JP3313708B2 - イミダゾ〔４，５−ｃ〕キノリン−４−アミンの製法 - Google Patents

イミダゾ〔４，５−ｃ〕キノリン−４−アミンの製法

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Publication number
JP3313708B2
JP3313708B2 JP50932392A JP50932392A JP3313708B2 JP 3313708 B2 JP3313708 B2 JP 3313708B2 JP 50932392 A JP50932392 A JP 50932392A JP 50932392 A JP50932392 A JP 50932392A JP 3313708 B2 JP3313708 B2 JP 3313708B2
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JP
Japan
Prior art keywords
carbon atoms
alkyl
group
phenyl
substituted
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
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JP50932392A
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English (en)
Japanese (ja)
Other versions
JPH06505499A (ja
Inventor
エフ． ジャースター，ジョン
Original Assignee
ミネソタ マイニング アンド マニュファクチャリング カンパニー
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Publication of JPH06505499A publication Critical patent/JPH06505499A/ja
Application granted granted Critical
Publication of JP3313708B2 publication Critical patent/JP3313708B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP50932392A 1991-03-01 1992-02-13 イミダゾ〔４，５−ｃ〕キノリン−４−アミンの製法 Expired - Lifetime JP3313708B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US663,110 1991-03-01
US07/663,110 US5175296A (en) 1991-03-01 1991-03-01 Imidazo[4,5-c]quinolin-4-amines and processes for their preparation
PCT/US1992/001212 WO1992015581A1 (en) 1991-03-01 1992-02-13 PROCESS FOR IMIDAZO[4,5-c]QUINOLIN-4-AMINES

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP03146599A Division JP3450736B2 (ja) 1991-03-01 1999-02-09 イミダゾ〔４，５−ｃ〕キノリン−４−アミンの中間体及びその製法

Publications (2)

Publication Number Publication Date
JPH06505499A JPH06505499A (ja) 1994-06-23
JP3313708B2 true JP3313708B2 (ja) 2002-08-12

Family

ID=24660514

Family Applications (2)

Application Number Title Priority Date Filing Date
JP50932392A Expired - Lifetime JP3313708B2 (ja) 1991-03-01 1992-02-13 イミダゾ〔４，５−ｃ〕キノリン−４−アミンの製法
JP03146599A Expired - Lifetime JP3450736B2 (ja) 1991-03-01 1999-02-09 イミダゾ〔４，５−ｃ〕キノリン−４−アミンの中間体及びその製法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP03146599A Expired - Lifetime JP3450736B2 (ja) 1991-03-01 1999-02-09 イミダゾ〔４，５−ｃ〕キノリン−４−アミンの中間体及びその製法

Country Status (17)

Country Link
US (1) US5175296A (https=)
EP (1) EP0575549B1 (https=)
JP (2) JP3313708B2 (https=)
KR (1) KR100226184B1 (https=)
AT (1) ATE142632T1 (https=)
AU (1) AU657958B2 (https=)
CA (1) CA2104781C (https=)
CZ (1) CZ291368B6 (https=)
DE (1) DE69213720T2 (https=)
DK (1) DK0575549T3 (https=)
ES (1) ES2091463T3 (https=)
HU (1) HU218219B (https=)
IE (1) IE920524A1 (https=)
IL (1) IL100998A (https=)
NO (1) NO301714B1 (https=)
NZ (1) NZ241645A (https=)
WO (1) WO1992015581A1 (https=)

Families Citing this family (171)

* Cited by examiner, † Cited by third party
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US5395937A (en) * 1993-01-29 1995-03-07 Minnesota Mining And Manufacturing Company Process for preparing quinoline amines
US5648516A (en) * 1994-07-20 1997-07-15 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
JPH09500128A (ja) * 1993-07-15 1997-01-07 ミネソタ マイニング アンド マニュファクチャリング カンパニー イミダゾ〔４，５−ｃ〕ピリジン−４−アミン
US5352784A (en) * 1993-07-15 1994-10-04 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
US5644063A (en) * 1994-09-08 1997-07-01 Minnesota Mining And Manufacturing Company Imidazo[4,5-c]pyridin-4-amine intermediates
US5693811A (en) * 1996-06-21 1997-12-02 Minnesota Mining And Manufacturing Company Process for preparing tetrahdroimidazoquinolinamines
US5741908A (en) * 1996-06-21 1998-04-21 Minnesota Mining And Manufacturing Company Process for reparing imidazoquinolinamines
UA67760C2 (uk) * 1997-12-11 2004-07-15 Міннесота Майнінг Енд Мануфакчурінг Компані Імідазонафтиридин та тетрагідроімідазонафтиридин, фармацевтична композиція, спосіб індукування біосинтезу цитокінів та спосіб лікування вірусної інфекції, проміжні сполуки
HU229441B1 (en) 1999-01-08 2013-12-30 3M Innovative Properties Co Formulations and methods for treating mucosal associated conditions with an immune response modifier
US6486168B1 (en) 1999-01-08 2002-11-26 3M Innovative Properties Company Formulations and methods for treatment of mucosal associated conditions with an immune response modifier
US20020058674A1 (en) 1999-01-08 2002-05-16 Hedenstrom John C. Systems and methods for treating a mucosal surface
US6558951B1 (en) * 1999-02-11 2003-05-06 3M Innovative Properties Company Maturation of dendritic cells with immune response modifying compounds
US6331539B1 (en) * 1999-06-10 2001-12-18 3M Innovative Properties Company Sulfonamide and sulfamide substituted imidazoquinolines
US6541485B1 (en) 1999-06-10 2003-04-01 3M Innovative Properties Company Urea substituted imidazoquinolines
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US6376669B1 (en) 1999-11-05 2002-04-23 3M Innovative Properties Company Dye labeled imidazoquinoline compounds
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CA2399136A1 (en) * 2000-02-09 2001-08-16 Hideo Kato 1h-imidazopyridine derivatives
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US6667312B2 (en) * 2000-12-08 2003-12-23 3M Innovative Properties Company Thioether substituted imidazoquinolines
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JP2005501550A (ja) * 2001-08-30 2005-01-20 スリーエム イノベイティブ プロパティズ カンパニー 免疫反応調整剤分子を用いた形質細胞様樹状細胞を成熟させる方法
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WO2003101949A2 (en) 2002-05-29 2003-12-11 3M Innovative Properties Company Process for imidazo[4,5-c]pyridin-4-amines
JP2005538057A (ja) * 2002-06-07 2005-12-15 スリーエム イノベイティブ プロパティズ カンパニー エーテル置換イミダゾピリジン
AU2003259226A1 (en) 2002-07-23 2004-02-09 Biogal Gyogyszergyar Rt Preparation of 1h-imidazo(4,5-c)quinolin-4-amines via1h-imidazo (4,5-c)quinolin-4-phthalimide intermediates
PT1539752E (pt) 2002-07-26 2007-05-31 Teva Gyogyszergyar Zartkoeruen Preparação de 1h-imidazo [4,5-c] quinolina-4-aminas via novos intermediários imidazo [4,5-c] quinolina-4-ciano e 1h-imidazo [4,5-c] quinolina-4-carboxamida
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JP2006503068A (ja) * 2002-09-26 2006-01-26 スリーエム イノベイティブ プロパティズ カンパニー １ｈ−イミダゾダイマー
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US7163947B2 (en) * 2003-03-07 2007-01-16 3M Innovative Properties Company 1-Amino 1H-imidazoquinolines
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HUT66968A (en) 1995-01-30
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US5175296A (en) 1992-12-29
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ES2091463T3 (es) 1996-11-01
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