JP2022530985A5 - - Google Patents
Info
- Publication number
- JP2022530985A5 JP2022530985A5 JP2021564826A JP2021564826A JP2022530985A5 JP 2022530985 A5 JP2022530985 A5 JP 2022530985A5 JP 2021564826 A JP2021564826 A JP 2021564826A JP 2021564826 A JP2021564826 A JP 2021564826A JP 2022530985 A5 JP2022530985 A5 JP 2022530985A5
- Authority
- JP
- Japan
- Prior art keywords
- methylene
- succinate
- oxy
- oxobutanoyl
- methylene succinate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP19172051 | 2019-04-30 | ||
| EP19172051.5 | 2019-04-30 | ||
| EP19189910 | 2019-08-02 | ||
| EP19189910.3 | 2019-08-02 | ||
| EP19217846 | 2019-12-19 | ||
| EP19217846.5 | 2019-12-19 | ||
| EP20162494.7 | 2020-03-11 | ||
| EP20162494 | 2020-03-11 | ||
| PCT/GB2020/051060 WO2020222011A1 (en) | 2019-04-30 | 2020-04-30 | Itaconic acid derivatives and uses thereof in treating an inflammatory disease or a disease associated with an undesirable immune response |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022530985A JP2022530985A (ja) | 2022-07-05 |
| JP2022530985A5 true JP2022530985A5 (https=) | 2023-03-27 |
Family
ID=70480305
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021564826A Ceased JP2022530985A (ja) | 2019-04-30 | 2020-04-30 | 炎症性疾患または望ましくない免疫応答に関連する疾患の治療におけるイタコン酸誘導体およびその使用 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US12390437B2 (https=) |
| EP (2) | EP3962602B1 (https=) |
| JP (1) | JP2022530985A (https=) |
| KR (1) | KR20220002952A (https=) |
| CN (1) | CN113825740A (https=) |
| AU (1) | AU2020264773A1 (https=) |
| BR (1) | BR112021021301A2 (https=) |
| CA (1) | CA3135991A1 (https=) |
| CO (1) | CO2021015538A2 (https=) |
| CR (1) | CR20210578A (https=) |
| DO (1) | DOP2021000219A (https=) |
| EC (1) | ECSP21086530A (https=) |
| IL (1) | IL287444B2 (https=) |
| JO (3) | JOP20210291A1 (https=) |
| MA (2) | MA55796A (https=) |
| MX (1) | MX2021013299A (https=) |
| PE (1) | PE20220762A1 (https=) |
| SG (1) | SG11202110624YA (https=) |
| WO (2) | WO2020222010A1 (https=) |
Families Citing this family (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SMT202400306T1 (it) | 2018-03-30 | 2024-09-16 | Incyte Corp | Trattamento dell'idrosadenite suppurativa utilizzando inibitori di jak. |
| HUE065501T2 (hu) | 2018-08-20 | 2024-05-28 | Janssen Pharmaceutica Nv | A KEAP1-NRF2 protein-protein kölcsönhatás inhibitorok |
| WO2020232247A1 (en) | 2019-05-14 | 2020-11-19 | Provention Bio, Inc. | Methods and compositions for preventing type 1 diabetes |
| PE20230405A1 (es) * | 2019-10-29 | 2023-03-07 | Univ Johns Hopkins | Profarmacos de itaconato e itaconato de metilo desarrollo o investigacion patrocinados por el gobierno |
| BR112022008310A2 (pt) | 2019-10-29 | 2022-08-09 | Univ Johns Hopkins | Uso de itaconato e seus derivados/análogos para induzir crescimento capilar |
| IL298999A (en) | 2020-06-11 | 2023-02-01 | Provention Bio Inc | Methods and compositions for the prevention of type 1 diabetes |
| EP4192821A1 (en) | 2020-08-05 | 2023-06-14 | Sitryx Therapeutics Limited | Alpha,beta unsaturated methacrylic esters with anti-inflammatory properties |
| EP4237404A1 (en) * | 2020-10-29 | 2023-09-06 | Sitryx Therapeutics Limited | Novel compounds |
| CN114681450A (zh) * | 2020-12-28 | 2022-07-01 | 苏州澳宗生物科技有限公司 | 依达拉奉、衍生物、药学上可接受的盐、前药或多晶型物的新用途 |
| CN112812052B (zh) * | 2021-02-02 | 2023-12-01 | 成都阿奇生物医药科技有限公司 | 一种治疗溃疡性结肠炎的化合物及其制备方法和用途 |
