JP5960688B2 - プロテインキナーゼ調節物質としての新規3,5−二置換−3h−[1,2,3]トリアゾロ[4,5−b]ピリジン化合物 - Google Patents

プロテインキナーゼ調節物質としての新規3,5−二置換−3h−[1,2,3]トリアゾロ[4,5−b]ピリジン化合物 Download PDF

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JP5960688B2
JP5960688B2 JP2013510708A JP2013510708A JP5960688B2 JP 5960688 B2 JP5960688 B2 JP 5960688B2 JP 2013510708 A JP2013510708 A JP 2013510708A JP 2013510708 A JP2013510708 A JP 2013510708A JP 5960688 B2 JP5960688 B2 JP 5960688B2
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triazolo
pyridin
ylmethyl
quinolin
benzamide
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JP2013529207A (ja
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ムスッパラニアッパン,メイヤッパン
ヴィスワナダ,スリカント
バブ,ゴヴィンダラジュル
ヴァッカランカ,スワループ,ケー.ヴィ.エス.
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インコゼン セラピューティクス プライベート リミテッド
インコゼン セラピューティクス プライベート リミテッド
リーゼン ファーマシューティカルズ エス.エー.
リーゼン ファーマシューティカルズ エス.エー.
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
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JP2013510708A 2010-05-17 2011-05-13 プロテインキナーゼ調節物質としての新規3,5−二置換−3h−[1,2,3]トリアゾロ[4,5−b]ピリジン化合物 Expired - Fee Related JP5960688B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN1377CH2010 2010-05-17
IN1377/CHE/2010 2010-05-17
PCT/IB2011/052120 WO2011145035A1 (en) 2010-05-17 2011-05-13 Novel 3,5-disubstitued-3h-imidazo[4,5-b]pyridine and 3,5- disubstitued -3h-[1,2,3]triazolo[4,5-b] pyridine compounds as modulators of protein kinases

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JP2016081792A Division JP6286472B2 (ja) 2010-05-17 2016-04-15 プロテインキナーゼ調節物質としての新規3,5−二置換−3h−イミダゾ[4,5−b]ピリジン化合物および3,5−二置換−3h−[1,2,3]トリアゾロ[4,5−b]ピリジン化合物

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JP2013529207A JP2013529207A (ja) 2013-07-18
JP5960688B2 true JP5960688B2 (ja) 2016-08-02

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JP2016081792A Expired - Fee Related JP6286472B2 (ja) 2010-05-17 2016-04-15 プロテインキナーゼ調節物質としての新規3,5−二置換−3h−イミダゾ[4,5−b]ピリジン化合物および3,5−二置換−3h−[1,2,3]トリアゾロ[4,5−b]ピリジン化合物

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US (5) US8481739B2 (cg-RX-API-DMAC7.html)
EP (2) EP2571878B1 (cg-RX-API-DMAC7.html)
JP (2) JP5960688B2 (cg-RX-API-DMAC7.html)
KR (1) KR101871436B1 (cg-RX-API-DMAC7.html)
CN (2) CN107674073B (cg-RX-API-DMAC7.html)
AU (2) AU2011254242B2 (cg-RX-API-DMAC7.html)
CA (2) CA3084173A1 (cg-RX-API-DMAC7.html)
DK (1) DK2571878T3 (cg-RX-API-DMAC7.html)
EA (2) EA201690998A1 (cg-RX-API-DMAC7.html)
ES (1) ES2715611T3 (cg-RX-API-DMAC7.html)
IL (2) IL222977A (cg-RX-API-DMAC7.html)
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Cited By (1)

* Cited by examiner, † Cited by third party
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JP2016164184A (ja) * 2010-05-17 2016-09-08 インコゼン セラピューティクス プライベート リミテッド プロテインキナーゼ調節物質としての新規3,5−二置換−3h−イミダゾ[4,5−b]ピリジン化合物および3,5−二置換−3h−[1,2,3]トリアゾロ[4,5−b]ピリジン化合物

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