JP2021529813A5 - - Google Patents
Info
- Publication number
- JP2021529813A5 JP2021529813A5 JP2021500540A JP2021500540A JP2021529813A5 JP 2021529813 A5 JP2021529813 A5 JP 2021529813A5 JP 2021500540 A JP2021500540 A JP 2021500540A JP 2021500540 A JP2021500540 A JP 2021500540A JP 2021529813 A5 JP2021529813 A5 JP 2021529813A5
- Authority
- JP
- Japan
- Prior art keywords
- disorders
- disorder
- formula
- thiadiazine
- dioxo
- Prior art date
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024020524A JP2024056879A (ja) | 2018-07-13 | 2024-02-14 | チアジアジン誘導体 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HUP1800249 | 2018-07-13 | ||
| HUP1800249A HU231414B1 (hu) | 2018-07-13 | 2018-07-13 | Tiadiazin származékok |
| PCT/IB2019/055949 WO2020012423A1 (en) | 2018-07-13 | 2019-07-12 | Thiadiazine derivatives |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024020524A Division JP2024056879A (ja) | 2018-07-13 | 2024-02-14 | チアジアジン誘導体 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2021529813A JP2021529813A (ja) | 2021-11-04 |
| JP2021529813A5 true JP2021529813A5 (https=) | 2022-07-20 |
| JPWO2020012423A5 JPWO2020012423A5 (https=) | 2022-07-20 |
| JP7440486B2 JP7440486B2 (ja) | 2024-02-28 |
Family
ID=89992726
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021500540A Active JP7440486B2 (ja) | 2018-07-13 | 2019-07-12 | チアジアジン誘導体 |
| JP2024020524A Withdrawn JP2024056879A (ja) | 2018-07-13 | 2024-02-14 | チアジアジン誘導体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024020524A Withdrawn JP2024056879A (ja) | 2018-07-13 | 2024-02-14 | チアジアジン誘導体 |
Country Status (23)
| Country | Link |
|---|---|
| US (2) | US12194050B2 (https=) |
| EP (1) | EP3820865A1 (https=) |
| JP (2) | JP7440486B2 (https=) |
| KR (1) | KR20210033003A (https=) |
| CN (1) | CN112424198A (https=) |
| AR (1) | AR115783A1 (https=) |
| AU (1) | AU2019300515B2 (https=) |
| BR (1) | BR112020027016A2 (https=) |
| CA (1) | CA3104264A1 (https=) |
| CL (1) | CL2021000081A1 (https=) |
| CO (1) | CO2021001224A2 (https=) |
| CU (1) | CU24622B1 (https=) |
| EA (1) | EA202190246A1 (https=) |
| GE (2) | GEAP202215558A (https=) |
| HU (1) | HU231414B1 (https=) |
| IL (1) | IL279939B2 (https=) |
| MX (1) | MX2021000461A (https=) |
| MY (1) | MY207757A (https=) |
| PE (1) | PE20210465A1 (https=) |
| PH (1) | PH12021550007A1 (https=) |
| SG (1) | SG11202012769QA (https=) |
| TW (1) | TWI827628B (https=) |
| WO (1) | WO2020012423A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4103191A4 (en) * | 2020-02-14 | 2024-03-06 | University of Pittsburgh - of the Commonwealth System of Higher Education | HEAT SHOCK PROTEIN MODULATORS AND THERAPEUTIC AGENTS FOR HUNTINGTON'S DISEASE |
| TWI901650B (zh) | 2020-03-26 | 2025-10-21 | 匈牙利商羅特格登公司 | 啶及吡啶并〔３，４－ｃ〕嗒衍生物 |
| CN111454232B (zh) * | 2020-05-30 | 2021-11-23 | 南方医科大学 | 一种1,3,4-噻二嗪类化合物及其应用 |
| HU231691B1 (hu) | 2021-09-29 | 2025-10-28 | Richter Gedeon Nyrt | GABAA ALFA5 receptor modulátor hatású biciklusos aminszármazékok |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006016548A1 (ja) | 2004-08-09 | 2006-02-16 | Eisai R & D Management Co., Ltd. | ヘテロ環化合物を含有する新規な抗マラリア剤 |
| NZ566036A (en) | 2005-09-13 | 2010-06-25 | Janssen Pharmaceutica Nv | 2-Aniline-4-aryl substituted thiazole derivatives that modulate the alpha7 nicotinic receptor |
| ES2274729B1 (es) | 2005-11-11 | 2008-06-01 | Consejo Superior Investig. Cientificas | Derivados de 5-carboxilato y 5-carboxamida 2-sustituidos de 1,1-dioxo-1,2,6-tiadiazina con propiedades cannabinoides. |
| US20100298314A1 (en) | 2006-12-20 | 2010-11-25 | Schering Corporation | Novel jnk inhibitors |
| MX2010003155A (es) | 2007-10-04 | 2010-04-01 | Hoffmann La Roche | Derivados de ciclopropil aril amida y uso de los mismos. |
| MX2010003156A (es) | 2007-10-04 | 2010-04-01 | Hoffmann La Roche | Derivados de aril amida substituida con tetrazol y usos de los mismos. |
