JP2021531260A5 - - Google Patents
Info
- Publication number
- JP2021531260A5 JP2021531260A5 JP2021500532A JP2021500532A JP2021531260A5 JP 2021531260 A5 JP2021531260 A5 JP 2021531260A5 JP 2021500532 A JP2021500532 A JP 2021500532A JP 2021500532 A JP2021500532 A JP 2021500532A JP 2021531260 A5 JP2021531260 A5 JP 2021531260A5
- Authority
- JP
- Japan
- Prior art keywords
- disorders
- disorder
- methyl
- formula
- alkyl
- Prior art date
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HUP1800248A HU231333B1 (hu) | 2018-07-13 | 2018-07-13 | Spirokromán származékok |
| HUP1800248 | 2018-07-13 | ||
| PCT/IB2019/055948 WO2020012422A1 (en) | 2018-07-13 | 2019-07-12 | Spirochromane derivatives |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2021531260A JP2021531260A (ja) | 2021-11-18 |
| JP2021531260A5 true JP2021531260A5 (https=) | 2022-07-20 |
| JPWO2020012422A5 JPWO2020012422A5 (https=) | 2022-07-20 |
| JP7487167B2 JP7487167B2 (ja) | 2024-05-20 |
Family
ID=89992725
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021500532A Active JP7487167B2 (ja) | 2018-07-13 | 2019-07-12 | スピロクロマン誘導体 |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US20210330650A1 (https=) |
| EP (1) | EP3820869B1 (https=) |
| JP (1) | JP7487167B2 (https=) |
| KR (1) | KR20210033002A (https=) |
| CN (1) | CN112823157B (https=) |
| AR (1) | AR115782A1 (https=) |
| AU (1) | AU2019300514B2 (https=) |
| BR (1) | BR112020026996A2 (https=) |
| CA (1) | CA3104258A1 (https=) |
| CL (1) | CL2021000080A1 (https=) |
| CO (1) | CO2021001216A2 (https=) |
| CU (1) | CU24680B1 (https=) |
| EA (1) | EA202190245A1 (https=) |
| ES (1) | ES2964617T3 (https=) |
| GE (2) | GEAP202315557A (https=) |
| HU (2) | HU231333B1 (https=) |
| IL (1) | IL279938B2 (https=) |
| MX (1) | MX2021000460A (https=) |
| MY (1) | MY206779A (https=) |
| PE (1) | PE20211809A1 (https=) |
| PH (1) | PH12020552183A1 (https=) |
| SG (1) | SG11202012594RA (https=) |
| TW (1) | TWI821321B (https=) |
| WO (1) | WO2020012422A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU231414B1 (hu) | 2018-07-13 | 2023-08-28 | Richter Gedeon Nyrt. | Tiadiazin származékok |
| TWI901650B (zh) | 2020-03-26 | 2025-10-21 | 匈牙利商羅特格登公司 | 啶及吡啶并〔３，４－ｃ〕嗒衍生物 |
| CN115403579A (zh) * | 2021-05-27 | 2022-11-29 | 上海拓界生物医药科技有限公司 | 一种新的螺环衍生物及其用途 |
| HU231691B1 (hu) | 2021-09-29 | 2025-10-28 | Richter Gedeon Nyrt | GABAA ALFA5 receptor modulátor hatású biciklusos aminszármazékok |
| WO2025175249A1 (en) | 2024-02-14 | 2025-08-21 | Olema Pharmaceuticals, Inc. | Estrogen receptor modulators and uses thereof |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006016548A1 (ja) | 2004-08-09 | 2006-02-16 | Eisai R & D Management Co., Ltd. | ヘテロ環化合物を含有する新規な抗マラリア剤 |
| NZ566036A (en) | 2005-09-13 | 2010-06-25 | Janssen Pharmaceutica Nv | 2-Aniline-4-aryl substituted thiazole derivatives that modulate the alpha7 nicotinic receptor |
| CN101490056A (zh) * | 2006-05-17 | 2009-07-22 | 阿斯利康(瑞典)有限公司 | 烟碱乙酰胆碱受体的配体101 |
| TW200813067A (en) * | 2006-05-17 | 2008-03-16 | Astrazeneca Ab | Nicotinic acetylcholine receptor ligands |
| US20100298314A1 (en) | 2006-12-20 | 2010-11-25 | Schering Corporation | Novel jnk inhibitors |
| MX2010003156A (es) | 2007-10-04 | 2010-04-01 | Hoffmann La Roche | Derivados de aril amida substituida con tetrazol y usos de los mismos. |
