) | 2017-01-09 | 2018-07-12 | Ardelyx, Inc. | Compounds and methods for inhibiting nhe-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders |
| GB0916163D0 (en) * | 2009-09-15 | 2009-10-28 | Shire Llc | Prodrugs of guanfacine |
| BR112015025805A2 (pt) | 2013-04-12 | 2017-07-25 | Ardelyx Inc | compostos de ligação de nh3 e métodos para inibir o transporte de fosfato |
| WO2018129552A1 (en) | 2017-01-09 | 2018-07-12 | Ardelyx, Inc. | Compounds useful for treating gastrointestinal tract disorders |
| BR112019013963A2 (pt) | 2017-01-09 | 2020-04-28 | Ardelyx Inc | inibidores de antiporte mediado por nhe |
| CN114340631A (zh) | 2019-05-21 | 2022-04-12 | 阿德利克斯股份有限公司 | 用于降低患者的血清磷酸盐的组合 |
| CN116492469A (zh) * | 2023-05-22 | 2023-07-28 | 遵义医科大学附属医院 | 一种通道阻滞剂在制备治疗和/或预防肝纤维疾病药物中的应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3929582A1 (de) * | 1989-09-06 | 1991-03-07 | Hoechst Ag | Benzoylguanidine, verfahren zu ihrer herstellung, ihre verwendung als medikament sowie sie enthaltendes medikament |
| DE4421536A1 (de) * | 1994-06-20 | 1995-12-21 | Hoechst Ag | Perfluoralkylgruppen tragende phenylsubstituierte Alkenylcarbonsäure-guanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| SI0738712T1 (en) * | 1995-04-18 | 1999-12-31 | Hoechst Aktiengesellschaft | Anti-arrhythmic and cardioprotective substituted indenoylguanidines |
-
1996
- 1996-07-30 EP EP96112275A patent/EP0837055A1/en not_active Withdrawn
-
1997
- 1997-05-23 TW TW086106928A patent/TW445251B/zh active
- 1997-07-14 ID IDP972422A patent/ID17565A/id unknown
- 1997-07-24 PT PT97112674T patent/PT822182E/pt unknown
- 1997-07-24 ES ES97112674T patent/ES2164283T3/es not_active Expired - Lifetime
- 1997-07-24 AT AT97112674T patent/ATE207888T1/de not_active IP Right Cessation
- 1997-07-24 DE DE69707777T patent/DE69707777T2/de not_active Expired - Lifetime
- 1997-07-24 EP EP97112674A patent/EP0822182B1/en not_active Expired - Lifetime
- 1997-07-24 DK DK97112674T patent/DK0822182T3/da active
- 1997-07-24 SI SI9730260T patent/SI0822182T1/xx unknown
- 1997-07-28 CN CN97114777A patent/CN1064351C/zh not_active Expired - Fee Related
- 1997-07-28 TR TR97/00704A patent/TR199700704A2/xx unknown
- 1997-07-28 AU AU31554/97A patent/AU715187B2/en not_active Ceased
- 1997-07-28 NZ NZ328440A patent/NZ328440A/en unknown
- 1997-07-28 SK SK1034-97A patent/SK282128B6/sk unknown
- 1997-07-28 CZ CZ972411A patent/CZ241197A3/cs unknown
- 1997-07-28 IL IL12140797A patent/IL121407A0/xx unknown
- 1997-07-28 US US08/901,099 patent/US5900436A/en not_active Expired - Lifetime
- 1997-07-28 KR KR1019970035527A patent/KR980009236A/ko not_active Ceased
- 1997-07-28 AR ARP970103414A patent/AR008095A1/es unknown
- 1997-07-29 NO NO973486A patent/NO308213B1/no not_active IP Right Cessation
- 1997-07-29 BR BR9704131A patent/BR9704131A/pt active Search and Examination
- 1997-07-29 ZA ZA9706735A patent/ZA976735B/xx unknown
- 1997-07-29 RU RU97113146/04A patent/RU2176638C2/ru not_active IP Right Cessation
- 1997-07-29 HR HR970424A patent/HRP970424B1/xx not_active IP Right Cessation
- 1997-07-29 CA CA002211982A patent/CA2211982C/en not_active Expired - Fee Related
- 1997-07-29 JP JP20275697A patent/JP4039589B2/ja not_active Expired - Fee Related
- 1997-07-29 HU HU9701316A patent/HUP9701316A3/hu unknown
- 1997-07-29 MX MX9705737A patent/MX9705737A/es not_active IP Right Cessation
- 1997-07-29 PL PL97321392A patent/PL321392A1/xx unknown
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