JP4716980B2 - ベンゾチアゼピン及びベンゾチエピン誘導体 - Google Patents

ベンゾチアゼピン及びベンゾチエピン誘導体 Download PDF

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Publication number
JP4716980B2
JP4716980B2 JP2006502310A JP2006502310A JP4716980B2 JP 4716980 B2 JP4716980 B2 JP 4716980B2 JP 2006502310 A JP2006502310 A JP 2006502310A JP 2006502310 A JP2006502310 A JP 2006502310A JP 4716980 B2 JP4716980 B2 JP 4716980B2
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formula
solvate
pharmaceutically acceptable
salt
alkyl
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Expired - Fee Related
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JP2006518728A5 (enExample
JP2006518728A (ja
Inventor
スターク，インゲマー
アレンフォーク，スザンヌ
ノードバーグ，マッツ・ペーター
ダールストロム，ミカエル・ウルフ・ヨハン
ボストロム，スティグ・ヨナス
レムレル，マリン・アニタ
ウォールバーグ，アンドレアス・クリスター
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アルビレオ・アクチボラグ
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02—Seven-membered rings
    • C07D337/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/08—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2006502310A 2003-02-25 2004-02-23 ベンゾチアゼピン及びベンゾチエピン誘導体 Expired - Fee Related JP4716980B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0304194.4 2003-02-25
GBGB0304194.4A GB0304194D0 (en) 2003-02-25 2003-02-25 Chemical compounds
PCT/GB2004/000695 WO2004076430A1 (en) 2003-02-25 2004-02-23 Benzothiazepine and benzothiepine derivatives

Publications (3)

Publication Number Publication Date
JP2006518728A JP2006518728A (ja) 2006-08-17
JP2006518728A5 JP2006518728A5 (enExample) 2006-11-30
JP4716980B2 true JP4716980B2 (ja) 2011-07-06

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ID=9953554

Family Applications (1)

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JP2006502310A Expired - Fee Related JP4716980B2 (ja) 2003-02-25 2004-02-23 ベンゾチアゼピン及びベンゾチエピン誘導体

Country Status (5)

Country Link
US (1) US8067584B2 (enExample)
EP (1) EP1597245A1 (enExample)
JP (1) JP4716980B2 (enExample)
GB (1) GB0304194D0 (enExample)
WO (1) WO2004076430A1 (enExample)

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GB0314079D0 (en) * 2003-06-18 2003-07-23 Astrazeneca Ab Therapeutic agents
SE0104334D0 (sv) 2001-12-19 2001-12-19 Astrazeneca Ab Therapeutic agents
GB0201850D0 (en) 2002-01-26 2002-03-13 Astrazeneca Ab Therapeutic treatment
GB0209467D0 (en) * 2002-04-25 2002-06-05 Astrazeneca Ab Chemical compounds
GB0213669D0 (en) * 2002-06-14 2002-07-24 Astrazeneca Ab Chemical compounds
GB0216321D0 (en) 2002-07-13 2002-08-21 Astrazeneca Ab Therapeutic treatment
GB0304194D0 (en) 2003-02-25 2003-03-26 Astrazeneca Ab Chemical compounds
GB0307918D0 (en) 2003-04-05 2003-05-14 Astrazeneca Ab Therapeutic use

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GB0304194D0 (en) 2003-03-26
US20060094884A1 (en) 2006-05-04
US8067584B2 (en) 2011-11-29
JP2006518728A (ja) 2006-08-17
WO2004076430A1 (en) 2004-09-10

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