JP2022521119A - 組織の灌流の増加における使用のためのイノシトールリン酸化合物 - Google Patents

組織の灌流の増加における使用のためのイノシトールリン酸化合物 Download PDF

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JP2022521119A
JP2022521119A JP2021532911A JP2021532911A JP2022521119A JP 2022521119 A JP2022521119 A JP 2022521119A JP 2021532911 A JP2021532911 A JP 2021532911A JP 2021532911 A JP2021532911 A JP 2021532911A JP 2022521119 A JP2022521119 A JP 2022521119A
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JP2022521119A5 (https=
JPWO2020157362A5 (https=
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バッシッシ，モハンマド・フィラス
ロカ，カロリーナ サルセド
ベスタルド，フアン ペレロ
レイネス，ミゲル・ダビド フェレール
フェレール，マリア・デル・マール ペレス
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サニフィット・セラピューティクス・ソシエダッド・アノニマ
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/08—Esters of oxyacids of phosphorus
    • C07F9/09—Esters of phosphoric acids
    • C07F9/117—Esters of phosphoric acids with cycloaliphatic alcohols
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/661—Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • A61K31/6615—Compounds having two or more esterified phosphorus acid groups, e.g. inositol triphosphate, phytic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2021532911A 2019-01-30 2020-01-30 組織の灌流の増加における使用のためのイノシトールリン酸化合物 Pending JP2022521119A (ja)

Priority Applications (1)

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JP2024158993A JP2024175025A (ja) 2019-01-30 2024-09-13 組織の灌流の増加における使用のためのイノシトールリン酸化合物

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EP19382061.0 2019-01-30
EP19382061 2019-01-30
US201962913259P 2019-10-10 2019-10-10
US62/913,259 2019-10-10
PCT/ES2020/070070 WO2020157362A1 (en) 2019-01-30 2020-01-30 Inositol phosphate compounds for use in increasing tissular perfusion

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JP2024158993A Division JP2024175025A (ja) 2019-01-30 2024-09-13 組織の灌流の増加における使用のためのイノシトールリン酸化合物

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JP2022521119A true JP2022521119A (ja) 2022-04-06
JP2022521119A5 JP2022521119A5 (https=) 2022-09-14
JPWO2020157362A5 JPWO2020157362A5 (https=) 2022-09-14

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JP2024158993A Pending JP2024175025A (ja) 2019-01-30 2024-09-13 組織の灌流の増加における使用のためのイノシトールリン酸化合物

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US (2) US20220000889A1 (https=)
EP (1) EP3917535A1 (https=)
JP (2) JP2022521119A (https=)
KR (1) KR20210148078A (https=)
CN (1) CN113365636A (https=)
AU (1) AU2020213713B2 (https=)
BR (1) BR112021014897A2 (https=)
CA (1) CA3130735A1 (https=)
IL (1) IL285084A (https=)
MX (1) MX2021008966A (https=)
WO (1) WO2020157362A1 (https=)

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Publication number Priority date Publication date Assignee Title
AU2018445164B2 (en) 2018-10-11 2025-05-29 Vifor (International) Ltd. Inositol phosphates for the treatment of ectopic calcification
MX2023005931A (es) * 2020-11-20 2023-08-03 Vifor Int Ag Analogos de hexakisfosfato de inositol para el tratamiento de enfermedades renales asociadas con la calcificacion.
WO2024047037A1 (en) 2022-08-30 2024-03-07 ETH Zürich Compositions for parenteral sustained release delivery of hydrophilic drugs

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JP2003507430A (ja) * 1999-08-25 2003-02-25 ジーエムピー カンパニーズ，インコーポレーテッド 哺乳動物中で酸素運搬を向上する薬剤
JP2016514119A (ja) * 2013-03-15 2016-05-19 ラボラトリス サニフィット，エセ．エレ． 腎不全を患っている患者におけるｃ−ｏ−ｐ結合を含む誘導体の使用
WO2017098047A1 (en) * 2015-12-11 2017-06-15 ETH Zürich Inositol derivatives for use in pathological crystallization

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US5582837A (en) 1992-03-25 1996-12-10 Depomed, Inc. Alkyl-substituted cellulose-based sustained-release oral drug dosage forms
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ES2270982T3 (es) 2000-02-04 2007-04-16 Depomed, Inc. Forma de dosificacion de nucleo y carcasa que se aproxima a una liberacion del farmaco de orden cero.
US6488962B1 (en) 2000-06-20 2002-12-03 Depomed, Inc. Tablet shapes to enhance gastric retention of swellable controlled-release oral dosage forms
US20020142995A1 (en) * 2000-08-01 2002-10-03 Nicolau Yves Claude Ammonium salts of hemoglobin allosteric effectors, and uses thereof
WO2002010177A1 (en) * 2000-08-01 2002-02-07 Gmp Companies, Inc. Ammonium salts of inositol hexaphosphate and uses thereof
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JP3678144B2 (ja) 2000-12-22 2005-08-03 ウシオ電機株式会社 フィルム回路基板の周辺露光装置
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JP2016514119A (ja) * 2013-03-15 2016-05-19 ラボラトリス サニフィット，エセ．エレ． 腎不全を患っている患者におけるｃ−ｏ−ｐ結合を含む誘導体の使用
WO2017098047A1 (en) * 2015-12-11 2017-06-15 ETH Zürich Inositol derivatives for use in pathological crystallization

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CN113365636A (zh) 2021-09-07
AU2020213713B2 (en) 2025-08-21
US20220000889A1 (en) 2022-01-06
CA3130735A1 (en) 2020-08-06
MX2021008966A (es) 2021-11-04
US20230248749A1 (en) 2023-08-10
EP3917535A1 (en) 2021-12-08
AU2020213713A1 (en) 2021-07-22
IL285084A (en) 2021-09-30
JP2024175025A (ja) 2024-12-17
KR20210148078A (ko) 2021-12-07
BR112021014897A2 (pt) 2021-09-28
WO2020157362A1 (en) 2020-08-06

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