| WO2022223778A1 (en) * | 2021-04-23 | 2022-10-27 | Helmholtz-Zentrum für Infektionsforschung GmbH | Citraconic acid and derivatives thereof for use as a medicament |
| EP4330231A1 (en) | 2021-04-26 | 2024-03-06 | Sitryx Therapeutics Limited | 2-methylene-4-oxo-butanoic acid drivatives for the treatment of inflammation |
| JP2024520444A (ja) | 2021-05-24 | 2024-05-24 | プロヴェンション・バイオ・インコーポレイテッド | 1型糖尿病を治療するための方法 |
| EP4359390A1 (en) | 2021-06-22 | 2024-05-01 | Sitryx Therapeutics Limited | Acrylamide derivatives useful as anti-inflammatory agents |
| US20240360067A1 (en) | 2021-08-11 | 2024-10-31 | Sitryx Therapeutics Limited | Derivatives of itaconic acid and their use as anti-inflammatory agents |
| GB202203755D0 (en) * | 2022-03-17 | 2022-05-04 | Imperial College Innovations Ltd | Treatment or prevention of respiratory diseases characterised by, or involving, lung fibrosis |
| CN114557993B (zh) * | 2022-03-22 | 2023-05-12 | 中南大学湘雅三医院 | 4-衣康酸辛酯在制备胰腺提取胰岛前的注射制剂中的应用 |
| CN115969790B (zh) * | 2022-05-27 | 2024-09-06 | 哈尔滨医科大学 | 一种肺炎治疗药物pfc@4-oi及其制备方法与应用 |
| CN116139117A (zh) * | 2022-05-31 | 2023-05-23 | 西南医科大学附属医院 | 衣康酸及其衍生物在防治阿霉素诱导的心脏毒性中的应用 |
| AU2023287566A1 (en) | 2022-06-22 | 2025-01-16 | Sitryx Therapeutics Limited | Oxadiazole derivatives, preparation process thereof and their use in treating inflammatory diseases |
| CN115518060A (zh) * | 2022-09-30 | 2022-12-27 | 中国人民解放军空军军医大学 | 衣康酸及其衍生物在治疗白癜风药物上的应用及其治疗白癜风的药物 |
| WO2024089421A1 (en) | 2022-10-25 | 2024-05-02 | Sitryx Therapeutics Limited | Tetrazole derivatives |
| CN120712258A (zh) | 2022-12-15 | 2025-09-26 | 西特瑞治疗有限公司 | 用于治疗或预防炎性疾病或与不良免疫反应相关的疾病的取代吡啶类化合物 |
| CN116019975A (zh) * | 2023-01-06 | 2023-04-28 | 天津市天津医院 | 一种负载抗炎因子4-辛基衣康酸可注射水凝胶及其制备方法和应用 |
| CN117205194A (zh) * | 2023-05-10 | 2023-12-12 | 苏州大学 | 衣康酸或其衍生物在制备预防或治疗急性移植物抗宿主病药物中的应用 |
| CN117530944A (zh) * | 2023-12-25 | 2024-02-09 | 中国医学科学院放射医学研究所 | 衣康酸四辛酯在制备防治放射性肠损伤药物中的应用 |
| CN117599037A (zh) * | 2023-12-25 | 2024-02-27 | 中国医学科学院放射医学研究所 | 衣康酸四辛酯在制备防治辐射诱导骨髓抑制药物中的应用 |
| WO2025153532A1 (en) | 2024-01-16 | 2025-07-24 | NodThera Limited | Nlrp3 inhibitors and glp-1 agonists combination therapies |
| WO2026008955A1 (en) * | 2024-07-03 | 2026-01-08 | Cambridge Enterprise Limited | Treatment or prevention of central nervous system (cns) disorder |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4743657A (en) * | 1986-03-17 | 1988-05-10 | Milliken Research Corporation | Method for preparing polymer bound stabilizers made from non-homopolymerizable stabilizers |
| US5422349A (en) * | 1992-08-14 | 1995-06-06 | G. D. Seale & Co. | Morpholino-oxazinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension |
| KR100538968B1 (ko) * | 1997-02-18 | 2006-07-11 | 후지 샤신 필름 가부시기가이샤 | 포지티브감광성조성물 |
| US6235787B1 (en) * | 1997-06-30 | 2001-05-22 | Hoffmann-La Roche Inc. | Hydrazine derivatives |
| JP2001354625A (ja) * | 2000-04-12 | 2001-12-25 | Dainippon Ink & Chem Inc | 新規なイタコン酸エステル及びその製造方法 |
| JP4102014B2 (ja) * | 2000-10-03 | 2008-06-18 | 富士フイルム株式会社 | 感光性平版印刷版 |
| US6777155B2 (en) * | 2000-10-03 | 2004-08-17 | Fuji Photo Film Co., Ltd. | Photosensitive lithographic printing plate |
| JP3925288B2 (ja) * | 2002-04-22 | 2007-06-06 | チッソ株式会社 | イタコン酸誘導体およびその重合体 |
| JP4133376B2 (ja) * | 2002-09-03 | 2008-08-13 | 信越化学工業株式会社 | 高分子化合物及びポジ型レジスト材料並びにこれを用いたパターン形成方法 |
| JP2004315791A (ja) * | 2003-03-28 | 2004-11-11 | Tokyo Ohka Kogyo Co Ltd | ジカルボン酸モノエステル化合物およびその製造方法ならびに重合体 |
