JP2022502431A5 - - Google Patents
Info
- Publication number
- JP2022502431A5 JP2022502431A5 JP2021517292A JP2021517292A JP2022502431A5 JP 2022502431 A5 JP2022502431 A5 JP 2022502431A5 JP 2021517292 A JP2021517292 A JP 2021517292A JP 2021517292 A JP2021517292 A JP 2021517292A JP 2022502431 A5 JP2022502431 A5 JP 2022502431A5
- Authority
- JP
- Japan
- Prior art keywords
- integer
- formula
- alkyl
- ch2ch2o
- cycloalkanediyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024106489A JP7830555B2 (ja) | 2018-09-27 | 2024-07-01 | スルホマレイミドに基づくリンカーおよび対応する複合体 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP18306270 | 2018-09-27 | ||
| EP18306270.2 | 2018-09-27 | ||
| PCT/IB2019/001114 WO2020065408A1 (en) | 2018-09-27 | 2019-09-27 | Sulfomaleimide-based linkers and corresponding conjugates |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024106489A Division JP7830555B2 (ja) | 2018-09-27 | 2024-07-01 | スルホマレイミドに基づくリンカーおよび対応する複合体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022502431A JP2022502431A (ja) | 2022-01-11 |
| JP2022502431A5 true JP2022502431A5 (enExample) | 2022-10-11 |
Family
ID=63857832
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021517292A Pending JP2022502431A (ja) | 2018-09-27 | 2019-09-27 | スルホマレイミドに基づくリンカーおよび対応する複合体 |
| JP2024106489A Active JP7830555B2 (ja) | 2018-09-27 | 2024-07-01 | スルホマレイミドに基づくリンカーおよび対応する複合体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024106489A Active JP7830555B2 (ja) | 2018-09-27 | 2024-07-01 | スルホマレイミドに基づくリンカーおよび対応する複合体 |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US12011485B2 (enExample) |
| EP (1) | EP3856258B1 (enExample) |
| JP (2) | JP2022502431A (enExample) |
| KR (1) | KR102858995B1 (enExample) |
| CN (1) | CN113453724B (enExample) |
| AU (1) | AU2019350536B2 (enExample) |
| BR (1) | BR112021005655A2 (enExample) |
| CA (1) | CA3113378C (enExample) |
| MX (1) | MX2021003295A (enExample) |
| WO (1) | WO2020065408A1 (enExample) |
| ZA (1) | ZA202101990B (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201908886D0 (en) * | 2019-06-20 | 2019-08-07 | Almac Discovery Ltd | Anthracycline derivatives |
| CN118955614B (zh) * | 2022-07-05 | 2025-12-30 | 上海药明合联生物技术有限公司 | 偶联连接子 |
| CN120957756A (zh) * | 2023-05-12 | 2025-11-14 | 四川科伦博泰生物医药股份有限公司 | 稠环化合物及其制备方法和用途 |
| CN119751374A (zh) * | 2024-12-09 | 2025-04-04 | 中国科学院水生生物研究所 | 高抑菌活性、低生态毒性的异噻唑啉酮类化合物及其制备方法和应用 |
Family Cites Families (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4127687A (en) * | 1976-07-19 | 1978-11-28 | Rohm And Haas Company | Prevention of fouling of marine structures such as boat hulls |
| IL162181A (en) | 1988-12-28 | 2006-04-10 | Pdl Biopharma Inc | A method of producing humanized immunoglubulin, and polynucleotides encoding the same |
| US5530101A (en) | 1988-12-28 | 1996-06-25 | Protein Design Labs, Inc. | Humanized immunoglobulins |
| GB9014932D0 (en) | 1990-07-05 | 1990-08-22 | Celltech Ltd | Recombinant dna product and method |
| JPH04248881A (ja) | 1991-01-25 | 1992-09-04 | Mitsubishi Kasei Corp | 顔料分散型水性記録液 |
| JPH04261476A (ja) | 1991-02-15 | 1992-09-17 | Mitsubishi Kasei Corp | インクジェットプリンター用クリーニング液 |
| WO1994004679A1 (en) | 1991-06-14 | 1994-03-03 | Genentech, Inc. | Method for making humanized antibodies |
| JPH05244982A (ja) | 1991-12-06 | 1993-09-24 | Sumitomo Chem Co Ltd | 擬人化ｂ−ｂ１０ |
| US5639641A (en) | 1992-09-09 | 1997-06-17 | Immunogen Inc. | Resurfacing of rodent antibodies |
| TW258789B (enExample) * | 1992-09-28 | 1995-10-01 | Rohm & Haas | |