| KR20100124272A (ko) | 2008-02-07 | 2010-11-26 | 아보트 러보러터리즈 | 양성 알로스테릭 조절제로서의 아미드 유도체 및 이의 사용방법 |
| AR070936A1 (es) | 2008-03-19 | 2010-05-12 | Janssen Pharmaceutica Nv | 1,2,4 -triazoles trisustituidos |
| EP2110377A1 (en) | 2008-04-15 | 2009-10-21 | DAC S.r.l. | Spirocyclic derivatives as histone deacetylase inhibitors |
| WO2009127678A1 (en) | 2008-04-17 | 2009-10-22 | Glaxo Group Limited | Indoles as modulators of nicotinic acetylcholin receptor subtype alpha-71 |
| JP5486591B2 (ja) | 2008-05-09 | 2014-05-07 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | アセチルコリン受容体モジュレーターとしての三置換ピラゾール |
| CA2725940A1 (en) | 2008-05-30 | 2009-12-23 | Merck Sharp & Dohme Corp. | Novel substituted azabenzoxazoles |
| EP2488520B1 (en) * | 2009-10-13 | 2015-09-02 | Merck Sharp & Dohme B.V. | Condensed azine-derivatives for the treatment of diseases related to the acetylcholine receptor |
| EP3795573B1 (en) | 2009-12-31 | 2022-07-06 | Hutchison Medipharma Limited | Certain triazolopyrazines, compositions thereof and methods of use therefor |
| WO2012042915A1 (en) | 2010-10-01 | 2012-04-05 | Raqualia Pharma Inc. | Sulfamoyl benzoic acid heterobicyclic derivatives as trpm8 antagonists |
| SG192078A1 (en) * | 2011-02-03 | 2013-08-30 | Lupin Ltd | Pyrrole derivatives used as modulators of alpha7 nachr |
| US9617210B2 (en) * | 2013-03-13 | 2017-04-11 | Lupin Limited | Pyrrole derivatives as alpha 7 NACHR modulators |
| AR107928A1 (es) * | 2016-03-22 | 2018-06-28 | Merck Sharp & Dohme | Moduladores alostéricos de receptores de acetilcolina nicotínicos |
| US10870630B2 (en) | 2016-11-01 | 2020-12-22 | Merck Sharp & Dohme Corp. | Substituted bicyclic heteroaryl allosteric modulators of nicotinic acetylcholine receptors |
| WO2018112204A1 (en) | 2016-12-14 | 2018-06-21 | Cephalon, Inc. | Spiropiperidine derivatives |
| SG11201908012SA (en) | 2017-03-02 | 2019-09-27 | Assembly Biosciences Inc | Cyclic sulfamide compounds and methods of using same |
| HU231333B1 (hu) | 2018-07-13 | 2023-01-28 | Richter Gedeon Nyrt | Spirokromán származékok |
-
2018
- 2018-07-13 HU HUP1800249A patent/HU231414B1/hu unknown
-
2019
- 2019-06-27 TW TW108122604A patent/TWI827628B/zh active
- 2019-07-12 US US17/259,975 patent/US12194050B2/en active Active
- 2019-07-12 CA CA3104264A patent/CA3104264A1/en active Pending
- 2019-07-12 WO PCT/IB2019/055949 patent/WO2020012423A1/en not_active Ceased
- 2019-07-12 CN CN201980046660.4A patent/CN112424198A/zh active Pending
- 2019-07-12 BR BR112020027016-4A patent/BR112020027016A2/pt unknown
- 2019-07-12 IL IL279939A patent/IL279939B2/en unknown
- 2019-07-12 SG SG11202012769QA patent/SG11202012769QA/en unknown
- 2019-07-12 AR ARP190101992A patent/AR115783A1/es unknown
- 2019-07-12 EP EP19744869.9A patent/EP3820865A1/en active Pending
- 2019-07-12 PE PE2021000052A patent/PE20210465A1/es unknown
- 2019-07-12 KR KR1020217004286A patent/KR20210033003A/ko not_active Ceased
- 2019-07-12 GE GEAP202215558A patent/GEAP202215558A/en unknown
- 2019-07-12 AU AU2019300515A patent/AU2019300515B2/en not_active Expired - Fee Related
- 2019-07-12 MX MX2021000461A patent/MX2021000461A/es unknown
- 2019-07-12 JP JP2021500540A patent/JP7440486B2/ja active Active
- 2019-07-12 CU CU2020000109A patent/CU24622B1/es unknown
- 2019-07-12 GE GEAP201915558A patent/GEP20237459B/en unknown
- 2019-07-12 EA EA202190246A patent/EA202190246A1/ru unknown
- 2019-07-12 MY MYPI2020006712A patent/MY207757A/en unknown
-
2021
- 2021-01-04 PH PH12021550007A patent/PH12021550007A1/en unknown
- 2021-01-12 CL CL2021000081A patent/CL2021000081A1/es unknown
- 2021-02-03 CO CONC2021/0001224A patent/CO2021001224A2/es unknown
-
2024
- 2024-02-14 JP JP2024020524A patent/JP2024056879A/ja not_active Withdrawn
- 2024-11-14 US US18/947,529 patent/US20250064823A1/en active Pending
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