JP2022535577A5 - - Google Patents

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Publication number
JP2022535577A5
JP2022535577A5 JP2021572409A JP2021572409A JP2022535577A5 JP 2022535577 A5 JP2022535577 A5 JP 2022535577A5 JP 2021572409 A JP2021572409 A JP 2021572409A JP 2021572409 A JP2021572409 A JP 2021572409A JP 2022535577 A5 JP2022535577 A5 JP 2022535577A5
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JP
Japan
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JP2021572409A
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Japanese (ja)
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JP7541538B2 (ja
JPWO2020247475A5 (https=
JP2022535577A (ja
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JP2021572409A 2019-06-05 2020-06-03 癌を処置するためのprc2阻害剤としてのイミダゾ[1,2-c]ピリミジン誘導体 Active JP7541538B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962857515P 2019-06-05 2019-06-05
US62/857,515 2019-06-05
PCT/US2020/035891 WO2020247475A1 (en) 2019-06-05 2020-06-03 Imidazo[1,2-c]pyrimidine derivatives as prc2 inhibitors for treating cancer

Publications (4)

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JP2022535577A JP2022535577A (ja) 2022-08-09
JPWO2020247475A5 JPWO2020247475A5 (https=) 2023-05-08
JP2022535577A5 true JP2022535577A5 (https=) 2023-05-08
JP7541538B2 JP7541538B2 (ja) 2024-08-28

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JP2021572409A Active JP7541538B2 (ja) 2019-06-05 2020-06-03 癌を処置するためのprc2阻害剤としてのイミダゾ[1,2-c]ピリミジン誘導体

Country Status (9)

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US (2) US12252493B2 (https=)
EP (1) EP3980422A1 (https=)
JP (1) JP7541538B2 (https=)
KR (1) KR20220027933A (https=)
CN (1) CN114269748A (https=)
AU (1) AU2020288563A1 (https=)
CA (1) CA3142711A1 (https=)
IL (1) IL288529A (https=)
WO (1) WO2020247475A1 (https=)

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DK3746446T3 (da) 2018-01-31 2022-06-27 Mirati Therapeutics Inc PRC2-inhibitorer
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US12252493B2 (en) 2019-06-05 2025-03-18 Mirati Therapeutics, Inc. Imidazo[1,2-c]pyrimidine derivatives as PRC2 inhibitors for treating cancer
CN114907385A (zh) * 2021-02-10 2022-08-16 上海青煜医药科技有限公司 氮杂芳基化合物、其制备方法及应用
WO2023016511A1 (zh) * 2021-08-11 2023-02-16 上海青煜医药科技有限公司 氮杂芳基化合物、其制备方法及应用
WO2023049723A1 (en) * 2021-09-24 2023-03-30 Oric Pharmaceuticals, Inc. Prc2 inhibitors for use in treating blood disorders
EP4404932A4 (en) * 2021-09-24 2025-07-23 Oric Pharmaceuticals Inc PRC2 INHIBITORS FOR USE IN THE TREATMENT OF BLOOD DISORDERS
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IL326327A (en) * 2023-08-04 2026-04-01 Oric Pharmaceuticals Inc Prostate cancer treatment

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