JP4508651B2 - ２−フロ酸フルチカゾンの結晶性複合体 - Google Patents

２−フロ酸フルチカゾンの結晶性複合体 Download PDF

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Publication number
JP4508651B2
JP4508651B2 JP2003566027A JP2003566027A JP4508651B2 JP 4508651 B2 JP4508651 B2 JP 4508651B2 JP 2003566027 A JP2003566027 A JP 2003566027A JP 2003566027 A JP2003566027 A JP 2003566027A JP 4508651 B2 JP4508651 B2 JP 4508651B2
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complex
formula
compound
complex according
guest molecule
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Expired - Lifetime
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Japanese (ja)
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JP2005527497A (ja
JP2005527497A5 (enExample
Inventor
ビッガーダイク，キース
コーテ，スティーヴン，ジョン
クレイグ，アンドリュー
クロウェ，デヴィッド，マルコム
ジェスウィッツ，ヴィクター，ウィットールド
ミラン，マイケル，ジョン
ナイス，ロザリン，ケイ
ノガ，ブライアン
シーゲル，ジョン，フレデリック
セオフィラス，アンドリュー，リュイス
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Glaxo Group Ltd
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Glaxo Group Ltd
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
JP2003566027A 2002-02-04 2003-02-04 ２−フロ酸フルチカゾンの結晶性複合体 Expired - Lifetime JP4508651B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/067,010 US6777399B2 (en) 2000-08-05 2002-02-04 Anti-inflammatory androstane derivative compositions
PCT/GB2003/000478 WO2003066656A1 (en) 2002-02-04 2003-02-04 Crystalline complexes of fluticasone 2-furoate

Publications (3)

Publication Number Publication Date
JP2005527497A JP2005527497A (ja) 2005-09-15
JP2005527497A5 JP2005527497A5 (enExample) 2006-01-05
JP4508651B2 true JP4508651B2 (ja) 2010-07-21

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003566027A Expired - Lifetime JP4508651B2 (ja) 2002-02-04 2003-02-04 ２−フロ酸フルチカゾンの結晶性複合体

Country Status (8)

Country Link
US (3) US6777399B2 (enExample)
EP (1) EP1472272B1 (enExample)
JP (1) JP4508651B2 (enExample)
AT (1) ATE462711T1 (enExample)
AU (1) AU2003207019A1 (enExample)
DE (1) DE60331891D1 (enExample)
ES (1) ES2343315T3 (enExample)
WO (1) WO2003066656A1 (enExample)

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EP1472272B1 (en) 2010-03-31
US20040224932A1 (en) 2004-11-11
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DE60331891D1 (de) 2010-05-12
EP1472272A1 (en) 2004-11-03
US20050043284A1 (en) 2005-02-24
ATE462711T1 (de) 2010-04-15
US7592329B2 (en) 2009-09-22
ES2343315T3 (es) 2010-07-28
US20030153542A1 (en) 2003-08-14
AU2003207019A1 (en) 2003-09-02
WO2003066656A1 (en) 2003-08-14

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