| MX2010003155A (es) | 2007-10-04 | 2010-04-01 | Hoffmann La Roche | Derivados de ciclopropil aril amida y uso de los mismos. |
| KR20100124272A (ko) | 2008-02-07 | 2010-11-26 | 아보트 러보러터리즈 | 양성 알로스테릭 조절제로서의 아미드 유도체 및 이의 사용방법 |
| AR070936A1 (es) | 2008-03-19 | 2010-05-12 | Janssen Pharmaceutica Nv | 1,2,4 -triazoles trisustituidos |
| EP2110377A1 (en) * | 2008-04-15 | 2009-10-21 | DAC S.r.l. | Spirocyclic derivatives as histone deacetylase inhibitors |
| WO2009127678A1 (en) * | 2008-04-17 | 2009-10-22 | Glaxo Group Limited | Indoles as modulators of nicotinic acetylcholin receptor subtype alpha-71 |
| JP5486591B2 (ja) | 2008-05-09 | 2014-05-07 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | アセチルコリン受容体モジュレーターとしての三置換ピラゾール |
| CA2725940A1 (en) | 2008-05-30 | 2009-12-23 | Merck Sharp & Dohme Corp. | Novel substituted azabenzoxazoles |
| EP3795573B1 (en) | 2009-12-31 | 2022-07-06 | Hutchison Medipharma Limited | Certain triazolopyrazines, compositions thereof and methods of use therefor |
| WO2012042915A1 (en) | 2010-10-01 | 2012-04-05 | Raqualia Pharma Inc. | Sulfamoyl benzoic acid heterobicyclic derivatives as trpm8 antagonists |
| US9617210B2 (en) * | 2013-03-13 | 2017-04-11 | Lupin Limited | Pyrrole derivatives as alpha 7 NACHR modulators |
| AR107928A1 (es) | 2016-03-22 | 2018-06-28 | Merck Sharp & Dohme | Moduladores alostéricos de receptores de acetilcolina nicotínicos |
| US10870630B2 (en) | 2016-11-01 | 2020-12-22 | Merck Sharp & Dohme Corp. | Substituted bicyclic heteroaryl allosteric modulators of nicotinic acetylcholine receptors |
| WO2018112204A1 (en) * | 2016-12-14 | 2018-06-21 | Cephalon, Inc. | Spiropiperidine derivatives |
-
2018
- 2018-07-13 HU HUP1800248A patent/HU231333B1/hu unknown
-
2019
- 2019-06-27 TW TW108122548A patent/TWI821321B/zh active
- 2019-07-12 CA CA3104258A patent/CA3104258A1/en active Pending
- 2019-07-12 US US17/259,972 patent/US20210330650A1/en not_active Abandoned
- 2019-07-12 CU CU2020000108A patent/CU24680B1/es unknown
- 2019-07-12 AU AU2019300514A patent/AU2019300514B2/en not_active Ceased
- 2019-07-12 IL IL279938A patent/IL279938B2/en unknown
- 2019-07-12 WO PCT/IB2019/055948 patent/WO2020012422A1/en not_active Ceased
- 2019-07-12 PE PE2021000053A patent/PE20211809A1/es unknown
- 2019-07-12 KR KR1020217004264A patent/KR20210033002A/ko not_active Abandoned
- 2019-07-12 HU HUE19744868A patent/HUE064417T2/hu unknown
- 2019-07-12 GE GEAP202315557A patent/GEAP202315557A/en unknown
- 2019-07-12 JP JP2021500532A patent/JP7487167B2/ja active Active
- 2019-07-12 EA EA202190245A patent/EA202190245A1/ru unknown
- 2019-07-12 GE GEAP201915557A patent/GEP20237534B/en unknown
- 2019-07-12 BR BR112020026996-4A patent/BR112020026996A2/pt unknown
- 2019-07-12 EP EP19744868.1A patent/EP3820869B1/en active Active
- 2019-07-12 MY MYPI2020006684A patent/MY206779A/en unknown
- 2019-07-12 MX MX2021000460A patent/MX2021000460A/es unknown
- 2019-07-12 CN CN201980046665.7A patent/CN112823157B/zh active Active
- 2019-07-12 AR ARP190101991A patent/AR115782A1/es unknown
- 2019-07-12 SG SG11202012594RA patent/SG11202012594RA/en unknown
- 2019-07-12 ES ES19744868T patent/ES2964617T3/es active Active
-
2020
- 2020-12-16 PH PH12020552183A patent/PH12020552183A1/en unknown
-
2021
- 2021-01-12 CL CL2021000080A patent/CL2021000080A1/es unknown
- 2021-02-03 CO CONC2021/0001216A patent/CO2021001216A2/es unknown
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