JP2025502842A5 - - Google Patents

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Publication number
JP2025502842A5
JP2025502842A5 JP2024539928A JP2024539928A JP2025502842A5 JP 2025502842 A5 JP2025502842 A5 JP 2025502842A5 JP 2024539928 A JP2024539928 A JP 2024539928A JP 2024539928 A JP2024539928 A JP 2024539928A JP 2025502842 A5 JP2025502842 A5 JP 2025502842A5
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JP
Japan
Prior art keywords
crystalline form
alpha
compound
radiation source
measured
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024539928A
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English (en)
Japanese (ja)
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JP2025502842A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/087952 external-priority patent/WO2023126436A1/en
Publication of JP2025502842A publication Critical patent/JP2025502842A/ja
Publication of JP2025502842A5 publication Critical patent/JP2025502842A5/ja
Pending legal-status Critical Current

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JP2024539928A 2021-12-29 2022-12-28 薬学的に活性な化合物としての使用のための(5s)-{[2-(4-カルボキシフェニル)エチル][2-(2-{[3-クロロ-4’-(トリフルオロメチル)ビフェニル-4-イル]メトキシ}フェニル)エチル]アミノ}-5,6,7,8-テトラヒドロキノリン-2-カルボン酸及びその結晶形態を調製するための方法 Pending JP2025502842A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP21218163 2021-12-29
EP21218163.0 2021-12-29
PCT/EP2022/087952 WO2023126436A1 (en) 2021-12-29 2022-12-28 Process for preparing (5s)-{[2-(4-carboxyphenyl)ethyl] |2-(2-{|3-chloro-4'-(trifluoromethyl)biphenyl-4- yl]methoxy}phenyl)ethyl]aminol-5,6,7,8-tetrahydroquinoline-2-carboxylic acid and its crystalline forms for use as pharmaceutically active compound

Publications (2)

Publication Number Publication Date
JP2025502842A JP2025502842A (ja) 2025-01-28
JP2025502842A5 true JP2025502842A5 (enExample) 2026-01-09

Family

ID=79185525

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024539928A Pending JP2025502842A (ja) 2021-12-29 2022-12-28 薬学的に活性な化合物としての使用のための(5s)-{[2-(4-カルボキシフェニル)エチル][2-(2-{[3-クロロ-4’-(トリフルオロメチル)ビフェニル-4-イル]メトキシ}フェニル)エチル]アミノ}-5,6,7,8-テトラヒドロキノリン-2-カルボン酸及びその結晶形態を調製するための方法

Country Status (12)

Country Link
US (2) US12202805B2 (enExample)
EP (1) EP4457215A1 (enExample)
JP (1) JP2025502842A (enExample)
KR (1) KR20240144177A (enExample)
CN (1) CN118765272A (enExample)
AR (1) AR128147A1 (enExample)
AU (1) AU2022429647A1 (enExample)
CA (1) CA3244893A1 (enExample)
IL (1) IL313922A (enExample)
MX (1) MX2024008172A (enExample)
TW (1) TW202342012A (enExample)
WO (1) WO2023126436A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202342034A (zh) 2021-12-29 2023-11-01 德商拜耳廠股份有限公司 心肺病症之治療
AU2022429647A1 (en) 2021-12-29 2024-07-04 Bayer Aktiengesellschaft Process for preparing (5s)-{[2-(4-carboxyphenyl)ethyl] |2-(2-{|3-chloro-4'-(trifluoromethyl)biphenyl-4- yl]methoxy}phenyl)ethyl]aminol-5,6,7,8-tetrahydroquinoline-2-carboxylic acid and its crystalline forms for use as pharmaceutically active compound

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KR20230012494A (ko) 2020-05-20 2023-01-26 바이엘 악티엔게젤샤프트 부틸 (5s)-5-({2-[4-(부톡시카르보닐)페닐]에틸}[2-(2-{[3-클로로-4'-(트리플루오로메틸)[비페닐]-4-일]메톡시}페닐)에틸]아미노)-5,6,7,8-테트라히드로퀴놀린-2-카르복실레이트의 제조 방법
TW202342035A (zh) 2021-12-29 2023-11-01 德商拜耳廠股份有限公司 醫藥乾粉吸入配製物
TW202342034A (zh) 2021-12-29 2023-11-01 德商拜耳廠股份有限公司 心肺病症之治療
AU2022429647A1 (en) 2021-12-29 2024-07-04 Bayer Aktiengesellschaft Process for preparing (5s)-{[2-(4-carboxyphenyl)ethyl] |2-(2-{|3-chloro-4'-(trifluoromethyl)biphenyl-4- yl]methoxy}phenyl)ethyl]aminol-5,6,7,8-tetrahydroquinoline-2-carboxylic acid and its crystalline forms for use as pharmaceutically active compound

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