JP2022530866A5 - - Google Patents

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Publication number
JP2022530866A5
JP2022530866A5 JP2021562339A JP2021562339A JP2022530866A5 JP 2022530866 A5 JP2022530866 A5 JP 2022530866A5 JP 2021562339 A JP2021562339 A JP 2021562339A JP 2021562339 A JP2021562339 A JP 2021562339A JP 2022530866 A5 JP2022530866 A5 JP 2022530866A5
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JP
Japan
Prior art keywords
cancer
heterocyclyl
pharmaceutically acceptable
cancers
carcinoma
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JP2021562339A
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English (en)
Japanese (ja)
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JP2022530866A (ja
JP7624404B2 (ja
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Priority claimed from PCT/US2020/029118 external-priority patent/WO2020219448A1/en
Publication of JP2022530866A publication Critical patent/JP2022530866A/ja
Publication of JP2022530866A5 publication Critical patent/JP2022530866A5/ja
Application granted granted Critical
Publication of JP7624404B2 publication Critical patent/JP7624404B2/ja
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JP2021562339A 2019-04-22 2020-04-21 Ｐｒｃ２阻害剤としてのナフチリジン誘導体 Active JP7624404B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962836840P 2019-04-22 2019-04-22
US62/836,840 2019-04-22
PCT/US2020/029118 WO2020219448A1 (en) 2019-04-22 2020-04-21 Naphthyridine derivatives as prc2 inhibitors

Publications (3)

Publication Number Publication Date
JP2022530866A JP2022530866A (ja) 2022-07-04
JP2022530866A5 true JP2022530866A5 (https=) 2023-04-19
JP7624404B2 JP7624404B2 (ja) 2025-01-30

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JP2021562339A Active JP7624404B2 (ja) 2019-04-22 2020-04-21 Ｐｒｃ２阻害剤としてのナフチリジン誘導体

Country Status (4)

Country Link
US (1) US12421228B2 (https=)
EP (1) EP3959214A1 (https=)
JP (1) JP7624404B2 (https=)
WO (1) WO2020219448A1 (https=)

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US12421228B2 (en) 2019-04-22 2025-09-23 Mirati Therapeutics, Inc. Naphthyridine derivatives as PRC2 inhibitors
EP3980422A1 (en) 2019-06-05 2022-04-13 Mirati Therapeutics, Inc. Imidazo[1,2-c]pyrimidine derivatives as prc2 inhibitors for treating cancer
WO2022184116A1 (zh) * 2021-03-05 2022-09-09 江苏先声药业有限公司 新型sos1抑制剂及其制备方法和应用
CN113861172B (zh) * 2021-09-23 2024-04-16 北京大学深圳研究生院 基于苯并五元杂环的双极性荧光材料及其制备方法与有机电致发光器件
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WO2025117697A1 (en) * 2023-11-29 2025-06-05 Riboscience Llc 7-aza bicyclic heteroaryl derivatives as ectonucleotide pyrophosphatase phosphodiesterase 1 inhibitors

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