ATE210663T1 - Kondensierte imidazolderivate, ihre herstellung und verwendung - Google Patents

Kondensierte imidazolderivate, ihre herstellung und verwendung

Info

Publication number
ATE210663T1
ATE210663T1 AT95921968T AT95921968T ATE210663T1 AT E210663 T1 ATE210663 T1 AT E210663T1 AT 95921968 T AT95921968 T AT 95921968T AT 95921968 T AT95921968 T AT 95921968T AT E210663 T1 ATE210663 T1 AT E210663T1
Authority
AT
Austria
Prior art keywords
pct
production
date dec
condensed imidazole
imidazole derivatives
Prior art date
Application number
AT95921968T
Other languages
English (en)
Inventor
Muneo Takatani
Hitoshi Ikeda
Kyoko Iida
Hidenori Abe
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Application granted granted Critical
Publication of ATE210663T1 publication Critical patent/ATE210663T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
AT95921968T 1994-06-20 1995-06-15 Kondensierte imidazolderivate, ihre herstellung und verwendung ATE210663T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP13760094 1994-06-20
JP6412895 1995-03-24
PCT/JP1995/001192 WO1995035296A1 (en) 1994-06-20 1995-06-15 Condensed imidazole compounds, their production and use

Publications (1)

Publication Number Publication Date
ATE210663T1 true ATE210663T1 (de) 2001-12-15

Family

ID=26405261

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95921968T ATE210663T1 (de) 1994-06-20 1995-06-15 Kondensierte imidazolderivate, ihre herstellung und verwendung

Country Status (8)

Country Link
US (1) US5840732A (de)
EP (1) EP0767790B1 (de)
CN (1) CN1046725C (de)
AT (1) ATE210663T1 (de)
AU (1) AU2682695A (de)
CA (1) CA2191979A1 (de)
DE (1) DE69524598T2 (de)
WO (1) WO1995035296A1 (de)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ388598A3 (cs) * 1996-05-31 1999-07-14 Sankyo Company, Limited Léčivo proti autoimunní nemoci
US6455550B1 (en) 1997-08-22 2002-09-24 Hoffmann-La Roche Inc. N-alkanoylphenylalanine derivatives
SI1005445T1 (en) * 1997-08-22 2004-12-31 F. Hoffmann-La Roche Ag N-alkanoylphenylalanine derivatives
US6229011B1 (en) 1997-08-22 2001-05-08 Hoffman-La Roche Inc. N-aroylphenylalanine derivative VCAM-1 inhibitors
AU739511B2 (en) * 1997-08-22 2001-10-11 F. Hoffmann-La Roche Ag N-aroylphenylalanine derivatives
EP1050535A4 (de) 1997-11-11 2001-04-25 Ono Pharmaceutical Co Kondensierte pyrazinderivate
US6358971B1 (en) 1998-05-20 2002-03-19 Eli Lilly And Company Anti-viral compounds
US6867203B2 (en) 1998-12-29 2005-03-15 Abbott Laboratories Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
HUP0200343A3 (en) 1999-02-18 2005-04-28 Hoffmann La Roche Phenylalaninol derivatives, process for their preparation, pharmaceutical compositions containing them and their use
DE60014588T2 (de) 1999-02-18 2006-02-23 F. Hoffmann-La Roche Ag Thioamidderivate
MXPA02000625A (es) * 1999-07-21 2002-07-02 Boehringer Ingelheim Pharma Pequenas moleculas utiles en el tratamiento de enfermedades inflamatorias.
EP1478327B1 (de) * 2002-02-22 2015-04-29 Meda AB Verfahren zur reduzierung und behandlung von uvb-induzierter immunsuppression
ITFI20030058A1 (it) * 2003-03-06 2004-09-07 Univ Firenze Formulazioni farmaceutiche contenenti tiazolidinedioni
PL2121687T3 (pl) 2006-12-22 2016-03-31 Astex Therapeutics Ltd Pochodne amin tricyklicznych jako inhibitory białkowej kinazy tyrozynowej
JP5442448B2 (ja) 2006-12-22 2014-03-12 アステックス、セラピューティックス、リミテッド Ｆｇｆｒインヒビターとしての二環式ヘテロ環式化合物
GB0720038D0 (en) 2007-10-12 2007-11-21 Astex Therapeutics Ltd New compounds
GB0720041D0 (en) 2007-10-12 2007-11-21 Astex Therapeutics Ltd New Compounds
GB0810902D0 (en) 2008-06-13 2008-07-23 Astex Therapeutics Ltd New compounds
WO2010058402A1 (en) 2008-11-20 2010-05-27 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. Novel anti-biofilm agents
GB0906472D0 (en) 2009-04-15 2009-05-20 Astex Therapeutics Ltd New compounds
GB0906470D0 (en) 2009-04-15 2009-05-20 Astex Therapeutics Ltd New compounds
US10202376B2 (en) 2014-12-24 2019-02-12 Takeda Pharmaceutical Company Limited Heterocyclic compound
CN107286156A (zh) * 2016-04-05 2017-10-24 江苏新元素医药科技有限公司 新型urat1抑制剂及其在医药上的应用
KR20200088397A (ko) 2017-11-14 2020-07-22 칠드런'즈 메디컬 센터 코포레이션 신규 이미다조피리미딘 화합물 및 그의 용도
WO2019099578A1 (en) 2017-11-14 2019-05-23 Chidren's Medical Center Corporation Use of imidazopyrimidine for modulating human immune response
JP2021050161A (ja) 2019-09-25 2021-04-01 武田薬品工業株式会社 複素環化合物及びその用途

