JP2023508332A5 - - Google Patents

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Publication number
JP2023508332A5
JP2023508332A5 JP2022538232A JP2022538232A JP2023508332A5 JP 2023508332 A5 JP2023508332 A5 JP 2023508332A5 JP 2022538232 A JP2022538232 A JP 2022538232A JP 2022538232 A JP2022538232 A JP 2022538232A JP 2023508332 A5 JP2023508332 A5 JP 2023508332A5
Authority
JP
Japan
Prior art keywords
unsubstituted
cancer
substituted
compound
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022538232A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023508332A (ja
JP7750526B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/065410 external-priority patent/WO2021127045A1/en
Publication of JP2023508332A publication Critical patent/JP2023508332A/ja
Publication of JP2023508332A5 publication Critical patent/JP2023508332A5/ja
Application granted granted Critical
Publication of JP7750526B2 publication Critical patent/JP7750526B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022538232A 2019-12-20 2020-12-16 組み合わせ Active JP7750526B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962952032P 2019-12-20 2019-12-20
US62/952,032 2019-12-20
PCT/US2020/065410 WO2021127045A1 (en) 2019-12-20 2020-12-16 Combinations

Publications (3)

Publication Number Publication Date
JP2023508332A JP2023508332A (ja) 2023-03-02
JP2023508332A5 true JP2023508332A5 (enExample) 2023-12-25
JP7750526B2 JP7750526B2 (ja) 2025-10-07

Family

ID=76478077

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022538232A Active JP7750526B2 (ja) 2019-12-20 2020-12-16 組み合わせ

Country Status (12)

Country Link
US (1) US20230054854A1 (enExample)
EP (1) EP4069242A4 (enExample)
JP (1) JP7750526B2 (enExample)
KR (1) KR20220119420A (enExample)
CN (2) CN121102230A (enExample)
AU (1) AU2020404996A1 (enExample)
BR (1) BR112022012283A2 (enExample)
CA (1) CA3165474A1 (enExample)
IL (1) IL294094A (enExample)
MX (1) MX2022007623A (enExample)
TW (1) TWI875898B (enExample)
WO (1) WO2021127045A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4566612A3 (en) 2018-03-09 2025-08-20 Recurium IP Holdings, LLC Substituted 1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-ones
AU2020384291A1 (en) 2019-11-15 2022-05-26 Recurium Ip Holdings, Llc Chiral synthesis of a tertiary alcohol
WO2022011391A1 (en) 2020-07-09 2022-01-13 Recurium Ip Holdings, Llc Salts and forms of a wee1 inhibitor
US12084453B2 (en) 2021-12-10 2024-09-10 Incyte Corporation Bicyclic amines as CDK12 inhibitors
WO2023147297A2 (en) * 2022-01-25 2023-08-03 Verastem, Inc. Combination therapy for treating abnormal cell growth
WO2025193930A1 (en) * 2024-03-14 2025-09-18 Zeno Management, Inc. Wee1 inhibitor combination therapy

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102124715B1 (ko) * 2015-11-03 2020-06-18 제넨테크, 인크. 암의 치료를 위한 bcl-2 억제제 및 mek 억제제의 조합물
CN109422754A (zh) * 2017-08-24 2019-03-05 上海迪诺医药科技有限公司 吡唑并[3,4-d]嘧啶-3-酮衍生物、其药物组合物及应用
KR20200108301A (ko) * 2018-01-10 2020-09-17 리커리엄 아이피 홀딩스, 엘엘씨 벤즈아미드 화합물
WO2019165204A1 (en) * 2018-02-23 2019-08-29 Newave Pharmaceutical Inc. 1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidine-3-one compounds as inhibitors of wee-1 kinase
US12220415B2 (en) * 2018-02-28 2025-02-11 The Regents Of The University Of Colorado, A Body Corporate WEE1 kinase inhibitors and methods of treating cancer using the same
EP4566612A3 (en) * 2018-03-09 2025-08-20 Recurium IP Holdings, LLC Substituted 1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-ones

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