JP2024518554A5 - - Google Patents

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Publication number
JP2024518554A5
JP2024518554A5 JP2023570165A JP2023570165A JP2024518554A5 JP 2024518554 A5 JP2024518554 A5 JP 2024518554A5 JP 2023570165 A JP2023570165 A JP 2023570165A JP 2023570165 A JP2023570165 A JP 2023570165A JP 2024518554 A5 JP2024518554 A5 JP 2024518554A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
alkyl
diluent
acceptable salt
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023570165A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024518554A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/029102 external-priority patent/WO2022241171A1/en
Publication of JP2024518554A publication Critical patent/JP2024518554A/ja
Publication of JP2024518554A5 publication Critical patent/JP2024518554A5/ja
Pending legal-status Critical Current

Links

JP2023570165A 2021-05-14 2022-05-13 置換ヘテロ環化合物 Pending JP2024518554A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163188498P 2021-05-14 2021-05-14
US63/188,498 2021-05-14
US202263318149P 2022-03-09 2022-03-09
US63/318,149 2022-03-09
PCT/US2022/029102 WO2022241171A1 (en) 2021-05-14 2022-05-13 Substituted heterocyclic compounds

Publications (2)

Publication Number Publication Date
JP2024518554A JP2024518554A (ja) 2024-05-01
JP2024518554A5 true JP2024518554A5 (https=) 2025-03-12

Family

ID=81927926

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023570165A Pending JP2024518554A (ja) 2021-05-14 2022-05-13 置換ヘテロ環化合物

Country Status (13)

Country Link
US (3) US11866414B2 (https=)
EP (1) EP4337655A1 (https=)
JP (1) JP2024518554A (https=)
KR (1) KR20240008336A (https=)
AU (1) AU2022271794A1 (https=)
CA (1) CA3217332A1 (https=)
CL (1) CL2023003308A1 (https=)
CO (1) CO2023015226A2 (https=)
IL (1) IL308421A (https=)
MX (1) MX2023013445A (https=)
PE (1) PE20250262A1 (https=)
TW (1) TW202311247A (https=)
WO (1) WO2022241171A1 (https=)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2019373203B2 (en) * 2018-10-30 2024-10-24 Bristol-Myers Squibb Company Amide-substituted heterocyclic compounds for the treatment of conditions related to the modulation of IL-12, IL-23 and/or IFN-alpha
EP4146205A4 (en) 2020-05-05 2024-05-29 Nuvalent, Inc. HETEROAROMATIC MACROCYCLIC ETHERS AS CHEMOTHERAPEUTIC AGENTS
IL297832A (en) 2020-05-05 2023-01-01 Nuvalent Inc Macrocyclic heteroaromatic chemotherapeutic agents
US12492184B2 (en) 2020-12-22 2025-12-09 InventisBio Co., Ltd. Heteroaryl compounds, preparation methods and uses thereof
CA3208361A1 (en) 2021-02-19 2022-08-25 Anjali Pandey Tyk2 inhibitors and uses thereof
EP4294806A1 (en) 2021-02-19 2023-12-27 Sudo Biosciences Limited Tyk2 inhibitors and uses thereof
AU2022222470A1 (en) 2021-02-19 2023-09-21 Sudo Biosciences Limited Tyk2 inhibitors and uses thereof
BR112023019861A2 (pt) 2021-03-31 2023-11-07 Xinthera Inc Inibidores de mk2 e usos dos mesmos
US20240317718A1 (en) * 2021-05-14 2024-09-26 Bristol-Myers Squibb Company Substituted heterocyclic compounds
KR20240008337A (ko) * 2021-05-14 2024-01-18 브리스톨-마이어스 스큅 컴퍼니 치환된 헤테로시클릭 화합물
PE20250262A1 (es) * 2021-05-14 2025-01-29 Bristol Myers Squibb Co Compuestos heterociclicos sustituidos
US11884650B2 (en) * 2021-05-14 2024-01-30 Bristol-Myers Squibb Company Substituted heterocyclic compounds
JP2024518791A (ja) * 2021-05-14 2024-05-02 ブリストル-マイヤーズ スクイブ カンパニー 置換ヘテロ環化合物
CN115724830A (zh) * 2021-08-31 2023-03-03 浙江文达医药科技有限公司 作为tyk2/jak1假激酶结构域(jh2)抑制剂的化合物及合成和使用方法
TW202320768A (zh) 2021-10-01 2023-06-01 美商努法倫特公司 雜芳族大環醚化合物之固體形式、醫藥組成物及製備
WO2024044486A1 (en) * 2022-08-22 2024-02-29 Ajax Therapeutics, Inc. Jak2 inhibitor compounds
CN120152968A (zh) * 2022-11-08 2025-06-13 百时美施贵宝公司 取代的杂环化合物
CN118812511A (zh) * 2023-04-21 2024-10-22 浙江文达医药科技有限公司 作为tyk2抑制剂的杂环化合物及合成和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT3495358T (lt) * 2012-11-08 2022-05-25 Bristol-Myers Squibb Company Amidais pakeisti heterocikliniai junginiai, naudingi kaip il-12, il-23 ir (arba) ifn alfa atsako moduliatoriai
JP7113023B2 (ja) 2017-03-30 2022-08-04 ブリストル-マイヤーズ スクイブ カンパニー 6-(シクロプロパンアミド)-4-((2-メトキシ-3-(1-メチル-1h-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-n-(メチル-d3)ピリダジン-3-カルボキシアミドの製造方法
PE20250262A1 (es) * 2021-05-14 2025-01-29 Bristol Myers Squibb Co Compuestos heterociclicos sustituidos

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