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB656607A (en) * 1948-01-23 1951-08-29 Kodak Ltd Improvements in dyes for use in photographic materials
US4105767A (en) * 1977-03-28 1978-08-08 Merck & Co., Inc. Imidazo [1,2-a] pyridines substituted with a thienyl, thiazolyl, or thiadiazolyl group
CA1164459A (en) * 1980-11-11 1984-03-27 Yung-Hsiung Yang Process for preparing (imidazo¬1,2-a|pyridine- 2-yl)-carbostyril or -3,4-dihydrocarbostyryl derivatives
US4470986A (en) * 1982-12-21 1984-09-11 Ciba-Geigy Corporation Certain imidazo (1,5-A) pyridine aliphatic carboxylic acid derivatives and their use as selective thromboxane inhibitors
US4507481A (en) * 1983-07-29 1985-03-26 Pennwalt Corporation Pyrrolo[1,2-a]imidazoles and imidazo[1,2-a]pyridines
US4590196A (en) * 1984-08-23 1986-05-20 Bristol-Myers Company Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives
EP0228006A1 (de) * 1985-12-16 1987-07-08 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridinverbindungen und Verfahren zu ihrer Herstellung
JPS6383067A (ja) * 1986-09-26 1988-04-13 Sumitomo Pharmaceut Co Ltd 新規コハク酸イミド誘導体
JPS6383085A (ja) * 1986-09-26 1988-04-13 Sumitomo Pharmaceut Co Ltd 新規なイミド誘導体
EP0299470B1 (de) * 1987-07-16 1996-12-04 Byk Gulden Lomberg Chemische Fabrik GmbH Imidazo[1,2-a]pyridine
US5082838A (en) * 1989-06-21 1992-01-21 Takeda Chemical Industries, Ltd. Sulfur-containing fused pyrimidine derivatives, their production and use
ATE119774T1 (de) * 1990-07-30 1995-04-15 Takeda Chemical Industries Ltd Imidazopyridinderivate und ihre verwendung.
US5260303A (en) * 1991-03-07 1993-11-09 G. D. Searle & Co. Imidazopyridines as serotonergic 5-HT3 antagonists
DE69209576T4 (de) * 1991-05-10 1997-01-30 Takeda Chemical Industries Ltd Pyridinderivate, deren Herstellung und Anwendung
US5457102A (en) * 1994-07-07 1995-10-10 Janssen Pharmaceutica, N.V. Pyrroloimidazolyl and imidazopyridinyl substituted 1H-benzimidazole derivatives
IL108520A (en) * 1993-02-15 1997-09-30 Byk Gulden Lomberg Chem Fab 2, 3, 8-TRISUBSTITUTED IMIDAZO £1, 2-a| PYRIDINE DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Also Published As

Publication number Publication date
DE69524598D1 (de) 2002-01-24
CN1046725C (zh) 1999-11-24
AU2682695A (en) 1996-01-15
DE69524598T2 (de) 2002-07-11
US5840732A (en) 1998-11-24
EP0767790B1 (de) 2001-12-12
CN1151161A (zh) 1997-06-04
WO1995035296A1 (en) 1995-12-28
CA2191979A1 (en) 1995-12-28
EP0767790A1 (de) 1997-04-16

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties