JP5646598B2 - 治療に用いるためのｆｇｆｒキナーゼ阻害薬としてのイミダゾ［１，２‐ａ］ピリジン誘導体 - Google Patents

治療に用いるためのｆｇｆｒキナーゼ阻害薬としてのイミダゾ［１，２‐ａ］ピリジン誘導体 Download PDF

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JP5646598B2
JP5646598B2 JP2012505239A JP2012505239A JP5646598B2 JP 5646598 B2 JP5646598 B2 JP 5646598B2 JP 2012505239 A JP2012505239 A JP 2012505239A JP 2012505239 A JP2012505239 A JP 2012505239A JP 5646598 B2 JP5646598 B2 JP 5646598B2
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alkyl
alkoxy
heterocyclyl
compound
cancer
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JP2012524056A5 (enExample
JP2012524056A (ja
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ゴードン、サクスティ
バレリオ、ベルディーニ
クリストファー、ウィリアム、マレー
エディ、ジャン、エドガー、フレイヌ
ヤニク、エメ、エディ、リニー
パスカル、ジスレーン、アンドレ、ボネ
ベルトルト、ブロブロブスキー
アレクサンドラ、パパニコス
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Astex Therapeutics Ltd
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Astex Therapeutics Ltd
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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JP2012505239A 2009-04-15 2010-04-15 治療に用いるためのｆｇｆｒキナーゼ阻害薬としてのイミダゾ［１，２‐ａ］ピリジン誘導体 Expired - Fee Related JP5646598B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US16950309P 2009-04-15 2009-04-15
GBGB0906470.0A GB0906470D0 (en) 2009-04-15 2009-04-15 New compounds
US61/169,503 2009-04-15
GB0906470.0 2009-04-15
PCT/GB2010/050618 WO2010119285A1 (en) 2009-04-15 2010-04-15 Imidazo [1,2-a]pyridine derivatives as fgfr kinase inhibitors for use in therapy

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JP2012524056A JP2012524056A (ja) 2012-10-11
JP2012524056A5 JP2012524056A5 (enExample) 2013-05-16
JP5646598B2 true JP5646598B2 (ja) 2014-12-24

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US (1) US8722687B2 (enExample)
EP (1) EP2419428B1 (enExample)
JP (1) JP5646598B2 (enExample)
AU (1) AU2010238290B2 (enExample)
CA (1) CA2757326C (enExample)
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ES (1) ES2545215T3 (enExample)
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SI (1) SI2419428T1 (enExample)
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