JP2023504542A5 - - Google Patents

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Publication number
JP2023504542A5
JP2023504542A5 JP2022533451A JP2022533451A JP2023504542A5 JP 2023504542 A5 JP2023504542 A5 JP 2023504542A5 JP 2022533451 A JP2022533451 A JP 2022533451A JP 2022533451 A JP2022533451 A JP 2022533451A JP 2023504542 A5 JP2023504542 A5 JP 2023504542A5
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haloalkyl
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JP2022533451A
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Japanese (ja)
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JP7721143B2 (ja
JP2023504542A (ja
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Priority claimed from PCT/US2020/063383 external-priority patent/WO2021113690A1/en
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JP2022533451A 2019-12-04 2020-12-04 Masp-2阻害剤および使用方法 Active JP7721143B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962943622P 2019-12-04 2019-12-04
US62/943,622 2019-12-04
PCT/US2020/063383 WO2021113690A1 (en) 2019-12-04 2020-12-04 Masp-2 inhibitors and methods of use

Publications (3)

Publication Number Publication Date
JP2023504542A JP2023504542A (ja) 2023-02-03
JP2023504542A5 true JP2023504542A5 (https=) 2023-10-05
JP7721143B2 JP7721143B2 (ja) 2025-08-12

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JP2022533451A Active JP7721143B2 (ja) 2019-12-04 2020-12-04 Masp-2阻害剤および使用方法

Country Status (11)

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US (1) US11661418B2 (https=)
EP (1) EP4069678A1 (https=)
JP (1) JP7721143B2 (https=)
KR (1) KR20220110529A (https=)
CN (1) CN115052862A (https=)
AU (1) AU2020397894B2 (https=)
BR (1) BR112022010881A2 (https=)
CA (1) CA3159167A1 (https=)
IL (1) IL293551A (https=)
WO (1) WO2021113690A1 (https=)
ZA (1) ZA202409281B (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
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IL311042B1 (en) 2018-05-29 2026-04-01 Omeros Corp MASP-2 inhibitors and methods of use
EP4069676A1 (en) 2019-12-04 2022-10-12 Omeros Corporation Masp-2 inhibitors and methods of use
IL293588B1 (en) 2019-12-04 2026-04-01 Omeros Corp 3-Amino-1-methylpyrazin-2(H1)-one derivatives as MASP-2 inhibitors, compositions containing them and uses thereof
BR112022010895A2 (pt) 2019-12-04 2022-09-06 Omeros Corp Composto, composição farmacêutica, e, método para tratar uma doença ou distúrbio associado à serina protease-2 associada à lectina de ligação ao manan
TWI834025B (zh) 2020-03-06 2024-03-01 美商奥默羅斯公司 用於治療和/或預防冠狀病毒誘導的急性呼吸窘迫症候群的抑制masp-2的方法
EP4471023A4 (en) * 2022-01-28 2025-09-03 Wuhan Createrna Science And Tech Co Ltd MASP-2 INHIBITOR COMPOUND, PHARMACEUTICAL COMPOSITION, PREPARATION METHOD THEREOF AND USE THEREOF
WO2025207595A1 (en) * 2024-03-25 2025-10-02 Entasis Therapeutics, Inc. Modulators of mannan-binding lectin-associated protease

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KR102528260B1 (ko) 2016-01-05 2023-05-04 유니버시티 오브 레스터 필요로 하는 대상체에서 섬유증의 억제 방법
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JOP20170170B1 (ar) 2016-08-31 2022-09-15 Omeros Corp صيغ لجسم مضاد تثبيطية لـ masp-2 بتركيز عالي ولزوجة منخفضة وأطقم، وطرق
US20180105604A1 (en) 2016-10-13 2018-04-19 University Of Leicester Methods for reducing proteinuria in a human subject suffering from immunoglobulin a nephropathy
TWI881481B (zh) 2017-08-15 2025-04-21 美商歐米諾斯公司 用於治療和/或預防與造血幹細胞移植有關的移植物抗宿主病和/或瀰漫性肺泡出血和/或靜脈閉塞性病的方法
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IL311042B1 (en) * 2018-05-29 2026-04-01 Omeros Corp MASP-2 inhibitors and methods of use
EP4069676A1 (en) 2019-12-04 2022-10-12 Omeros Corporation Masp-2 inhibitors and methods of use
BR112022010895A2 (pt) 2019-12-04 2022-09-06 Omeros Corp Composto, composição farmacêutica, e, método para tratar uma doença ou distúrbio associado à serina protease-2 associada à lectina de ligação ao manan
IL293588B1 (en) 2019-12-04 2026-04-01 Omeros Corp 3-Amino-1-methylpyrazin-2(H1)-one derivatives as MASP-2 inhibitors, compositions containing them and uses thereof

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