JP5932642B2 - 多量体ペプチドコンジュゲートおよびその使用 - Google Patents

多量体ペプチドコンジュゲートおよびその使用 Download PDF

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JP5932642B2
JP5932642B2 JP2012518704A JP2012518704A JP5932642B2 JP 5932642 B2 JP5932642 B2 JP 5932642B2 JP 2012518704 A JP2012518704 A JP 2012518704A JP 2012518704 A JP2012518704 A JP 2012518704A JP 5932642 B2 JP5932642 B2 JP 5932642B2
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glp
disease
pain
gly
cancer
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JP2012531467A5 (cg-RX-API-DMAC10.html
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デムール，ミシェル
シェ，クリスティアン
ティオット，カリーン
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アンジオケム インコーポレーテッド
アンジオケム インコーポレーテッド
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/62—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
    • A61K47/64—Drug-peptide, drug-protein or drug-polyamino acid conjugates, i.e. the modifying agent being a peptide, protein or polyamino acid which is covalently bonded or complexed to a therapeutically active agent
    • A—HUMAN NECESSITIES
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

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  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Molecular Biology (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Anesthesiology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Physical Education & Sports Medicine (AREA)
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  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2012518704A 2009-07-02 2010-06-30 多量体ペプチドコンジュゲートおよびその使用 Expired - Fee Related JP5932642B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US22278509P 2009-07-02 2009-07-02
US61/222,785 2009-07-02
US25202409P 2009-10-15 2009-10-15
US61/252,024 2009-10-15
PCT/CA2010/001014 WO2011000095A1 (en) 2009-07-02 2010-06-30 Multimeric peptide conjugates and uses thereof

Publications (3)

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JP2012531467A JP2012531467A (ja) 2012-12-10
JP2012531467A5 JP2012531467A5 (cg-RX-API-DMAC10.html) 2013-08-15
JP5932642B2 true JP5932642B2 (ja) 2016-06-08

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US (1) US9161988B2 (cg-RX-API-DMAC10.html)
EP (1) EP2448965A4 (cg-RX-API-DMAC10.html)
JP (1) JP5932642B2 (cg-RX-API-DMAC10.html)
CN (1) CN102596993A (cg-RX-API-DMAC10.html)
AU (1) AU2010268726A1 (cg-RX-API-DMAC10.html)
BR (1) BRPI1015918A2 (cg-RX-API-DMAC10.html)
CA (1) CA2766537A1 (cg-RX-API-DMAC10.html)
IN (1) IN2012DN00248A (cg-RX-API-DMAC10.html)
MX (1) MX2012000016A (cg-RX-API-DMAC10.html)
RU (1) RU2012103240A (cg-RX-API-DMAC10.html)
WO (1) WO2011000095A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201109324B (cg-RX-API-DMAC10.html)

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