| KR20070110327A (ko) | 2005-03-08 | 2007-11-16 | 미쓰비시 가가꾸 가부시키가이샤 | 이방성 색소 필름용 조성물, 이방성 색소 필름 및 편광소자 |
| JP2007025635A (ja) * | 2005-06-17 | 2007-02-01 | Fujitsu Hitachi Plasma Display Ltd | プラズマディスプレイ装置及びその処理方法 |
| US20060293374A1 (en) | 2005-06-24 | 2006-12-28 | Beers Scott A | Substituted isothiazolones |
| CN101397280A (zh) | 2008-11-04 | 2009-04-01 | 东华大学 | 反应性异噻唑啉酮类抗菌整理剂的制备方法 |
| DE102012213321A1 (de) | 2012-07-30 | 2014-01-30 | Robert Bosch Gmbh | Verfahren und Vorrichtung zum Betreiben eines Fahrzeugs |
| FR3005051A1 (fr) | 2013-04-25 | 2014-10-31 | Pf Medicament | Derives de la dolastatine 10 et d'auristatines |
| JP2016524593A (ja) | 2013-04-29 | 2016-08-18 | メモリアル スローン−ケタリング キャンサー センター | セカンドメッセンジャーのシグナル伝達を変えるための組成物及び方法 |
| WO2014197866A1 (en) * | 2013-06-06 | 2014-12-11 | Igenica Biotherapeutics, Inc. | Modified antibodies and related compounds, compositions, and methods of use |
| US10533010B2 (en) | 2014-03-27 | 2020-01-14 | Vanderbilt University | Substituted indole Mcl-1 inhibitors |
| CN106459204B (zh) | 2014-04-25 | 2021-02-02 | 皮埃尔法布雷医药公司 | Igf-1r抗体及其作为定位载体用于治疗癌症的用途 |
| MX378281B (es) * | 2014-04-25 | 2025-03-10 | Pf Medicament | Conjugado farmaco-anticuerpo y su uso para el tratamiento contra el cancer. |
| MA39909B1 (fr) | 2014-04-25 | 2019-05-31 | Pf Medicament | Conjugué anticorps de l'igf-1r-médicament et son utilisation pour le traitement du cancer |
| CN104230916B (zh) | 2014-09-30 | 2020-04-28 | 上海化学试剂研究所有限公司 | 一种异噻唑啉酮类化合物及其制备方法和应用 |
| US20190209704A1 (en) | 2014-10-20 | 2019-07-11 | Igenica Biotherapeutics, Inc. | Novel antibody-drug conjugates and related compounds, compositions and methods of use |
| DK3233882T3 (da) | 2014-12-16 | 2020-01-27 | Kayla Therapeutics | Fluorinerede cykliske dinukleotider til cytokininduktion |
| TWI706958B (zh) | 2015-03-10 | 2020-10-11 | 美商艾杜諾生物科技公司 | 活化「干擾素基因刺激因子」依賴性訊息傳導之組合物及方法 |
| EP3307749A4 (en) * | 2015-06-15 | 2019-06-19 | Hangzhou Dac Biotech Co., Ltd | HYDROPHILIC LINKER FOR CONJUGATION |
| WO2017051254A1 (en) * | 2015-09-25 | 2017-03-30 | Legochem Biosciences, Inc. | Compositions and methods related to anti-egfr antibody drug conjugates |
| US20180369268A1 (en) | 2015-12-16 | 2018-12-27 | Aduro Biotech, Inc. | Methods for identifying inhibitors of "stimulator of interferon gene"- dependent interferon production |
| HK1259487A1 (zh) | 2016-02-04 | 2019-11-29 | Hangzhou Dac Biotech Co. Ltd. | 特定的共轭连接子，特定的免疫共轭物，制造和使用这些共轭物的方法 |
| WO2018100558A2 (en) | 2016-12-01 | 2018-06-07 | Takeda Pharmaceutical Company Limited | Cyclic dinucleotide |
-
2019
- 2019-09-27 CN CN201980077950.5A patent/CN113453724B/zh active Active
- 2019-09-27 AU AU2019350536A patent/AU2019350536B2/en active Active
- 2019-09-27 CA CA3113378A patent/CA3113378C/en active Active
- 2019-09-27 US US17/280,800 patent/US12011485B2/en active Active
- 2019-09-27 WO PCT/IB2019/001114 patent/WO2020065408A1/en not_active Ceased
- 2019-09-27 MX MX2021003295A patent/MX2021003295A/es unknown
- 2019-09-27 JP JP2021517292A patent/JP2022502431A/ja active Pending
- 2019-09-27 KR KR1020217012389A patent/KR102858995B1/ko active Active
- 2019-09-27 BR BR112021005655-6A patent/BR112021005655A2/pt unknown
- 2019-09-27 EP EP19813935.4A patent/EP3856258B1/en active Active
-
2021
- 2021-03-24 ZA ZA2021/01990A patent/ZA202101990B/en unknown
-
2024
- 2024-03-29 US US18/622,613 patent/US20240350657A1/en active Pending
- 2024-07-01 JP JP2024106489A patent/JP7830555B2/ja active Active
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