JP7061076B2 - アイバカフトール類似体を含有するケイ素原子 - Google Patents

アイバカフトール類似体を含有するケイ素原子 Download PDF

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JP7061076B2
JP7061076B2 JP2018552693A JP2018552693A JP7061076B2 JP 7061076 B2 JP7061076 B2 JP 7061076B2 JP 2018552693 A JP2018552693 A JP 2018552693A JP 2018552693 A JP2018552693 A JP 2018552693A JP 7061076 B2 JP7061076 B2 JP 7061076B2
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disease
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tert
cftr
compound
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JP2019513741A5 (enExample
JP2019513741A (ja
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ムノーズ，ベニート
パークス，ダニエル
バストス，セシリア，エム．
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プロテオステイシス セラピューティクス，インコーポレイテッド
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    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
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    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2018552693A 2016-04-07 2017-04-07 アイバカフトール類似体を含有するケイ素原子 Active JP7061076B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662319439P 2016-04-07 2016-04-07
US62/319,439 2016-04-07
PCT/US2017/026579 WO2017177124A1 (en) 2016-04-07 2017-04-07 Silicone atoms containing ivacaftor analogues

Publications (3)

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JP2019513741A JP2019513741A (ja) 2019-05-30
JP2019513741A5 JP2019513741A5 (enExample) 2020-05-14
JP7061076B2 true JP7061076B2 (ja) 2022-04-27

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US (5) US10662207B2 (enExample)
EP (1) EP3440057B1 (enExample)
JP (1) JP7061076B2 (enExample)
KR (1) KR102448404B1 (enExample)
CN (1) CN109563047A (enExample)
AR (1) AR108203A1 (enExample)
AU (1) AU2017248253B2 (enExample)
BR (1) BR112018070747B1 (enExample)
CA (1) CA3019663C (enExample)
IL (1) IL262030B (enExample)
MA (1) MA43775A (enExample)
MX (1) MX386698B (enExample)
NZ (1) NZ746793A (enExample)
SA (1) SA518400164B1 (enExample)
SG (1) SG11201808682XA (enExample)
WO (1) WO2017177124A1 (enExample)

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WO2017177124A1 (en) 2016-04-07 2017-10-12 Proteostasis Therapeutics, Inc. Silicone atoms containing ivacaftor analogues
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CN109663129B (zh) * 2019-02-27 2021-05-11 四川大学华西第二医院 扩张型心肌病治疗药物及其应用
TWI848092B (zh) 2019-04-03 2024-07-11 美商維泰克斯製藥公司 囊腫纖維化跨膜傳導調節蛋白調節劑
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TWI899097B (zh) 2019-08-14 2025-10-01 美商維泰克斯製藥公司 製備cftr調節劑之方法
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