JP2022543250A5 - - Google Patents
Info
- Publication number
- JP2022543250A5 JP2022543250A5 JP2022506745A JP2022506745A JP2022543250A5 JP 2022543250 A5 JP2022543250 A5 JP 2022543250A5 JP 2022506745 A JP2022506745 A JP 2022506745A JP 2022506745 A JP2022506745 A JP 2022506745A JP 2022543250 A5 JP2022543250 A5 JP 2022543250A5
- Authority
- JP
- Japan
- Prior art keywords
- pyridine
- fluorophenyl
- oxo
- carboxamide
- oxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20190094455 | 2019-08-02 | ||
| KR10-2019-0094455 | 2019-08-02 | ||
| PCT/KR2020/010204 WO2021025407A1 (ko) | 2019-08-02 | 2020-08-03 | 옥소-피리딘 융합고리 유도체 및 이를 포함하는 약학적 조성물 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022543250A JP2022543250A (ja) | 2022-10-11 |
| JP2022543250A5 true JP2022543250A5 (https=) | 2023-08-10 |
Family
ID=74503219
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022506745A Pending JP2022543250A (ja) | 2019-08-02 | 2020-08-03 | オキソ-ピリジン縮合環誘導体、およびそれを含む医薬組成物 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20220235064A1 (https=) |
| EP (1) | EP4011885A4 (https=) |
| JP (1) | JP2022543250A (https=) |
| KR (1) | KR20210015730A (https=) |
| CN (1) | CN114206883A (https=) |
| WO (1) | WO2021025407A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2023513675A (ja) * | 2020-02-06 | 2023-04-03 | ウェルマーカー・バイオ・カンパニー・リミテッド | Kras変異に関連する癌の予防または治療のための医薬組成物 |
| KR20210111711A (ko) * | 2020-03-03 | 2021-09-13 | 웰마커바이오 주식회사 | Kras 돌연변이 및 활성화된 ron이 존재하는 암의 예방 또는 치료용 약학 조성물 |
| JP2023526443A (ja) * | 2020-05-18 | 2023-06-21 | ウェルマーカー バイオ カンパニー リミテッド | Ron変異が関与する非小細胞肺がんの予防又は治療用医薬組成物及びその使用方法 |
| US20230202992A1 (en) * | 2020-05-18 | 2023-06-29 | Wellmarker Bio Co., Ltd. | Pharmaceutical composition for preventing or treating small-cell lung cancer associated with ron mutants and method using same |
| KR20210142555A (ko) * | 2020-05-18 | 2021-11-25 | 웰마커바이오 주식회사 | Ron 돌연변이와 관련된 췌장암 예방 또는 치료용 약학 조성물 및 이를 이용한 방법 |
| KR20220152155A (ko) * | 2021-05-07 | 2022-11-15 | 웰마커바이오 주식회사 | Ron 돌연변이와 관련된 담도암 예방 또는 치료용 약학 조성물 |
| KR20220170766A (ko) * | 2021-06-22 | 2022-12-30 | 주식회사 엘지화학 | 단백질 키나아제 억제제로서의 신규한 화합물 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009526761A (ja) * | 2006-01-30 | 2009-07-23 | アレイ バイオファーマ、インコーポレイテッド | ヘテロ二環式チオフェン化合物および使用の方法 |
| JP2009539878A (ja) * | 2006-06-08 | 2009-11-19 | アレイ バイオファーマ、インコーポレイテッド | キノリン化合物および使用方法 |
| SI2089364T1 (sl) * | 2006-11-08 | 2013-10-30 | Bristol-Myers Squibb Company | Spojine piridinona |
| EP2423208A1 (en) * | 2010-08-28 | 2012-02-29 | Lead Discovery Center GmbH | Pharmaceutically active compounds as Axl inhibitors |
| JP2014513724A (ja) * | 2011-05-16 | 2014-06-05 | オーエスアイ・ファーマシューティカルズ,エルエルシー | 融合二環キナーゼ阻害剤 |
| CN102816175B (zh) * | 2011-06-09 | 2015-12-16 | 上海汇伦生命科技有限公司 | 一种杂环并吡啶酮类化合物,其中间体、制备方法和用途 |
| WO2013022519A1 (en) * | 2011-08-10 | 2013-02-14 | Merck Patent Gmbh | Pyrido-pyrimidine derivatives |
| DK2820009T3 (en) | 2012-03-01 | 2018-04-16 | Array Biopharma Inc | Serine / threonine kinase inhibitors |
| WO2014038881A2 (ko) * | 2012-09-06 | 2014-03-13 | 씨제이제일제당 (주) | 피리돈 유도체를 포함하는 단백질 키나제 억제제 |
| CN103965107B (zh) * | 2013-02-06 | 2016-08-17 | 沈阳药科大学 | 2-芳基取代喹啉类化合物及其用途 |
| US20150299219A1 (en) * | 2014-04-22 | 2015-10-22 | Calitor Sciences, Llc | Bicyclic pyrazolone compounds and methods of use |
| US11946934B2 (en) * | 2014-09-03 | 2024-04-02 | Wellmarker Bio Co., Ltd. | Biomarker for predicting the sensitivity to a protein kinase inhibitor and a use thereof |
| ES2749726T3 (es) * | 2014-12-25 | 2020-03-23 | Ono Pharmaceutical Co | Derivado de quinolina |
| US11623923B2 (en) * | 2017-11-24 | 2023-04-11 | Medshine Discovery, Inc. | Uracil compound as c-MET/AXL inhibitor |
| CN108314682A (zh) * | 2018-01-31 | 2018-07-24 | 江西科技师范大学 | 6,7-双取代-4-芳杂喹啉类化合物的制备及应用 |
| WO2019182274A1 (en) * | 2018-03-08 | 2019-09-26 | Wellmarker Bio Co., Ltd. | Thienopyridine derivatives and pharmaceutical composition comprising same |
| CN109096250A (zh) * | 2018-09-25 | 2018-12-28 | 辽宁大学 | 含哒嗪酮的4-苯氧基吡啶类化合物及其应用 |
| KR20210111711A (ko) * | 2020-03-03 | 2021-09-13 | 웰마커바이오 주식회사 | Kras 돌연변이 및 활성화된 ron이 존재하는 암의 예방 또는 치료용 약학 조성물 |
-
2020
- 2020-08-03 US US17/596,388 patent/US20220235064A1/en not_active Abandoned
- 2020-08-03 JP JP2022506745A patent/JP2022543250A/ja active Pending
- 2020-08-03 EP EP20849599.4A patent/EP4011885A4/en not_active Withdrawn
- 2020-08-03 KR KR1020200096979A patent/KR20210015730A/ko not_active Ceased
- 2020-08-03 WO PCT/KR2020/010204 patent/WO2021025407A1/ko not_active Ceased
- 2020-08-03 CN CN202080056144.2A patent/CN114206883A/zh active Pending
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