| JP2007086285A (ja) * | 2005-09-21 | 2007-04-05 | Fujifilm Corp | レジスト組成物及びそれを用いたパターン形成方法 |
| EP2145920A1 (en) | 2008-07-15 | 2010-01-20 | Lanxess Deutschland GmbH | Vulcanizable polymer compositions |
| EP2373617B1 (de) | 2008-12-04 | 2015-02-25 | Basf Se | Mischungen aus itaconsäure oder itaconsäurederivaten und primären aminen zur herstellung von 1,3- und 1,4-alkylmethylpyrrolidonen |
| JP5526693B2 (ja) * | 2009-10-09 | 2014-06-18 | 日油株式会社 | 感光性樹脂組成物およびその用途 |
| EP2423178A1 (en) | 2010-07-28 | 2012-02-29 | Chemo Ibérica, S.A. | Process for the production of sitagliptin |
| JP5732306B2 (ja) * | 2011-04-20 | 2015-06-10 | 東京応化工業株式会社 | 化合物、高分子化合物、酸発生剤、レジスト組成物、レジストパターン形成方法 |
| KR102085557B1 (ko) | 2013-03-14 | 2020-03-06 | 엘커메스 파마 아일랜드 리미티드 | 푸마레이트의 프로드럭 및 다양한 질환을 치료하는데 있어서의 이들의 용도 |
| EP3416634A4 (en) | 2016-02-15 | 2019-10-09 | Artyomov, Maxim | IMMUNOMODULATORY AGENTS AND METHOD FOR USE THEREOF |
| US10047100B2 (en) | 2016-04-08 | 2018-08-14 | Regents Of The University Of Minnesota | Compounds from renewable resources |
| WO2019036509A1 (en) * | 2017-08-14 | 2019-02-21 | Washington University | METHODS AND COMPOSITIONS FOR TREATING DISEASES ASSOCIATED WITH CANCER, INFLAMMATION OR IMMUNE RESPONSE |
| WO2019064827A1 (ja) * | 2017-09-26 | 2019-04-04 | Jnc株式会社 | 重合性極性化合物、液晶組成物および液晶表示素子 |
| US12060310B2 (en) | 2018-06-29 | 2024-08-13 | Ergon Pharmaceuticals Llc | Compositions and methods of using itaconic acid derivatives |
| CN110731955B (zh) | 2019-10-28 | 2023-05-02 | 中山大学 | 衣康酸二甲酯在预防和治疗溃疡性结肠炎及其癌变中的应用 |
| MX2022007846A (es) | 2019-12-23 | 2022-07-19 | Sitryx Therapeutics Ltd | Derivados carboxi con propiedades antiinflamatorias. |
-
2020
- 2020-04-30 MX MX2021013299A patent/MX2021013299A/es unknown
- 2020-04-30 US US17/606,884 patent/US12390437B2/en active Active
- 2020-04-30 MA MA055796A patent/MA55796A/fr unknown
- 2020-04-30 EP EP20723186.1A patent/EP3962602B1/en active Active
- 2020-04-30 IL IL287444A patent/IL287444B2/en unknown
- 2020-04-30 AU AU2020264773A patent/AU2020264773A1/en not_active Abandoned
- 2020-04-30 JP JP2021564826A patent/JP2022530985A/ja not_active Ceased
- 2020-04-30 CR CR20210578A patent/CR20210578A/es unknown
- 2020-04-30 KR KR1020217036775A patent/KR20220002952A/ko not_active Ceased
- 2020-04-30 EP EP20723187.9A patent/EP3962888A1/en not_active Withdrawn
- 2020-04-30 PE PE2021001799A patent/PE20220762A1/es unknown
- 2020-04-30 MA MA055795A patent/MA55795A/fr unknown
- 2020-04-30 SG SG11202110624YA patent/SG11202110624YA/en unknown
- 2020-04-30 CN CN202080032325.1A patent/CN113825740A/zh active Pending
- 2020-04-30 CA CA3135991A patent/CA3135991A1/en active Pending
- 2020-04-30 BR BR112021021301A patent/BR112021021301A2/pt not_active Application Discontinuation
- 2020-04-30 WO PCT/GB2020/051059 patent/WO2020222010A1/en not_active Ceased
- 2020-04-30 WO PCT/GB2020/051060 patent/WO2020222011A1/en not_active Ceased
-
2021
- 2021-10-28 DO DO2021000219A patent/DOP2021000219A/es unknown
- 2021-10-28 JO JOP/2021/0291A patent/JOP20210291A1/ar unknown
- 2021-10-28 JO JOP/2021/0290A patent/JOP20210290A1/ar unknown
- 2021-10-28 JO JOP/2021/0292A patent/JOP20210292A1/ar unknown
- 2021-11-18 CO CONC2021/0015538A patent/CO2021015538A2/es unknown
- 2021-11-30 EC ECSENADI202186530A patent/ECSP21086530A/es unknown
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