JPH0560479B2 - - Google Patents

Info

Publication number
JPH0560479B2
JPH0560479B2 JP24739285A JP24739285A JPH0560479B2 JP H0560479 B2 JPH0560479 B2 JP H0560479B2 JP 24739285 A JP24739285 A JP 24739285A JP 24739285 A JP24739285 A JP 24739285A JP H0560479 B2 JPH0560479 B2 JP H0560479B2
Authority
JP
Japan
Prior art keywords
formula
group
compound
ascamycin
amino acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP24739285A
Other languages
English (en)
Japanese (ja)
Other versions
JPS62108897A (ja
Inventor
Kyoshi Isono
Makoto Ubukata
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
RIKEN
Original Assignee
RIKEN
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by RIKEN filed Critical RIKEN
Priority to JP24739285A priority Critical patent/JPS62108897A/ja
Publication of JPS62108897A publication Critical patent/JPS62108897A/ja
Publication of JPH0560479B2 publication Critical patent/JPH0560479B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
JP24739285A 1985-11-05 1985-11-05 アスカマイシン誘導体及びその合成法並びに制癌剤 Granted JPS62108897A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP24739285A JPS62108897A (ja) 1985-11-05 1985-11-05 アスカマイシン誘導体及びその合成法並びに制癌剤

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP24739285A JPS62108897A (ja) 1985-11-05 1985-11-05 アスカマイシン誘導体及びその合成法並びに制癌剤

Publications (2)

Publication Number Publication Date
JPS62108897A JPS62108897A (ja) 1987-05-20
JPH0560479B2 true JPH0560479B2 (enExample) 1993-09-02

Family

ID=17162742

Family Applications (1)

Application Number Title Priority Date Filing Date
JP24739285A Granted JPS62108897A (ja) 1985-11-05 1985-11-05 アスカマイシン誘導体及びその合成法並びに制癌剤

Country Status (1)

Country Link
JP (1) JPS62108897A (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5824657A (en) * 1997-03-18 1998-10-20 Cubist Pharmaceuticals, Inc. Aminoacyl sulfamides for the treatment of hyperproliferative disorders
DE10340068A1 (de) * 2003-08-28 2005-03-24 TransMIT Gesellschaft für Technologietransfer mbH Substrate für die Inhibierung der Adenylierungsdomänen nicht-ribosomaler Peptidsynthetasen
EP1848718B1 (en) 2005-02-04 2012-08-01 Millennium Pharmaceuticals, Inc. Inhibitors of e1 activating enzymes
CN106008512B (zh) 2006-02-02 2019-03-12 千禧药品公司 E1活化酶抑制剂
CN102421780A (zh) 2009-05-14 2012-04-18 米伦纽姆医药公司 氨基磺酸((1s，2s，4r)-4-{4-[(1s)-2，3-二氢-1h-茚-1-基氨基]-7h-吡咯并[2，3-d]嘧啶-7-基}-2-羟基环戊基)甲酯盐酸盐

Also Published As

Publication number Publication date
JPS62108897A (ja) 1987-05-20

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