JP5536049B2 - 新規な置換ピリジン−２−オン及びピリダジン−３−オン - Google Patents

新規な置換ピリジン−２−オン及びピリダジン−３−オン Download PDF

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JP5536049B2
JP5536049B2 JP2011514004A JP2011514004A JP5536049B2 JP 5536049 B2 JP5536049 B2 JP 5536049B2 JP 2011514004 A JP2011514004 A JP 2011514004A JP 2011514004 A JP2011514004 A JP 2011514004A JP 5536049 B2 JP5536049 B2 JP 5536049B2
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formula
alkyl
arthritis
methyl
halogen
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JP2011524404A (ja
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デュードニー，ノーラン・ジェームス
コンドル，ラマ・ケィ
ロエ，ブラッドリー・イー
ロウ，イェン
マッキントッシュ，ジョエル
オーエンズ，ティモシー・ディー
ソス，マイケル
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F Hoffmann La Roche AG
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    • C07—ORGANIC CHEMISTRY
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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  • Chemical Kinetics & Catalysis (AREA)
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  • Immunology (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Transplantation (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
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  • Psychiatry (AREA)
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  • Gastroenterology & Hepatology (AREA)
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JP2011514004A 2008-06-24 2009-06-15 新規な置換ピリジン−２−オン及びピリダジン−３−オン Expired - Fee Related JP5536049B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US7527708P 2008-06-24 2008-06-24
US61/075,277 2008-06-24
PCT/EP2009/057320 WO2009156284A1 (en) 2008-06-24 2009-06-15 Novel substituted pyridin-2-ones and pyridazin-3-ones

Publications (2)

Publication Number Publication Date
JP2011524404A JP2011524404A (ja) 2011-09-01
JP5536049B2 true JP5536049B2 (ja) 2014-07-02

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JP2011514004A Expired - Fee Related JP5536049B2 (ja) 2008-06-24 2009-06-15 新規な置換ピリジン−２−オン及びピリダジン−３−オン

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US (4) US7902194B2 (es)
EP (1) EP2297142B1 (es)
JP (1) JP5536049B2 (es)
KR (1) KR101299867B1 (es)
CN (3) CN103709148B (es)
AR (1) AR072272A1 (es)
AU (1) AU2009264400B2 (es)
BR (1) BRPI0914657A2 (es)
CA (1) CA2728016C (es)
CL (1) CL2010001483A1 (es)
CO (1) CO6382183A2 (es)
CR (1) CR11815A (es)
EC (1) ECSP10010709A (es)
ES (1) ES2552320T3 (es)
HK (2) HK1152940A1 (es)
IL (1) IL209141A0 (es)
MA (1) MA32487B1 (es)
MX (1) MX2010013191A (es)
NZ (2) NZ588819A (es)
PE (1) PE20100851A1 (es)
RU (1) RU2500680C2 (es)
TW (1) TWI396537B (es)
UA (1) UA103327C2 (es)
WO (1) WO2009156284A1 (es)
ZA (1) ZA201007816B (es)

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UA103327C2 (en) 2013-10-10
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US8618098B2 (en) 2013-12-31
CA2728016A1 (en) 2009-12-30
CR11815A (es) 2011-01-10
RU2011101774A (ru) 2012-07-27
US20110105479A1 (en) 2011-05-05
CO6382183A2 (es) 2012-02-15
CL2010001483A1 (es) 2011-05-13
US8822457B2 (en) 2014-09-02
TW201002683A (en) 2010-01-16
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US7902194B2 (en) 2011-03-08
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RU2500680C2 (ru) 2013-12-10
HK1196358A1 (en) 2014-12-12
CN103709148B (zh) 2015-10-21
US8124604B2 (en) 2012-02-28
MX2010013191A (es) 2010-12-17
KR20110011706A (ko) 2011-02-08
EP2297142A1 (en) 2011-03-23
EP2297142B1 (en) 2015-10-14
BRPI0914657A2 (pt) 2019-09-24
CN102066366A (zh) 2011-05-18
KR101299867B1 (ko) 2013-08-23
JP2011524404A (ja) 2011-09-01
CA2728016C (en) 2017-02-28
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